NO995549L - Anvendelse av 5-(4-(2-(M-metyl-N-(2-pyridyl)amino)-etoksy)bensyl)2,4-tiazolidindion ved behandling av polycystisk ovairiesyndrom og gestationell diabetes - Google Patents

Anvendelse av 5-(4-(2-(M-metyl-N-(2-pyridyl)amino)-etoksy)bensyl)2,4-tiazolidindion ved behandling av polycystisk ovairiesyndrom og gestationell diabetes

Info

Publication number
NO995549L
NO995549L NO995549A NO995549A NO995549L NO 995549 L NO995549 L NO 995549L NO 995549 A NO995549 A NO 995549A NO 995549 A NO995549 A NO 995549A NO 995549 L NO995549 L NO 995549L
Authority
NO
Norway
Prior art keywords
thiazolidinedione
pyridyl
ethoxy
benzyl
amino
Prior art date
Application number
NO995549A
Other languages
English (en)
Other versions
NO995549D0 (no
Inventor
Tammy Antonucci
Dean Lockwood
Rebecca Norris
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of NO995549L publication Critical patent/NO995549L/no
Publication of NO995549D0 publication Critical patent/NO995549D0/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Nye metoder for anvendelse av tiazolidinonderivater og beslektede antihy- perglykemiske midler for å behandle populasjoner med risiko for utvikling av ikke- insulinavhengig diabetes mellitus (NIDDM) og komplikasjoner som stammer der- fra, er beskrevet, l en utførelsesform blir forbindelsene ifølge foreliggende oppfin- nelse anvendt for å behandle polycystisk ovariesyndrom for å forhindre eller ut- sette opptreden av ikke-insulinavhengig diabetes mellitus. Ved en annen utførel- sesform blir forbindelsene ifølge foreliggende oppfinnelse anvendt for å behandle svangerskapsdiabetes for å forhindre eller utsette opptreden av ikke-insulin- avhengig diabetes mellitus.
NO995549A 1997-05-15 1999-11-12 Anvendelse av 5-(4-(2-(M-metyl-N-(2-pyridyl)amino)-etoksy)bensyl)2,4-tiazolidindion ved behandling av polycystisk ovairiesyndrom og gestationell diabetes NO995549D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/856,987 US5874454A (en) 1993-09-15 1997-05-15 Use of thiazolidinedione derivatives in the treatment of polycystic ovary syndrome, gestational diabetes and disease states at risk for progressing to noninsulin-dependent diabetes mellitus
PCT/US1998/010113 WO1998051305A1 (en) 1997-05-15 1998-05-14 Use of 5-(4-(2-(n-methyl-n-(2-pyridyl)amino)-ethoxy)benzyl)2,4-thiazolidinedione in the treatment of polycystic ovary syndrome and gestational diabetes

Publications (2)

Publication Number Publication Date
NO995549L true NO995549L (no) 1999-11-12
NO995549D0 NO995549D0 (no) 1999-11-12

Family

ID=25324901

Family Applications (1)

Application Number Title Priority Date Filing Date
NO995549A NO995549D0 (no) 1997-05-15 1999-11-12 Anvendelse av 5-(4-(2-(M-metyl-N-(2-pyridyl)amino)-etoksy)bensyl)2,4-tiazolidindion ved behandling av polycystisk ovairiesyndrom og gestationell diabetes

Country Status (14)

Country Link
US (1) US5874454A (no)
EP (1) EP0981346A1 (no)
JP (1) JP2001525827A (no)
KR (1) KR20010012556A (no)
AU (1) AU731690B2 (no)
BR (1) BR9809120A (no)
CA (1) CA2282473A1 (no)
HU (1) HUP0003397A3 (no)
IL (1) IL132125A0 (no)
IS (1) IS5177A (no)
NO (1) NO995549D0 (no)
PL (1) PL336764A1 (no)
WO (1) WO1998051305A1 (no)
ZA (1) ZA984084B (no)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6046222A (en) * 1993-09-15 2000-04-04 Warner-Lambert Company Use of thiazolidinedione derivatives in the treatment of polycystic ovary syndrome, gestational diabetes and disease states at risk for progressing to noninsulin-dependent diabetes mellitus
JP2001072592A (ja) 1999-07-01 2001-03-21 Kyowa Hakko Kogyo Co Ltd テロメラーゼ阻害剤
GB0019223D0 (en) * 2000-08-04 2000-09-27 Smithkline Beecham Plc Novel pharmaceutical
GB0021865D0 (en) * 2000-09-06 2000-10-18 Smithkline Beecham Plc Novel pharmaceutical
US6452014B1 (en) 2000-12-22 2002-09-17 Geron Corporation Telomerase inhibitors and methods of their use
CN104163864B (zh) 2007-03-30 2017-08-01 Ambrx公司 经修饰fgf‑21多肽和其用途
US9339458B2 (en) * 2009-02-18 2016-05-17 Itf Research Pharma, S.L.U. Use of vaginal insulin sensitizing agents
ES2344183B1 (es) * 2009-02-18 2011-06-10 Italfarmaco, S.A. Uso de agentes sensibilizantes a insulina por via vaginal.
KR20240024362A (ko) 2014-10-24 2024-02-23 브리스톨-마이어스 스큅 컴퍼니 변형된 fgf-21 폴리펩티드 및 그의 용도
RU2665969C1 (ru) * 2017-05-04 2018-09-05 Федеральное государственное бюджетное образовательное учреждение дополнительного профессионального образования "Российская медицинская академия непрерывного профессионального образования" Министерства здравоохранения Российской Федерации (ФГБОУ ДПО РМАНПО Минздрава России) Способ лечения синдрома поликистозных яичников

