NO972450L - Substituerte 2-(fosfinyloksymetyl)-1,2,5-tiadiazolidin-3-on 1,1-dioksider og preparater og metode for anvendelse derav - Google Patents
Substituerte 2-(fosfinyloksymetyl)-1,2,5-tiadiazolidin-3-on 1,1-dioksider og preparater og metode for anvendelse deravInfo
- Publication number
- NO972450L NO972450L NO972450A NO972450A NO972450L NO 972450 L NO972450 L NO 972450L NO 972450 A NO972450 A NO 972450A NO 972450 A NO972450 A NO 972450A NO 972450 L NO972450 L NO 972450L
- Authority
- NO
- Norway
- Prior art keywords
- phosphinyloxymethyl
- thiadiazolidin
- dioxides
- substituted
- preparations
- Prior art date
Links
- NETOYMSVSRIRKE-UHFFFAOYSA-N [PH2](=O)OCN1S(NCC1=O)(=O)=O Chemical class [PH2](=O)OCN1S(NCC1=O)(=O)=O NETOYMSVSRIRKE-UHFFFAOYSA-N 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 238000002360 preparation method Methods 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000015122 neurodegenerative disease Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6536—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and sulfur atoms with or without oxygen atoms, as the only ring hetero atoms
- C07F9/6539—Five-membered rings
- C07F9/65392—Five-membered rings containing two nitrogen atoms
- C07F9/65397—Five-membered rings containing two nitrogen atoms having the two nitrogen atoms in positions 1 and 3
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Molecular Biology (AREA)
- Public Health (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Cosmetics (AREA)
- Detergent Compositions (AREA)
Abstract
Substituerte 2-(fosfinyloksymetyl)-l,2,5-tiadiazolidin-3-on 1,1-dioksider, farmasøytiske preparater inneholdende slike forbindelser og metoder for behandling av degenerative sykdommer under anvendelse derav.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/348,411 US5541168A (en) | 1994-12-02 | 1994-12-02 | Substituted 2-(phosphinyloxymethyl)-1,2,5-thiadiazolidin-3-one 1,1-dioxides and compositions and method of use thereof |
PCT/US1995/015565 WO1996016970A1 (en) | 1994-12-02 | 1995-11-30 | Substituted 2-(phosphinyloxymethyl)-1,2,5-thiadiazolidin-3-one 1,1-dioxides and compositions and method of use thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
NO972450D0 NO972450D0 (no) | 1997-05-29 |
NO972450L true NO972450L (no) | 1997-05-29 |
Family
ID=23367928
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO972450A NO972450L (no) | 1994-12-02 | 1997-05-29 | Substituerte 2-(fosfinyloksymetyl)-1,2,5-tiadiazolidin-3-on 1,1-dioksider og preparater og metode for anvendelse derav |
Country Status (12)
Country | Link |
---|---|
US (1) | US5541168A (no) |
EP (1) | EP0794956A4 (no) |
JP (1) | JP2001520626A (no) |
CN (1) | CN1173179A (no) |
AU (1) | AU704233B2 (no) |
CA (1) | CA2205950A1 (no) |
FI (1) | FI972310A (no) |
HU (1) | HUT78043A (no) |
MX (1) | MX9704035A (no) |
NO (1) | NO972450L (no) |
NZ (1) | NZ297344A (no) |
WO (1) | WO1996016970A1 (no) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6420401B1 (en) | 1997-08-22 | 2002-07-16 | Wichita State University | 1,2,5, thiadiazolidin-3-one 1,1-dioxide derivatives |
GT200000203A (es) | 1999-12-01 | 2002-05-24 | Compuestos, composiciones y metodos para estimular el crecimiento y elongacion de neuronas. | |
ATE432074T1 (de) * | 2002-12-30 | 2009-06-15 | Vertex Pharma | Sulfhydantoine als phosphatisostere zur verwendung als phosphatasehemmer bei der behandlung von krebs und autoimmunerkrankungen |
CN113372368B (zh) * | 2020-03-09 | 2022-04-12 | 苏州爱科百发生物医药技术有限公司 | 一种弹性蛋白酶抑制剂前药及其用途 |
WO2024179381A1 (zh) * | 2023-02-28 | 2024-09-06 | 四川科伦博泰生物医药股份有限公司 | 一类化学偶联连接子及其用途 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5236917A (en) * | 1989-05-04 | 1993-08-17 | Sterling Winthrop Inc. | Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof |
DE4141218A1 (de) * | 1991-12-13 | 1993-06-17 | Luitpold Werk Chem Pharm | Thiadiazincarbonsaeureamidderivate, verfahren zu ihrer herstellung und arzneimittel |
US5378720A (en) * | 1991-12-19 | 1995-01-03 | Sterling Winthrop Inc. | Saccharin derivative proteolytic enzyme inhibitors |
AU668694B2 (en) * | 1991-12-19 | 1996-05-16 | Sanofi-Synthelabo | Saccharin derivative proteolytic enzyme inhibitors |
US5187173A (en) * | 1991-12-27 | 1993-02-16 | Sterling Winthrop Inc. | 2-saccharinylmethyl and 4,5,6,7-tetrahydro-2-saccharinylmethyl phosphates, phosphonates and phosphinates useful as proteolytic enzyme inhibitors and compositions and method of use thereof |
US5296496A (en) * | 1991-12-27 | 1994-03-22 | Sterling Winthrop Inc. | 2-saccharinylmethyl phosphates, phosphonates and phosphinates useful as proteolytic enzyme inhibitors and compositions and method of use thereof |
-
1994
- 1994-12-02 US US08/348,411 patent/US5541168A/en not_active Expired - Fee Related
-
1995
- 1995-11-30 WO PCT/US1995/015565 patent/WO1996016970A1/en not_active Application Discontinuation
- 1995-11-30 HU HU9900832A patent/HUT78043A/hu unknown
- 1995-11-30 MX MX9704035A patent/MX9704035A/es unknown
- 1995-11-30 EP EP95940884A patent/EP0794956A4/en not_active Withdrawn
- 1995-11-30 JP JP51905896A patent/JP2001520626A/ja active Pending
- 1995-11-30 AU AU42485/96A patent/AU704233B2/en not_active Ceased
- 1995-11-30 CA CA002205950A patent/CA2205950A1/en not_active Abandoned
- 1995-11-30 NZ NZ297344A patent/NZ297344A/en unknown
- 1995-11-30 CN CN95197438A patent/CN1173179A/zh active Pending
-
1997
- 1997-05-29 NO NO972450A patent/NO972450L/no unknown
- 1997-05-30 FI FI972310A patent/FI972310A/fi unknown
Also Published As
Publication number | Publication date |
---|---|
NO972450D0 (no) | 1997-05-29 |
CN1173179A (zh) | 1998-02-11 |
WO1996016970A1 (en) | 1996-06-06 |
NZ297344A (en) | 1998-11-25 |
US5541168A (en) | 1996-07-30 |
EP0794956A1 (en) | 1997-09-17 |
FI972310A0 (fi) | 1997-05-30 |
AU4248596A (en) | 1996-06-19 |
MX9704035A (es) | 1998-02-28 |
JP2001520626A (ja) | 2001-10-30 |
EP0794956A4 (en) | 1998-02-11 |
FI972310A (fi) | 1997-07-21 |
CA2205950A1 (en) | 1996-06-06 |
AU704233B2 (en) | 1999-04-15 |
HUT78043A (hu) | 1999-07-28 |
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