NZ193471A - Method for preparation of h-sar-lys-sar-gln-nh2;dipeptide and protected tetrapeptide intermediates - Google Patents

Method for preparation of h-sar-lys-sar-gln-nh2;dipeptide and protected tetrapeptide intermediates

Info

Publication number
NZ193471A
NZ193471A NZ193471A NZ19347180A NZ193471A NZ 193471 A NZ193471 A NZ 193471A NZ 193471 A NZ193471 A NZ 193471A NZ 19347180 A NZ19347180 A NZ 19347180A NZ 193471 A NZ193471 A NZ 193471A
Authority
NZ
New Zealand
Prior art keywords
sar
gln
cbz
lys
loweralkyl
Prior art date
Application number
NZ193471A
Other languages
English (en)
Inventor
G Heavner
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/095,744 external-priority patent/US4250086A/en
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of NZ193471A publication Critical patent/NZ193471A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
    • C07K5/1008—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NZ193471A 1979-04-26 1980-04-17 Method for preparation of h-sar-lys-sar-gln-nh2;dipeptide and protected tetrapeptide intermediates NZ193471A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3364179A 1979-04-26 1979-04-26
US06/095,744 US4250086A (en) 1979-11-19 1979-11-19 Method and composition for preparation of H-SAR-LYS-SAR-GLN-NH2

Publications (1)

Publication Number Publication Date
NZ193471A true NZ193471A (en) 1984-07-06

Family

ID=26709949

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ193471A NZ193471A (en) 1979-04-26 1980-04-17 Method for preparation of h-sar-lys-sar-gln-nh2;dipeptide and protected tetrapeptide intermediates

Country Status (16)

Country Link
EP (1) EP0018793B1 (https=)
JP (3) JPH01193297A (https=)
AU (1) AU536981B2 (https=)
CA (1) CA1156220A (https=)
DE (1) DE3065502D1 (https=)
DK (1) DK149631C (https=)
ES (1) ES8105269A1 (https=)
FI (1) FI801344A7 (https=)
GR (1) GR67297B (https=)
IE (1) IE49765B1 (https=)
IL (1) IL59918A (https=)
NO (1) NO152050C (https=)
NZ (1) NZ193471A (https=)
PH (2) PH17633A (https=)
PT (1) PT71146B (https=)
YU (1) YU42666B (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4298523A (en) * 1980-06-17 1981-11-03 Ortho Pharmaceutical Corporation Methods and compositions for preparation of H-ARG-X-Z-Y-TYR-R
CN103351324A (zh) * 2013-07-01 2013-10-16 太仓市恒益医药化工原料厂 一种用于9-芴甲氧羰酰琥珀酰亚胺制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2932635A (en) * 1957-02-22 1960-04-12 Roussel Uclaf Alpha-peptides of lysine and method of preparing same
FR2391994A1 (fr) * 1977-05-25 1978-12-22 Anvar Nouveaux polypeptides a activite thymique ou a activite antagoniste et leurs procedes de synthese
NZ189101A (en) * 1977-12-08 1984-07-06 Ortho Pharma Corp Polypeptides having the ability to induce differentiation of both th-1+ t-lymphocytes and bu-1+ b-lymphocytes;pharmaceutical compositions

Also Published As

Publication number Publication date
YU42666B (en) 1988-10-31
AU5775980A (en) 1980-10-30
JPH01193297A (ja) 1989-08-03
DK149631B (da) 1986-08-18
NO801215L (no) 1980-10-27
EP0018793A2 (en) 1980-11-12
PH17633A (en) 1984-10-12
IL59918A0 (en) 1980-06-30
GR67297B (https=) 1981-06-29
ES490945A0 (es) 1981-05-16
DK149631C (da) 1987-01-26
PH16655A (en) 1983-12-09
DE3065502D1 (en) 1983-12-15
YU114780A (en) 1984-02-29
IE49765B1 (en) 1985-12-11
ES8105269A1 (es) 1981-05-16
IE800838L (en) 1980-10-26
CA1156220A (en) 1983-11-01
JPH01193296A (ja) 1989-08-03
FI801344A7 (fi) 1980-10-27
NO152050B (no) 1985-04-15
PT71146B (en) 1981-08-07
IL59918A (en) 1983-05-15
NO152050C (no) 1985-07-24
DK180480A (da) 1980-10-27
EP0018793A3 (en) 1981-01-07
JPH01193298A (ja) 1989-08-03
EP0018793B1 (en) 1983-11-09
PT71146A (en) 1980-05-01
AU536981B2 (en) 1984-05-31

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