NO981501L - Dimer-selektive RXR modulatorer og fremgangsmÕte for anvendelse derav - Google Patents

Dimer-selektive RXR modulatorer og fremgangsmÕte for anvendelse derav

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Publication number
NO981501L
NO981501L NO981501A NO981501A NO981501L NO 981501 L NO981501 L NO 981501L NO 981501 A NO981501 A NO 981501A NO 981501 A NO981501 A NO 981501A NO 981501 L NO981501 L NO 981501L
Authority
NO
Norway
Prior art keywords
dimer
image
selective rxr
rxr
rxr modulators
Prior art date
Application number
NO981501A
Other languages
English (en)
Other versions
NO313186B1 (no
NO981501D0 (no
Inventor
Lin Zhang
Alex M Nadzan
Richard A Heyman
Ranjan Mukherjee
Deepak S Lala
Luc J Farmer
Stacie Canan-Koch
Chan Kou Hwang
Marcus F Boehm
Beth Ann Badea
Laura J Dardashti
Original Assignee
Ligand Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27485410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO981501(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ligand Pharm Inc filed Critical Ligand Pharm Inc
Publication of NO981501D0 publication Critical patent/NO981501D0/no
Publication of NO981501L publication Critical patent/NO981501L/no
Publication of NO313186B1 publication Critical patent/NO313186B1/no

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    • C07D317/10Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/30Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
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    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Mechanical Treatment Of Semiconductor (AREA)
NO19981501A 1995-10-06 1998-04-02 Dimer-selektive RXR modulatorer, farmasöytisk preparat omfattende samme og anvendelse derav for fremstilling avmedikament NO313186B1 (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US489795P 1995-10-06 1995-10-06
US988496P 1996-01-10 1996-01-10
US1831896P 1996-05-24 1996-05-24
US2183996P 1996-07-10 1996-07-10
PCT/US1996/014876 WO1997012853A1 (en) 1995-10-06 1996-09-17 Dimer-selective rxr modulators and methods for their use

Publications (3)

Publication Number Publication Date
NO981501D0 NO981501D0 (no) 1998-04-02
NO981501L true NO981501L (no) 1998-06-02
NO313186B1 NO313186B1 (no) 2002-08-26

Family

ID=27485410

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19981501A NO313186B1 (no) 1995-10-06 1998-04-02 Dimer-selektive RXR modulatorer, farmasöytisk preparat omfattende samme og anvendelse derav for fremstilling avmedikament

Country Status (14)

Country Link
US (2) US6545049B1 (no)
EP (2) EP1336600A3 (no)
JP (1) JP2002515025A (no)
KR (1) KR100625255B1 (no)
AT (1) ATE236115T1 (no)
AU (1) AU726450B2 (no)
BR (1) BR9610875A (no)
CA (1) CA2233888A1 (no)
DE (1) DE69627193T2 (no)
DK (1) DK0873295T3 (no)
ES (1) ES2190479T3 (no)
NO (1) NO313186B1 (no)
PT (1) PT873295E (no)
WO (1) WO1997012853A1 (no)

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US6403638B1 (en) 1998-10-01 2002-06-11 Allergan Sales, Inc. 2,4-pentadienoic acid derivatives having selective activity for retinoid X (RXR) receptors
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US6147224A (en) * 1998-10-01 2000-11-14 Allergan Sales, Inc. 2,4-pentadienoic acid derivatives having selective activity for retinoid X (RXR) receptors
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AU6941200A (en) 1999-08-27 2001-03-26 Ligand Pharmaceuticals Incorporated 8-substituted-6-trifluoromethyl-9-pyrido(3,2-g)quinoline compounds as androgen receptor modulators
BR0013597A (pt) 1999-08-27 2002-07-16 Ligand Pharm Inc Compostos e métodos moduladores de receptor de androgênio
AU1291901A (en) * 1999-09-01 2001-03-26 University Of British Columbia, The Compositions and methods for modulating hdl cholesterol and triglyceride levels
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US7026484B2 (en) 2001-02-23 2006-04-11 Ligand Pharmaceuticals Incorporated Tricyclic androgen receptor modulator compounds and methods
EP1385549A2 (en) * 2001-03-12 2004-02-04 Novartis AG Combination of nateglinide or repaglinide with at least one further antidiabetic compound
MXPA03008229A (es) * 2001-03-14 2004-11-12 Lilly Co Eli Trienos fluorados y su uso como moduladores rxr.
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CA2233888A1 (en) 1997-04-10
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EP1336600A2 (en) 2003-08-20
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US6545049B1 (en) 2003-04-08
AU726450B2 (en) 2000-11-09
EP1336600A3 (en) 2004-07-07
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US20040019072A1 (en) 2004-01-29

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