NO20076345L - Bisykliske derivater som P38-kinaseinhibitorer - Google Patents

Bisykliske derivater som P38-kinaseinhibitorer

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Publication number
NO20076345L
NO20076345L NO20076345A NO20076345A NO20076345L NO 20076345 L NO20076345 L NO 20076345L NO 20076345 A NO20076345 A NO 20076345A NO 20076345 A NO20076345 A NO 20076345A NO 20076345 L NO20076345 L NO 20076345L
Authority
NO
Norway
Prior art keywords
kinase inhibitors
bicyclic derivatives
derivatives
bicyclic
meanings
Prior art date
Application number
NO20076345A
Other languages
English (en)
Norwegian (no)
Inventor
Marina Virgili Bernando
Carmen Almansa Rosales
Original Assignee
Palau Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Palau Pharma Sa filed Critical Palau Pharma Sa
Publication of NO20076345L publication Critical patent/NO20076345L/no

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    • C07C233/65—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
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    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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NO20076345A 2005-06-29 2007-12-11 Bisykliske derivater som P38-kinaseinhibitorer NO20076345L (no)

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PCT/EP2006/006256 WO2007000340A2 (en) 2005-06-29 2006-06-28 Bicyclic derivatives as p38 kinase inhibitors

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EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
US20090082368A1 (en) * 2007-09-24 2009-03-26 Painceptor Pharma Corporation Methods of modulating neurotrophin-mediated activity
AU2008313733A1 (en) 2007-10-18 2009-04-23 Boehringer Ingelheim International Gmbh CGRP antagonists
EP2065381A1 (de) 2007-10-18 2009-06-03 Boehringer Ingelheim Pharma GmbH & Co. KG CGRP Antagonisten
CA2705405A1 (en) 2007-11-22 2009-05-28 Boehringer Ingelheim International Gmbh New compounds
WO2009065922A2 (de) * 2007-11-22 2009-05-28 Boehringer Ingelheim International Gmbh Organische verbindungen
EP2062889A1 (de) * 2007-11-22 2009-05-27 Boehringer Ingelheim Pharma GmbH & Co. KG Verbindungen
WO2009072581A1 (ja) * 2007-12-05 2009-06-11 Aska Pharmaceutical Co., Ltd. ラクタム化合物又はその塩及びｐｐａｒ活性化剤
US10513515B2 (en) 2017-08-25 2019-12-24 Biotheryx, Inc. Ether compounds and uses thereof
US11236103B2 (en) 2018-07-27 2022-02-01 Biotheryx, Inc. Bifunctional compounds
EP4143329A4 (en) 2020-04-28 2024-10-16 Anwita Biosciences Inc INTERLEUKIN-2 POLYPEPTIDES AND FUSION PROTEINS THEREOF, AS WELL AS THEIR PHARMACEUTICAL COMPOSITIONS AND THERAPEUTIC APPLICATIONS
WO2023229685A2 (en) * 2022-02-24 2023-11-30 Microbiotix, Inc. Broad-spectrum inhibitors of cytomegalovirus

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WO2004108672A1 (en) 2003-06-02 2004-12-16 Abbott Laboratories Isoindolin-1-one compounds as kinase inhibitors
US20050182061A1 (en) 2003-10-02 2005-08-18 Jeremy Green Phthalimide compounds useful as protein kinase inhibitors
JP2007008816A (ja) 2003-10-15 2007-01-18 Ube Ind Ltd 新規イソキノリン誘導体

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AR055344A1 (es) 2007-08-22
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WO2007000340A3 (en) 2007-03-29
BRPI0613958A2 (pt) 2011-02-22
WO2007000340A8 (en) 2007-05-18
CN101213175A (zh) 2008-07-02
RU2008103218A (ru) 2009-08-10
KR20080029976A (ko) 2008-04-03
CA2612008A1 (en) 2007-01-04
JP2008544965A (ja) 2008-12-11
WO2007000340A2 (en) 2007-01-04
IL188027A0 (en) 2008-03-20
US20100222363A1 (en) 2010-09-02
EP1907358A2 (en) 2008-04-09

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