Family Cites Families (18)

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Publication number Priority date Publication date Assignee Title
JPS5522636A (en) * 1978-08-04 1980-02-18 Takeda Chem Ind Ltd Thiazoliding derivative
JPS6051189A (ja) * 1983-08-30 1985-03-22 Sankyo Co Ltd チアゾリジン誘導体およびその製造法
AR240698A1 (es) * 1985-01-19 1990-09-28 Takeda Chemical Industries Ltd Procedimiento para preparar compuestos de 5-(4-(2-(5-etil-2-piridil)-etoxi)benzil)-2,4-tiazolidindiona y sus sales
US4873255A (en) * 1987-02-04 1989-10-10 Sankyo Company Limited Thiazolidinone derivatives, their preparation and their use
EP0306228B1 (en) * 1987-09-04 1999-11-17 Beecham Group Plc Substituted thiazolidinedione derivatives
MX15171A (es) * 1988-03-08 1993-05-01 Pfizer Derivados de tiazolidinodiona hipoglicemicos
US5223522A (en) * 1988-03-08 1993-06-29 Pfizer Inc. Thiazolidinedione hypoglycemic agents
US5120754A (en) * 1988-03-08 1992-06-09 Pfizer Inc. Thiazolidinedione hypoglycemic agents
WO1989008650A1 (en) * 1988-03-08 1989-09-21 Pfizer Inc. Thiazolidinedione hypoglycemic agents
US4897405A (en) * 1989-04-21 1990-01-30 American Home Products Corporation Novel naphthalenylalkyl-3H-1,2,3,5-oxathiadiazole 2-oxides useful as antihyperglycemic agents
GB8919417D0 (en) * 1989-08-25 1989-10-11 Beecham Group Plc Novel compounds
GB8919434D0 (en) * 1989-08-25 1989-10-11 Beecham Group Plc Novel compounds
CA2071629C (en) * 1990-02-09 1997-12-30 Jerry R. Colca Use of insulin sensitizing agents to treat hypertension
GB9023585D0 (en) * 1990-10-30 1990-12-12 Beecham Group Plc Novel compounds
GB9023583D0 (en) * 1990-10-30 1990-12-12 Beecham Group Plc Novel compounds
DE69213738T2 (de) * 1991-06-25 1997-01-30 Pfizer Thiazolidindione als hypoglykämische wirkstoffe
EP0719140B1 (en) * 1993-09-15 2007-10-31 Daiichi Sankyo Company, Limited Use of thiazolidinediones to prevent or delay onset of niddm
US5457109A (en) * 1993-09-15 1995-10-10 Warner-Lambert Company Use of thiazolidinedione derivatives and related antihyperglycemic agents in the treatment of disease states at risk for progressing to noninsulin-dependent diabetes mellitus

Also Published As

Publication number Publication date
PL336764A1 (en) 2000-07-17
KR20010012556A (ko) 2001-02-15
EP0981346A1 (en) 2000-03-01
JP2001525827A (ja) 2001-12-11
CA2282473A1 (en) 1998-11-19
ZA984084B (en) 1998-11-20
AU731690B2 (en) 2001-04-05
HUP0003397A2 (hu) 2002-01-28
IL132125A0 (en) 2001-03-19
US5874454A (en) 1999-02-23
WO1998051305A1 (en) 1998-11-19
AU7494998A (en) 1998-12-08
HUP0003397A3 (en) 2002-02-28
NO995549D0 (no) 1999-11-12
IS5177A (is) 1999-09-10
BR9809120A (pt) 2000-08-01

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