NZ193471A - Method for preparation of h-sar-lys-sar-gln-nh2;dipeptide and protected tetrapeptide intermediates - Google Patents

Method for preparation of h-sar-lys-sar-gln-nh2;dipeptide and protected tetrapeptide intermediates

Info

Publication number
NZ193471A
NZ193471A NZ193471A NZ19347180A NZ193471A NZ 193471 A NZ193471 A NZ 193471A NZ 193471 A NZ193471 A NZ 193471A NZ 19347180 A NZ19347180 A NZ 19347180A NZ 193471 A NZ193471 A NZ 193471A
Authority
NZ
New Zealand
Prior art keywords
sar
gln
cbz
lys
loweralkyl
Prior art date
Application number
NZ193471A
Other languages
English (en)
Inventor
G Heavner
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/095,744 external-priority patent/US4250086A/en
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of NZ193471A publication Critical patent/NZ193471A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
    • C07K5/1008—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NZ193471A 1979-04-26 1980-04-17 Method for preparation of h-sar-lys-sar-gln-nh2;dipeptide and protected tetrapeptide intermediates NZ193471A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3364179A 1979-04-26 1979-04-26
US06/095,744 US4250086A (en) 1979-11-19 1979-11-19 Method and composition for preparation of H-SAR-LYS-SAR-GLN-NH2

Publications (1)

Publication Number Publication Date
NZ193471A true NZ193471A (en) 1984-07-06

Family

ID=26709949

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ193471A NZ193471A (en) 1979-04-26 1980-04-17 Method for preparation of h-sar-lys-sar-gln-nh2;dipeptide and protected tetrapeptide intermediates

Country Status (16)

Country Link
EP (1) EP0018793B1 (enExample)
JP (3) JPH01193298A (enExample)
AU (1) AU536981B2 (enExample)
CA (1) CA1156220A (enExample)
DE (1) DE3065502D1 (enExample)
DK (1) DK149631C (enExample)
ES (1) ES8105269A1 (enExample)
FI (1) FI801344A7 (enExample)
GR (1) GR67297B (enExample)
IE (1) IE49765B1 (enExample)
IL (1) IL59918A (enExample)
NO (1) NO152050C (enExample)
NZ (1) NZ193471A (enExample)
PH (2) PH17633A (enExample)
PT (1) PT71146B (enExample)
YU (1) YU42666B (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4298523A (en) * 1980-06-17 1981-11-03 Ortho Pharmaceutical Corporation Methods and compositions for preparation of H-ARG-X-Z-Y-TYR-R
CN103351324A (zh) * 2013-07-01 2013-10-16 太仓市恒益医药化工原料厂 一种用于9-芴甲氧羰酰琥珀酰亚胺制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2932635A (en) * 1957-02-22 1960-04-12 Roussel Uclaf Alpha-peptides of lysine and method of preparing same
FR2391994A1 (fr) * 1977-05-25 1978-12-22 Anvar Nouveaux polypeptides a activite thymique ou a activite antagoniste et leurs procedes de synthese
NZ189101A (en) * 1977-12-08 1984-07-06 Ortho Pharma Corp Polypeptides having the ability to induce differentiation of both th-1+ t-lymphocytes and bu-1+ b-lymphocytes;pharmaceutical compositions

Also Published As

Publication number Publication date
DK149631C (da) 1987-01-26
IL59918A (en) 1983-05-15
EP0018793A3 (en) 1981-01-07
NO152050C (no) 1985-07-24
PH17633A (en) 1984-10-12
IL59918A0 (en) 1980-06-30
GR67297B (enExample) 1981-06-29
JPH01193296A (ja) 1989-08-03
NO801215L (no) 1980-10-27
FI801344A7 (fi) 1980-10-27
AU536981B2 (en) 1984-05-31
CA1156220A (en) 1983-11-01
EP0018793B1 (en) 1983-11-09
PT71146A (en) 1980-05-01
ES490945A0 (es) 1981-05-16
ES8105269A1 (es) 1981-05-16
JPH01193298A (ja) 1989-08-03
IE800838L (en) 1980-10-26
NO152050B (no) 1985-04-15
YU42666B (en) 1988-10-31
PH16655A (en) 1983-12-09
EP0018793A2 (en) 1980-11-12
DK180480A (da) 1980-10-27
JPH01193297A (ja) 1989-08-03
DK149631B (da) 1986-08-18
IE49765B1 (en) 1985-12-11
AU5775980A (en) 1980-10-30
PT71146B (en) 1981-08-07
DE3065502D1 (en) 1983-12-15
YU114780A (en) 1984-02-29

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