NO20090125L - Benzimidazolderivater som skal anvendes som antagonist for CB1-reseptor - Google Patents
Benzimidazolderivater som skal anvendes som antagonist for CB1-reseptorInfo
- Publication number
- NO20090125L NO20090125L NO20090125A NO20090125A NO20090125L NO 20090125 L NO20090125 L NO 20090125L NO 20090125 A NO20090125 A NO 20090125A NO 20090125 A NO20090125 A NO 20090125A NO 20090125 L NO20090125 L NO 20090125L
- Authority
- NO
- Norway
- Prior art keywords
- antagonist
- receptor
- benzimidazole derivatives
- compounds
- treatment
- Prior art date
Links
- 102000009132 CB1 Cannabinoid Receptor Human genes 0.000 title 1
- 108010073366 CB1 Cannabinoid Receptor Proteins 0.000 title 1
- 239000005557 antagonist Substances 0.000 title 1
- 229940058303 antinematodal benzimidazole derivative Drugs 0.000 title 1
- 125000003785 benzimidazolyl group Chemical class N1=C(NC2=C1C=CC=C2)* 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/14—Antitussive agents
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/08—Radicals containing only hydrogen and carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Immunology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychology (AREA)
- Pulmonology (AREA)
- Cardiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Transplantation (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Hospice & Palliative Care (AREA)
- Virology (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Anesthesiology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Forbindelser med formel I, eller farmasøytisk akseptable salter derav, hvori X, A, R1, R2, R3 og R4 er som definert i beskrivelsen så vel som salter og farmasøytiske sammensetninger som inkluderer forbindelsene, er fremstilt. De anvendes ved behandling, særlig for behandling av smerte.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US80459906P | 2006-06-13 | 2006-06-13 | |
PCT/SE2007/000562 WO2007145563A1 (en) | 2006-06-13 | 2007-06-11 | Benzimidazole derivatives which are to be used as antagonist for the cb1-receptor |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20090125L true NO20090125L (no) | 2009-03-09 |
Family
ID=38831987
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20090125A NO20090125L (no) | 2006-06-13 | 2009-01-09 | Benzimidazolderivater som skal anvendes som antagonist for CB1-reseptor |
Country Status (19)
Country | Link |
---|---|
US (1) | US20100305140A1 (no) |
EP (1) | EP2035409A4 (no) |
JP (1) | JP2009539972A (no) |
KR (1) | KR20090021216A (no) |
CN (1) | CN101501022A (no) |
AR (1) | AR061444A1 (no) |
AU (1) | AU2007259425B2 (no) |
BR (1) | BRPI0712305A2 (no) |
CA (1) | CA2654250A1 (no) |
CL (1) | CL2007001715A1 (no) |
EC (1) | ECSP088968A (no) |
IL (1) | IL195426A0 (no) |
MX (1) | MX2008015157A (no) |
NO (1) | NO20090125L (no) |
RU (1) | RU2008148905A (no) |
TW (1) | TW200808772A (no) |
UY (1) | UY30412A1 (no) |
WO (1) | WO2007145563A1 (no) |
ZA (1) | ZA200809977B (no) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE0302573D0 (sv) * | 2003-09-26 | 2003-09-26 | Astrazeneca Ab | Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof |
US20110086853A1 (en) * | 2009-10-08 | 2011-04-14 | William Brown | Therapeutic Compounds |
WO2022087422A1 (en) * | 2020-10-22 | 2022-04-28 | Chulalongkorn University | Pyrrolidine-3-carboxamide derivatives and related uses |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP3295277B2 (ja) * | 1994-06-01 | 2002-06-24 | 呉羽化学工業株式会社 | 抗腎疾患剤及びベンズイミダゾール誘導体 |
US6348032B1 (en) * | 1998-11-23 | 2002-02-19 | Cell Pathways, Inc. | Method of inhibiting neoplastic cells with benzimidazole derivatives |
PA8535601A1 (es) * | 2000-12-21 | 2002-11-28 | Pfizer | Derivados benzimidazol y piridilimidazol como ligandos para gabaa |
SE0101387D0 (sv) * | 2001-04-20 | 2001-04-20 | Astrazeneca Ab | Novel compounds |
SE0301699D0 (sv) * | 2003-06-10 | 2003-06-10 | Astrazeneca Ab | Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof |
SE0301698D0 (sv) * | 2003-06-10 | 2003-06-10 | Astrazeneca Ab | Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof |
WO2006033630A1 (en) * | 2004-09-24 | 2006-03-30 | Astrazeneca Ab | Compounds, compositions containing them, preparation thereof and uses thereof iii |
-
2007
- 2007-06-04 TW TW096119997A patent/TW200808772A/zh unknown
- 2007-06-11 CN CNA2007800302283A patent/CN101501022A/zh active Pending
- 2007-06-11 MX MX2008015157A patent/MX2008015157A/es not_active Application Discontinuation
- 2007-06-11 JP JP2009515341A patent/JP2009539972A/ja active Pending
- 2007-06-11 BR BRPI0712305-1A patent/BRPI0712305A2/pt not_active IP Right Cessation
- 2007-06-11 RU RU2008148905/04A patent/RU2008148905A/ru not_active Application Discontinuation
- 2007-06-11 US US12/303,643 patent/US20100305140A1/en not_active Abandoned
- 2007-06-11 WO PCT/SE2007/000562 patent/WO2007145563A1/en active Application Filing
- 2007-06-11 AU AU2007259425A patent/AU2007259425B2/en not_active Expired - Fee Related
- 2007-06-11 EP EP07748225A patent/EP2035409A4/en not_active Withdrawn
- 2007-06-11 KR KR1020097000549A patent/KR20090021216A/ko not_active Application Discontinuation
- 2007-06-11 CA CA002654250A patent/CA2654250A1/en not_active Abandoned
- 2007-06-12 CL CL2007001715A patent/CL2007001715A1/es unknown
- 2007-06-12 AR ARP070102564A patent/AR061444A1/es unknown
- 2007-06-13 UY UY30412A patent/UY30412A1/es unknown
-
2008
- 2008-11-20 IL IL195426A patent/IL195426A0/en unknown
- 2008-11-24 ZA ZA200809977A patent/ZA200809977B/xx unknown
- 2008-12-12 EC EC2008008968A patent/ECSP088968A/es unknown
-
2009
- 2009-01-09 NO NO20090125A patent/NO20090125L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
JP2009539972A (ja) | 2009-11-19 |
WO2007145563A8 (en) | 2008-11-13 |
CA2654250A1 (en) | 2007-12-21 |
UY30412A1 (es) | 2008-01-31 |
BRPI0712305A2 (pt) | 2012-01-17 |
EP2035409A4 (en) | 2012-01-04 |
ZA200809977B (en) | 2010-04-28 |
US20100305140A1 (en) | 2010-12-02 |
AU2007259425A8 (en) | 2009-01-29 |
AU2007259425A1 (en) | 2007-12-21 |
TW200808772A (en) | 2008-02-16 |
ECSP088968A (es) | 2009-01-30 |
KR20090021216A (ko) | 2009-02-27 |
AR061444A1 (es) | 2008-08-27 |
CN101501022A (zh) | 2009-08-05 |
AU2007259425B2 (en) | 2011-09-08 |
RU2008148905A (ru) | 2010-07-20 |
IL195426A0 (en) | 2009-08-03 |
MX2008015157A (es) | 2008-12-12 |
CL2007001715A1 (es) | 2008-01-18 |
WO2007145563A1 (en) | 2007-12-21 |
EP2035409A1 (en) | 2009-03-18 |
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