NZ525720A - The use of triptorelin and exemestane in the manner of a medicament for treating a sex steroid dependent cancer - Google Patents
The use of triptorelin and exemestane in the manner of a medicament for treating a sex steroid dependent cancerInfo
- Publication number
- NZ525720A NZ525720A NZ525720A NZ52572001A NZ525720A NZ 525720 A NZ525720 A NZ 525720A NZ 525720 A NZ525720 A NZ 525720A NZ 52572001 A NZ52572001 A NZ 52572001A NZ 525720 A NZ525720 A NZ 525720A
- Authority
- NZ
- New Zealand
- Prior art keywords
- use according
- cancer
- medicament
- exemestane
- triptorelin
- Prior art date
Links
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- RWHUEXWOYVBUCI-ITQXDASVSA-N nafarelin Chemical compound C([C@@H](C(=O)N[C@H](CC=1C=C2C=CC=CC2=CC=1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1[C@@H](CCC1)C(=O)NCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CC=1C2=CC=CC=C2NC=1)NC(=O)[C@H](CC=1NC=NC=1)NC(=O)[C@H]1NC(=O)CC1)C1=CC=C(O)C=C1 RWHUEXWOYVBUCI-ITQXDASVSA-N 0.000 description 1
- 230000024717 negative regulation of secretion Effects 0.000 description 1
- 210000003635 pituitary gland Anatomy 0.000 description 1
- 239000000843 powder Substances 0.000 description 1
- 239000000583 progesterone congener Substances 0.000 description 1
- 229940097325 prolactin Drugs 0.000 description 1
- 108010092834 ramorelix Proteins 0.000 description 1
- 229950000277 ramorelix Drugs 0.000 description 1
- 108020003175 receptors Proteins 0.000 description 1
- 230000002829 reductive effect Effects 0.000 description 1
- 230000002441 reversible effect Effects 0.000 description 1
- 230000028327 secretion Effects 0.000 description 1
- 210000002966 serum Anatomy 0.000 description 1
- 239000000243 solution Substances 0.000 description 1
- 150000003431 steroids Chemical class 0.000 description 1
- 239000000725 suspension Substances 0.000 description 1
- 238000013268 sustained release Methods 0.000 description 1
- 239000012730 sustained-release form Substances 0.000 description 1
- 208000024891 symptom Diseases 0.000 description 1
- 239000006188 syrup Substances 0.000 description 1
- 235000020357 syrup Nutrition 0.000 description 1
- 239000003826 tablet Substances 0.000 description 1
- 229950011372 teverelix Drugs 0.000 description 1
- 229940124597 therapeutic agent Drugs 0.000 description 1
- 231100000331 toxic Toxicity 0.000 description 1
- 230000002588 toxic effect Effects 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Reproductive Health (AREA)
- Oncology (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US71460500A | 2000-11-16 | 2000-11-16 | |
| PCT/US2001/043847 WO2002039995A2 (en) | 2000-11-16 | 2001-11-06 | Combination therapy for estrogen-dependent disorders |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ525720A true NZ525720A (en) | 2006-12-22 |
Family
ID=24870727
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ525720A NZ525720A (en) | 2000-11-16 | 2001-11-06 | The use of triptorelin and exemestane in the manner of a medicament for treating a sex steroid dependent cancer |
Country Status (16)
| Country | Link |
|---|---|
| EP (1) | EP1341549A2 (cs) |
| JP (1) | JP2004536022A (cs) |
| KR (1) | KR20030051828A (cs) |
| CN (1) | CN1498112A (cs) |
| AU (1) | AU2002230464A1 (cs) |
| BR (1) | BR0115423A (cs) |
| CA (1) | CA2428249A1 (cs) |
| CZ (1) | CZ20031349A3 (cs) |
| EA (1) | EA200300572A1 (cs) |
| IL (1) | IL155817A0 (cs) |
| MX (1) | MXPA03004195A (cs) |
| NO (1) | NO20032206L (cs) |
