NO324873B1 - 3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom - Google Patents

3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom Download PDF

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Publication number
NO324873B1
NO324873B1 NO20025106A NO20025106A NO324873B1 NO 324873 B1 NO324873 B1 NO 324873B1 NO 20025106 A NO20025106 A NO 20025106A NO 20025106 A NO20025106 A NO 20025106A NO 324873 B1 NO324873 B1 NO 324873B1
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Norway
Prior art keywords
compound
compound according
mmol
substituted
solution
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Application number
NO20025106A
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English (en)
Norwegian (no)
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NO20025106L (no
NO20025106D0 (no
Inventor
Jeffery R Raymond
Claudia E Kasserra
Yaning Shen
Original Assignee
Inflazyme Pharm Ltd
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Publication of NO20025106D0 publication Critical patent/NO20025106D0/no
Publication of NO20025106L publication Critical patent/NO20025106L/no
Publication of NO324873B1 publication Critical patent/NO324873B1/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0011—Unsubstituted amino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0042—Nitrogen only
    • C07J71/0047—Nitrogen only at position 2(3)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0057—Nitrogen and oxygen
    • C07J71/0063—Nitrogen and oxygen at position 2(3)
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Virology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20025106A 2000-04-28 2002-10-24 3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom NO324873B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20061700P 2000-04-28 2000-04-28
PCT/CA2001/000581 WO2001083512A1 (en) 2000-04-28 2001-04-30 3-nitrogen-6,7-dioxygen steroids and uses related thereto

Publications (3)

Publication Number Publication Date
NO20025106D0 NO20025106D0 (no) 2002-10-24
NO20025106L NO20025106L (no) 2002-12-18
NO324873B1 true NO324873B1 (no) 2007-12-17

Family

ID=22742458

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20025106A NO324873B1 (no) 2000-04-28 2002-10-24 3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom

Country Status (33)

Country Link
US (4) US20040034216A1 (cg-RX-API-DMAC10.html)
EP (1) EP1278763B1 (cg-RX-API-DMAC10.html)
JP (1) JP2003531916A (cg-RX-API-DMAC10.html)
KR (1) KR20030045671A (cg-RX-API-DMAC10.html)
CN (1) CN1214039C (cg-RX-API-DMAC10.html)
AP (1) AP1825A (cg-RX-API-DMAC10.html)
AT (1) ATE353909T1 (cg-RX-API-DMAC10.html)
AU (2) AU2001252084B2 (cg-RX-API-DMAC10.html)
BG (1) BG107289A (cg-RX-API-DMAC10.html)
BR (1) BR0110419A (cg-RX-API-DMAC10.html)
CA (1) CA2418748A1 (cg-RX-API-DMAC10.html)
CO (1) CO5590904A2 (cg-RX-API-DMAC10.html)
DE (1) DE60126597T2 (cg-RX-API-DMAC10.html)
DK (1) DK1278763T3 (cg-RX-API-DMAC10.html)
DZ (1) DZ3355A1 (cg-RX-API-DMAC10.html)
EE (1) EE200200613A (cg-RX-API-DMAC10.html)
ES (1) ES2282247T3 (cg-RX-API-DMAC10.html)
HR (1) HRP20020944A2 (cg-RX-API-DMAC10.html)
HU (1) HUP0300908A2 (cg-RX-API-DMAC10.html)
IL (2) IL152448A0 (cg-RX-API-DMAC10.html)
MA (1) MA25808A1 (cg-RX-API-DMAC10.html)
MX (1) MXPA02010645A (cg-RX-API-DMAC10.html)
NO (1) NO324873B1 (cg-RX-API-DMAC10.html)
NZ (1) NZ522181A (cg-RX-API-DMAC10.html)
OA (1) OA12255A (cg-RX-API-DMAC10.html)
PL (1) PL365798A1 (cg-RX-API-DMAC10.html)
PT (1) PT1278763E (cg-RX-API-DMAC10.html)
RU (1) RU2291873C2 (cg-RX-API-DMAC10.html)
SK (1) SK15692002A3 (cg-RX-API-DMAC10.html)
UA (1) UA79229C2 (cg-RX-API-DMAC10.html)
WO (1) WO2001083512A1 (cg-RX-API-DMAC10.html)
YU (1) YU88102A (cg-RX-API-DMAC10.html)
ZA (1) ZA200208631B (cg-RX-API-DMAC10.html)

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US10100056B2 (en) 2013-03-14 2018-10-16 Aquinox Pharmaceuticals (Canada) Inc. SHIP1 modulators and methods related thereto
SG11201505926VA (en) 2013-03-15 2015-09-29 Biogen Ma Inc Factor ix polypeptide formulations
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Also Published As

Publication number Publication date
CN1430625A (zh) 2003-07-16
NO20025106L (no) 2002-12-18
PL365798A1 (en) 2005-01-10
US20040138186A1 (en) 2004-07-15
WO2001083512A1 (en) 2001-11-08
DE60126597D1 (de) 2007-03-29
US6635629B2 (en) 2003-10-21
MA25808A1 (fr) 2003-07-01
NO20025106D0 (no) 2002-10-24
AU2001252084B2 (en) 2006-07-06
ATE353909T1 (de) 2007-03-15
DK1278763T3 (da) 2007-06-11
IL152448A (en) 2006-12-31
MXPA02010645A (es) 2004-04-20
CA2418748A1 (en) 2001-11-08
AU5208401A (en) 2001-11-12
IL152448A0 (en) 2003-05-29
US7112580B2 (en) 2006-09-26
HK1050694A1 (en) 2003-07-04
CN1214039C (zh) 2005-08-10
SK15692002A3 (sk) 2003-11-04
EP1278763A1 (en) 2003-01-29
YU88102A (sh) 2006-01-16
JP2003531916A (ja) 2003-10-28
EP1278763B1 (en) 2007-02-14
HUP0300908A2 (hu) 2003-07-28
US20040034216A1 (en) 2004-02-19
HRP20020944A2 (en) 2004-02-29
NZ522181A (en) 2005-04-29
US20020072510A1 (en) 2002-06-13
BG107289A (bg) 2003-07-31
US20050215534A9 (en) 2005-09-29
PT1278763E (pt) 2007-05-31
ZA200208631B (en) 2004-02-23
DZ3355A1 (fr) 2001-11-08
EE200200613A (et) 2004-04-15
BR0110419A (pt) 2004-02-25
US20070060553A1 (en) 2007-03-15
CO5590904A2 (es) 2005-12-30
AP1825A (en) 2008-02-03
AP2002002659A0 (en) 2002-12-31
OA12255A (en) 2006-05-11
DE60126597T2 (de) 2007-10-31
ES2282247T3 (es) 2007-10-16
UA79229C2 (en) 2007-06-11
KR20030045671A (ko) 2003-06-11
RU2291873C2 (ru) 2007-01-20

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