NZ247032A - Phenyl-substituted quinazoline and thiazolo[2,3-b]quinazoline derivatives; pharmaceutical compositions and preparatory processes thereof - Google Patents

Phenyl-substituted quinazoline and thiazolo[2,3-b]quinazoline derivatives; pharmaceutical compositions and preparatory processes thereof

Info

Publication number
NZ247032A
NZ247032A NZ247032A NZ24703293A NZ247032A NZ 247032 A NZ247032 A NZ 247032A NZ 247032 A NZ247032 A NZ 247032A NZ 24703293 A NZ24703293 A NZ 24703293A NZ 247032 A NZ247032 A NZ 247032A
Authority
NZ
New Zealand
Prior art keywords
hydrogen
compound
formula
carbon atoms
chloro
Prior art date
Application number
NZ247032A
Other languages
English (en)
Inventor
Paul Leroy Anderson
William Joseph Houlihan
Prasad Koteswara Kapa
Andrew Kucerovy
Paul Gerard Mattner
Original Assignee
Sandoz Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ltd filed Critical Sandoz Ltd
Publication of NZ247032A publication Critical patent/NZ247032A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/91Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/582Recycling of unreacted starting or intermediate materials

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
NZ247032A 1992-03-03 1993-03-01 Phenyl-substituted quinazoline and thiazolo[2,3-b]quinazoline derivatives; pharmaceutical compositions and preparatory processes thereof NZ247032A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US84512392A 1992-03-03 1992-03-03

Publications (1)

Publication Number Publication Date
NZ247032A true NZ247032A (en) 1994-11-25

Family

ID=25294463

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ247032A NZ247032A (en) 1992-03-03 1993-03-01 Phenyl-substituted quinazoline and thiazolo[2,3-b]quinazoline derivatives; pharmaceutical compositions and preparatory processes thereof

Country Status (14)

Country Link
EP (1) EP0564397A1 (enrdf_load_stackoverflow)
JP (1) JPH0649076A (enrdf_load_stackoverflow)
KR (1) KR930019642A (enrdf_load_stackoverflow)
CN (1) CN1076445A (enrdf_load_stackoverflow)
AU (1) AU3387593A (enrdf_load_stackoverflow)
CA (1) CA2090635A1 (enrdf_load_stackoverflow)
CZ (1) CZ30293A3 (enrdf_load_stackoverflow)
FI (1) FI930922A7 (enrdf_load_stackoverflow)
HU (1) HUT63629A (enrdf_load_stackoverflow)
IL (1) IL104892A0 (enrdf_load_stackoverflow)
NO (1) NO930739L (enrdf_load_stackoverflow)
NZ (1) NZ247032A (enrdf_load_stackoverflow)
TW (1) TW227563B (enrdf_load_stackoverflow)
ZA (1) ZA931516B (enrdf_load_stackoverflow)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1655289A1 (en) * 2004-11-04 2006-05-10 Embl Quinazoline derivatives, process for their preparation, their use as antimitotics and pharmaceutical compositions comprising said derivatives
WO2012168359A1 (en) * 2011-06-10 2012-12-13 Chiesi Farmaceutici S.P.A. Compounds having muscarinic receptor antagonist and beta2 adrenergic receptor agonist activity
CN104119231A (zh) * 2013-04-27 2014-10-29 重庆华邦制药有限公司 二苯甲胺类化合物的制备方法及中间体
WO2015120059A1 (en) * 2014-02-04 2015-08-13 Yates Charles Ryan Inhibitors of paxillin function and related compositions and methods

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1242863A (en) * 1968-05-10 1971-08-18 Pharmacia As 2,3-DIHYDRO-5H-THIAZOLO[2,3-b]QUINAZOLINES AND PROCESSES FOR THE PREPARATION THEREOF
DE3734909A1 (de) * 1987-10-15 1989-04-27 Boehringer Ingelheim Kg Verwendung von oxochinazolinderivaten bei der behandlung der hyperlipidaemie

Also Published As

Publication number Publication date
HUT63629A (en) 1993-09-28
CN1076445A (zh) 1993-09-22
KR930019642A (ko) 1993-10-18
IL104892A0 (en) 1993-07-08
CZ30293A3 (en) 1993-12-15
AU3387593A (en) 1993-09-09
FI930922A7 (fi) 1993-09-04
CA2090635A1 (en) 1993-09-04
JPH0649076A (ja) 1994-02-22
ZA931516B (en) 1994-09-03
FI930922A0 (fi) 1993-03-02
HU9300556D0 (en) 1993-05-28
NO930739L (no) 1993-09-06
TW227563B (enrdf_load_stackoverflow) 1994-08-01
NO930739D0 (no) 1993-03-01
EP0564397A1 (en) 1993-10-06

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