| NZ (1) | NZ525720A (cs) |
| PL (1) | PL365904A1 (cs) |
| WO (1) | WO2002039995A2 (cs) |
| ZA (1) | ZA200303669B (cs) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL153218A0 (en) | 2000-06-02 | 2003-07-06 | Univ Texas | Ethylenedicysteine (ec) -drug conjugates |
| US9050378B2 (en) | 2003-12-10 | 2015-06-09 | Board Of Regents, The University Of Texas System | N2S2 chelate-targeting ligand conjugates |
| GB0506759D0 (en) * | 2005-04-02 | 2005-05-11 | Medical Res Council | Combination treatment methods |
| EP1891964A1 (en) * | 2006-08-08 | 2008-02-27 | AEterna Zentaris GmbH | Application of initial doses of LHRH analogues and maintenance doses of LHRH antagonists for the treatment of hormone-dependent cancers and corresponding pharmaceutical kits |
| US10925977B2 (en) | 2006-10-05 | 2021-02-23 | Ceil>Point, LLC | Efficient synthesis of chelators for nuclear imaging and radiotherapy: compositions and applications |
| US20080261933A1 (en) * | 2007-04-23 | 2008-10-23 | Jens Hoffmann | Combination of progesterone-receptor antagonist together with a lutein-hormone-releasing hormone agonist and antagonist for use in brca mediated diseases |
| CN101775054B (zh) * | 2010-02-05 | 2012-12-26 | 常州佳尔科药业集团有限公司 | 4-羟基-4-烯-3-酮甾族化合物的合成方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9911582D0 (en) * | 1999-05-18 | 1999-07-21 | Pharmacia & Upjohn Spa | Combined method of treatment comprising an aromatase inhibitor and a further biologically active compound |
| GB9930839D0 (en) * | 1999-12-30 | 2000-02-16 | Pharmacia & Upjohn Spa | Process for treating gynecomastia |
-
2001
- 2001-11-06 KR KR10-2003-7006608A patent/KR20030051828A/ko not_active Withdrawn
- 2001-11-06 EA EA200300572A patent/EA200300572A1/ru unknown
- 2001-11-06 CZ CZ20031349A patent/CZ20031349A3/cs unknown
- 2001-11-06 AU AU2002230464A patent/AU2002230464A1/en not_active Abandoned
- 2001-11-06 BR BR0115423-0A patent/BR0115423A/pt not_active IP Right Cessation
- 2001-11-06 NZ NZ525720A patent/NZ525720A/en unknown
- 2001-11-06 PL PL01365904A patent/PL365904A1/xx not_active Application Discontinuation
- 2001-11-06 MX MXPA03004195A patent/MXPA03004195A/es unknown
- 2001-11-06 IL IL15581701A patent/IL155817A0/xx unknown
- 2001-11-06 EP EP01990699A patent/EP1341549A2/en not_active Withdrawn
- 2001-11-06 CN CNA018189385A patent/CN1498112A/zh active Pending
- 2001-11-06 JP JP2002542370A patent/JP2004536022A/ja active Pending
- 2001-11-06 WO PCT/US2001/043847 patent/WO2002039995A2/en not_active Ceased
- 2001-11-06 CA CA002428249A patent/CA2428249A1/en not_active Abandoned
-
2003
- 2003-05-13 ZA ZA200303669A patent/ZA200303669B/en unknown
- 2003-05-15 NO NO20032206A patent/NO20032206L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CZ20031349A3 (cs) | 2004-05-12 |
| KR20030051828A (ko) | 2003-06-25 |
| NO20032206L (no) | 2003-07-15 |
| JP2004536022A (ja) | 2004-12-02 |
| NO20032206D0 (no) | 2003-05-15 |
| BR0115423A (pt) | 2005-12-13 |
| CN1498112A (zh) | 2004-05-19 |
| EP1341549A2 (en) | 2003-09-10 |
| AU2002230464A1 (en) | 2002-05-27 |
| CA2428249A1 (en) | 2002-05-23 |
| EA200300572A1 (ru) | 2004-06-24 |
| PL365904A1 (en) | 2005-01-10 |
| IL155817A0 (en) | 2003-12-23 |
| MXPA03004195A (es) | 2003-09-22 |
| WO2002039995A9 (en) | 2003-02-06 |
| WO2002039995A2 (en) | 2002-05-23 |
| ZA200303669B (en) | 2004-05-13 |
| WO2002039995A3 (en) | 2003-05-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RENW | Renewal (renewal fees accepted) | ||
| PSEA | Patent sealed |