NO20084688L - lmidazo[4,5-b]pyridin-2-on og oksazol[4,5-b]pyridin-2-onforbindelser og analoger derav cancerterapeutiske forbindelser - Google Patents

lmidazo[4,5-b]pyridin-2-on og oksazol[4,5-b]pyridin-2-onforbindelser og analoger derav cancerterapeutiske forbindelser

Info

Publication number
NO20084688L
NO20084688L NO20084688A NO20084688A NO20084688L NO 20084688 L NO20084688 L NO 20084688L NO 20084688 A NO20084688 A NO 20084688A NO 20084688 A NO20084688 A NO 20084688A NO 20084688 L NO20084688 L NO 20084688L
Authority
NO
Norway
Prior art keywords
independently
linker
compounds
raf
pyridin
Prior art date
Application number
NO20084688A
Other languages
English (en)
Norwegian (no)
Inventor
Richard Malcolm Marais
Harmen Dijkstra
Dan Niculescu-Duvaz
Caroline Spriger
Delphine Menard
Ion Niculescu-Duvaz
Lawrence Davies
Arnaud Nourry
Original Assignee
Inst Of Cancer Res The Royal C
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB0608268.9A external-priority patent/GB0608268D0/en
Application filed by Inst Of Cancer Res The Royal C filed Critical Inst Of Cancer Res The Royal C
Publication of NO20084688L publication Critical patent/NO20084688L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20084688A 2006-04-26 2008-11-06 lmidazo[4,5-b]pyridin-2-on og oksazol[4,5-b]pyridin-2-onforbindelser og analoger derav cancerterapeutiske forbindelser NO20084688L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US74563306P 2006-04-26 2006-04-26
GBGB0608268.9A GB0608268D0 (en) 2006-04-26 2006-04-26 Therapeutic compounds
PCT/GB2007/001534 WO2007125330A1 (fr) 2006-04-26 2007-04-26 Composés d'imidazo[4,5-b]pyridin-2-one et d'oxazolo[4,5- b]pyridin-2-one et leurs analogues en tant que composés de traitement du cancer

Publications (1)

Publication Number Publication Date
NO20084688L true NO20084688L (no) 2009-01-26

Family

ID=38421488

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20084688A NO20084688L (no) 2006-04-26 2008-11-06 lmidazo[4,5-b]pyridin-2-on og oksazol[4,5-b]pyridin-2-onforbindelser og analoger derav cancerterapeutiske forbindelser

Country Status (7)

Country Link
US (1) US7951819B2 (fr)
EP (1) EP2013207B1 (fr)
JP (1) JP2009534457A (fr)
AU (1) AU2007245495A1 (fr)
CA (1) CA2649994A1 (fr)
NO (1) NO20084688L (fr)
WO (1) WO2007125330A1 (fr)

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CN110446523B (zh) 2017-01-12 2022-06-10 加利福尼亚大学董事会 用于重症护理的血管内灌流增强
EP3612086A4 (fr) 2017-04-21 2021-01-20 The Regents of the University of California, A California Corporation Débitmètre aortique et pompe pour occlusion aortique partielle
BR112020015581A2 (pt) 2018-01-31 2021-02-02 Deciphera Pharmaceuticals, Llc terapia de combinação para o tratamento de tumores estromais gastrointestinais
CA3149846A1 (fr) 2019-08-08 2021-02-11 B.C.I. Pharma Derives d'isoquinoline utilises comme inhibiteurs de proteine kinase
MX2022001863A (es) 2019-08-12 2022-05-30 Deciphera Pharmaceuticals Llc Metodos para tratar los tumores del estroma gastrointestinal.
WO2021030405A1 (fr) 2019-08-12 2021-02-18 Deciphera Pharmaceuticals, Llc Ripretinib pour le traitement de tumeurs stromales gastro-intestinales
WO2021057696A1 (fr) * 2019-09-27 2021-04-01 隆泰申医药科技(南京)有限公司 Composé hétéroaryle et ses applications
EP4084779A1 (fr) 2019-12-30 2022-11-09 Deciphera Pharmaceuticals, LLC Compositions de 1-(4-bromo-5-(1-éthyl-7-(méthylamino)-2-oxo-1,2-dihydro -1,6-naphthyridine-3-yl)-2-fluorophényl)-3-phényluree
AU2020419197B2 (en) 2019-12-30 2023-08-31 Deciphera Pharmaceuticals, Llc Amorphous kinase inhibitor formulations and methods of use thereof
JP2023519191A (ja) 2020-03-16 2023-05-10 サータス クリティカル ケア， インコーポレイテッド 血流制御デバイス、システム、及び方法、並びにそれらのエラー検出
US11629143B2 (en) 2020-10-01 2023-04-18 Vibliome Therapeutics, Llc HipK4 inhibitors and uses thereof
TWI812301B (zh) * 2021-06-24 2023-08-11 南韓商Ｌｇ化學股份有限公司 作為ｒｏｎ抑制劑之新穎尿素衍生物化合物
US11779572B1 (en) 2022-09-02 2023-10-10 Deciphera Pharmaceuticals, Llc Methods of treating gastrointestinal stromal tumors

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Also Published As

Publication number Publication date
CA2649994A1 (fr) 2007-11-08
US20090325945A1 (en) 2009-12-31
US7951819B2 (en) 2011-05-31
JP2009534457A (ja) 2009-09-24
WO2007125330A1 (fr) 2007-11-08
AU2007245495A1 (en) 2007-11-08
EP2013207B1 (fr) 2012-04-25
EP2013207A1 (fr) 2009-01-14

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