NZ246558A - 5-amino (and azaheterocyclyl)-3-oxazolyl imidazoquinazoline derivatives, preparation and pharmaceutical compositions - Google Patents
5-amino (and azaheterocyclyl)-3-oxazolyl imidazoquinazoline derivatives, preparation and pharmaceutical compositionsInfo
- Publication number
- NZ246558A NZ246558A NZ246558A NZ24655892A NZ246558A NZ 246558 A NZ246558 A NZ 246558A NZ 246558 A NZ246558 A NZ 246558A NZ 24655892 A NZ24655892 A NZ 24655892A NZ 246558 A NZ246558 A NZ 246558A
- Authority
- NZ
- New Zealand
- Prior art keywords
- quinazoline
- compound
- cyclopropyl
- imidazo
- oxadiazol
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK912042A DK204291D0 (da) | 1991-12-20 | 1991-12-20 | Heterocykliske forbindelser deres fremstilling og anvendelse |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ246558A true NZ246558A (en) | 1995-07-26 |
Family
ID=8109668
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ246558A NZ246558A (en) | 1991-12-20 | 1992-12-18 | 5-amino (and azaheterocyclyl)-3-oxazolyl imidazoquinazoline derivatives, preparation and pharmaceutical compositions |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP0619820A1 (enExample) |
| JP (1) | JPH07502278A (enExample) |
| AU (1) | AU673814B2 (enExample) |
| CA (1) | CA2125854A1 (enExample) |
| DK (1) | DK204291D0 (enExample) |
| FI (1) | FI942963L (enExample) |
| IL (1) | IL104099A (enExample) |
| NO (1) | NO942301L (enExample) |
| NZ (1) | NZ246558A (enExample) |
| TW (1) | TW211568B (enExample) |
| WO (1) | WO1993013103A1 (enExample) |
| ZA (1) | ZA929770B (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK151890D0 (da) * | 1990-06-22 | 1990-06-22 | Ferrosan As | Heterocykliske forbindelser deres fremstilling og brug |
| CN1052724C (zh) * | 1996-07-01 | 2000-05-24 | 瑞安大药厂股份有限公司 | 新的光学活性的2,3－二氢咪唑并[1,2－c]喹唑啉衍生物及其制备方法和用途 |
| KR100864364B1 (ko) | 2005-12-13 | 2008-10-17 | 주식회사 엘지화학 | 신규한 이미다조퀴나졸린 유도체, 이의 제조방법 및 이를이용한 유기전기소자 |
| CA2678577A1 (en) | 2007-02-26 | 2008-09-04 | Vitae Pharmaceuticals, Inc. | Cyclic urea and carbamate inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1 |
| AR069207A1 (es) | 2007-11-07 | 2010-01-06 | Vitae Pharmaceuticals Inc | Ureas ciclicas como inhibidores de la 11 beta - hidroxi-esteroide deshidrogenasa 1 |
| JP5490014B2 (ja) | 2007-12-11 | 2014-05-14 | ヴァイティー ファーマシューティカルズ，インコーポレイテッド | １１β−ヒドロキシステロイドデヒドロゲナーゼ１型の環状尿素阻害剤 |
| US8846668B2 (en) | 2008-07-25 | 2014-09-30 | Vitae Pharmaceuticals, Inc. | Inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
| KR20110050459A (ko) | 2008-07-25 | 2011-05-13 | 비타이 파마슈티컬즈, 인코포레이티드 | 11베타-하이드록시스테로이드 탈수소효소 1의 고리형 억제제 |
| WO2010089303A1 (en) | 2009-02-04 | 2010-08-12 | Boehringer Ingelheim International Gmbh | CYCLIC INHIBITORS OF 11 β-HYDROXYSTEROID DEHYDROGENASE 1 |
| MA33216B1 (fr) | 2009-04-30 | 2012-04-02 | Boehringer Ingelheim Int | Inhibiteurs cycliques de la 11béta-hydroxysteroïde déshydrogénase 1 |
