IL199909A0 - Napadisylate salt of a muscarinic m3 antagonist - Google Patents

Napadisylate salt of a muscarinic m3 antagonist

Info

Publication number
IL199909A0
IL199909A0 IL199909A IL19990909A IL199909A0 IL 199909 A0 IL199909 A0 IL 199909A0 IL 199909 A IL199909 A IL 199909A IL 19990909 A IL19990909 A IL 19990909A IL 199909 A0 IL199909 A0 IL 199909A0
Authority
IL
Israel
Prior art keywords
muscarinic
antagonist
napadisylate salt
napadisylate
salt
Prior art date
Application number
IL199909A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Argenta Discovery Ltd
Avitabile Barbara Giuseppina
Sullivan David O
Bull Richard James
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB0702416.9A external-priority patent/GB0702416D0/en
Priority claimed from GBGB0702385.6A external-priority patent/GB0702385D0/en
Application filed by Astrazeneca Ab, Argenta Discovery Ltd, Avitabile Barbara Giuseppina, Sullivan David O, Bull Richard James filed Critical Astrazeneca Ab
Publication of IL199909A0 publication Critical patent/IL199909A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/10—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D263/12—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with radicals containing only hydrogen and carbon atoms
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
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  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
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IL199909A 2007-02-07 2009-07-16 Napadisylate salt of a muscarinic m3 antagonist IL199909A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0702416.9A GB0702416D0 (en) 2007-02-07 2007-02-07 New combination
GBGB0702385.6A GB0702385D0 (en) 2007-02-07 2007-02-07 New combination
PCT/GB2008/000434 WO2008096149A2 (en) 2007-02-07 2008-02-06 Napadisylate salt of a muscarinic m3 antagonist

Publications (1)

Publication Number Publication Date
IL199909A0 true IL199909A0 (en) 2010-04-15

Family

ID=39485211

Family Applications (1)

Application Number Title Priority Date Filing Date
IL199909A IL199909A0 (en) 2007-02-07 2009-07-16 Napadisylate salt of a muscarinic m3 antagonist

Country Status (13)

Country Link
US (1) US7846955B2 (OSRAM)
EP (1) EP2118078A2 (OSRAM)
JP (1) JP5373634B2 (OSRAM)
KR (1) KR20090119757A (OSRAM)
AU (1) AU2008212673B2 (OSRAM)
BR (1) BRPI0807004A2 (OSRAM)
CA (1) CA2675629A1 (OSRAM)
EC (1) ECSP099566A (OSRAM)
IL (1) IL199909A0 (OSRAM)
MX (1) MX2009008364A (OSRAM)
NZ (1) NZ578475A (OSRAM)
RU (1) RU2459810C2 (OSRAM)
WO (1) WO2008096149A2 (OSRAM)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0516313D0 (en) * 2005-08-08 2005-09-14 Argenta Discovery Ltd Azole derivatives and their uses
TW200825084A (en) 2006-11-14 2008-06-16 Astrazeneca Ab New compounds 521
NZ589091A (en) 2008-05-13 2011-07-29 Astrazeneca Ab Quinuclidine derivatives as muscarinic m3 receptor antagonists
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
ES2725784T3 (es) 2011-07-20 2019-09-27 Univ Brigham Young Compuestos de ceragenina hidrófobos y dispositivos que incorporan al mismo
US11524015B2 (en) 2013-03-15 2022-12-13 Brigham Young University Methods for treating inflammation, autoimmune disorders and pain
CN110420211A (zh) 2013-03-15 2019-11-08 布莱阿姆青年大学 治疗炎症、自身免疫性疾病和疼痛的方法
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US20150203527A1 (en) 2014-01-23 2015-07-23 Brigham Young University Cationic steroidal antimicrobials
CA2991726C (en) * 2015-04-22 2022-07-19 Brigham Young University Cationic steroidal antimicrobial salts
US10226550B2 (en) 2016-03-11 2019-03-12 Brigham Young University Cationic steroidal antimicrobial compositions for the treatment of dermal tissue
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JP7152122B2 (ja) * 2017-10-13 2022-10-12 ツリーウェイ ティーダブリュー００１ ビー．ブイ． エダラボン塩
US12186328B2 (en) 2019-05-23 2025-01-07 Brigham Young University Use of CSA compounds to stimulate stem cells and hair growth
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MX2009008364A (es) 2009-08-20
AU2008212673B2 (en) 2011-04-28
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US20100093816A1 (en) 2010-04-15
US7846955B2 (en) 2010-12-07
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BRPI0807004A2 (pt) 2014-04-15
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AU2008212673A1 (en) 2008-08-14
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