| JP5656986B2 (ja) | 2009-06-11 | 2015-01-21 | ヴァイティー ファーマシューティカルズ，インコーポレイテッド | １，３−オキサジナン−２−オン構造に基づく１１β−ヒドロキシステロイドデヒドロゲナーゼ１の環状阻害剤 |
| US8883778B2 (en) | 2009-07-01 | 2014-11-11 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11 beta-hydroxysteroid dehydrogenase 1 |
| US8933072B2 (en) | 2010-06-16 | 2015-01-13 | Vitae Pharmaceuticals, Inc. | Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use |
| EP2585444B1 (en) | 2010-06-25 | 2014-10-22 | Boehringer Ingelheim International GmbH | Azaspirohexanones as inhibitors of 11-beta-hsd1 for the treatment of metabolic disorders |
| CA2813671A1 (en) | 2010-11-02 | 2012-05-10 | Boehringer Ingelheim International Gmbh | Pharmaceutical combinations for the treatment of metabolic disorders |
| CA3195592A1 (en) * | 2020-10-16 | 2022-04-21 | Xiaohui Liu | Triheterocyclic derivative, and pharmaceutical composition and application thereof |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE44381T1 (de) * | 1985-10-17 | 1989-07-15 | Ferrosan As | Heterocyclische verbindungen und ihre herstellung und verwendung. |
| DK155524C (da) * | 1987-03-18 | 1989-09-11 | Ferrosan As | Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse |
| DK443589D0 (da) * | 1989-09-08 | 1989-09-08 | Ferrosan As | Heterocykliske forbindelser, deres fremstilling og anvendelse |
| DK151890D0 (da) * | 1990-06-22 | 1990-06-22 | Ferrosan As | Heterocykliske forbindelser deres fremstilling og brug |
-
1991
- 1991-12-20 DK DK912042A patent/DK204291D0/da not_active Application Discontinuation
-
1992
- 1992-12-15 IL IL10409992A patent/IL104099A/en not_active IP Right Cessation
- 1992-12-17 ZA ZA929770A patent/ZA929770B/xx unknown
- 1992-12-18 FI FI942963A patent/FI942963L/fi not_active Application Discontinuation
- 1992-12-18 JP JP5511363A patent/JPH07502278A/ja active Pending
- 1992-12-18 WO PCT/DK1992/000385 patent/WO1993013103A1/en not_active Ceased
- 1992-12-18 CA CA002125854A patent/CA2125854A1/en not_active Abandoned
- 1992-12-18 NZ NZ246558A patent/NZ246558A/en unknown
- 1992-12-18 TW TW081110173A patent/TW211568B/zh active
- 1992-12-18 AU AU33448/93A patent/AU673814B2/en not_active Ceased
- 1992-12-18 EP EP93902092A patent/EP0619820A1/en not_active Withdrawn
-
1994
- 1994-06-17 NO NO942301A patent/NO942301L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO942301D0 (no) | 1994-06-17 |
| FI942963A7 (fi) | 1994-06-20 |
| EP0619820A1 (en) | 1994-10-19 |
| NO942301L (no) | 1994-08-19 |
| TW211568B (enExample) | 1993-08-21 |
| FI942963A0 (fi) | 1994-06-20 |
| AU3344893A (en) | 1993-07-28 |
| DK204291D0 (da) | 1991-12-20 |
| ZA929770B (en) | 1994-06-17 |
| FI942963L (fi) | 1994-06-20 |
| IL104099A0 (en) | 1993-05-13 |
| AU673814B2 (en) | 1996-11-28 |
| JPH07502278A (ja) | 1995-03-09 |
| CA2125854A1 (en) | 1993-07-08 |
| IL104099A (en) | 1996-07-23 |
| WO1993013103A1 (en) | 1993-07-08 |
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