NO20071616L - Benzoksazin- og kinoksalinderivater og anvendelser - Google Patents

Benzoksazin- og kinoksalinderivater og anvendelser

Info

Publication number
NO20071616L
NO20071616L NO20071616A NO20071616A NO20071616L NO 20071616 L NO20071616 L NO 20071616L NO 20071616 A NO20071616 A NO 20071616A NO 20071616 A NO20071616 A NO 20071616A NO 20071616 L NO20071616 L NO 20071616L
Authority
NO
Norway
Prior art keywords
cinoxaline
benzoxazine
derivatives
medicaments
manufacture
Prior art date
Application number
NO20071616A
Other languages
English (en)
Norwegian (no)
Inventor
Shu-Hai Zhao
Douglas William Bonhaus
Renee Sharon Martin
Steven Sethofer
Li Zhang
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO20071616L publication Critical patent/NO20071616L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/536Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/341,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/361,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20071616A 2004-09-30 2007-03-27 Benzoksazin- og kinoksalinderivater og anvendelser NO20071616L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US61470504P 2004-09-30 2004-09-30
US63060804P 2004-11-24 2004-11-24
PCT/EP2005/010238 WO2006037481A1 (en) 2004-09-30 2005-09-22 Benzoxazine and quinoxaline derivatives and uses

Publications (1)

Publication Number Publication Date
NO20071616L true NO20071616L (no) 2007-04-25

Family

ID=35385358

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20071616A NO20071616L (no) 2004-09-30 2007-03-27 Benzoksazin- og kinoksalinderivater og anvendelser

Country Status (17)

Country Link
EP (1) EP1797051B1 (de)
JP (1) JP2008514662A (de)
KR (1) KR100875041B1 (de)
AR (1) AR051115A1 (de)
AT (1) ATE477248T1 (de)
AU (1) AU2005291541B2 (de)
BR (1) BRPI0516754A (de)
CA (1) CA2581921A1 (de)
DE (1) DE602005022896D1 (de)
IL (1) IL182304A0 (de)
MX (1) MX2007003911A (de)
MY (1) MY139409A (de)
NO (1) NO20071616L (de)
NZ (1) NZ553848A (de)
RU (1) RU2382036C2 (de)
TW (1) TW200626567A (de)
WO (1) WO2006037481A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2301625B1 (de) * 2004-09-30 2017-07-19 F. Hoffmann-La Roche AG Zusammensetzungen und verfahren zur behandlung kognitiver störungen
CL2007003044A1 (es) * 2006-10-24 2008-07-04 Wyeth Corp Compuestos derivados de benzoxazina; composicion farmaceutica que los comprende; y uso para el tratamiento de un trastorno psicotico, bipolar, depresivo y abuso o dependencia de sustancias entre otros.
BRPI0920520A2 (pt) * 2008-09-08 2015-12-22 Hoffmann La Roche benzoxazinas 5-subistituídas
CA2953004C (en) * 2014-07-08 2023-02-21 Sunshine Lake Pharma Co., Ltd. Aromatic heterocyclic derivatives and pharmaceutical applications thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW224941B (de) * 1989-11-08 1994-06-11 Yamanouchi Pharma Co Ltd
KR20010108025A (ko) * 1998-12-17 2001-12-07 이곤 이 버그 5HT2C 효능제인2,3,4,4a-테트라하이드로-1H-피라지노(1,2-a)퀴녹살린-5(6H)온 유도체
WO2003029238A1 (en) * 2001-10-04 2003-04-10 Wyeth Chroman derivatives as 5-hydroxytryptamine-6 ligands
WO2003095434A1 (en) * 2002-05-13 2003-11-20 F. Hoffmann-La Roche Ag Benzoxazine derivatives as 5-ht6 modulators and uses thereof
EP2301625B1 (de) * 2004-09-30 2017-07-19 F. Hoffmann-La Roche AG Zusammensetzungen und verfahren zur behandlung kognitiver störungen

Also Published As

Publication number Publication date
AR051115A1 (es) 2006-12-20
IL182304A0 (en) 2007-07-24
EP1797051B1 (de) 2010-08-11
AU2005291541B2 (en) 2011-03-10
KR20070047844A (ko) 2007-05-07
MX2007003911A (es) 2007-05-21
MY139409A (en) 2009-09-30
KR100875041B1 (ko) 2008-12-19
JP2008514662A (ja) 2008-05-08
ATE477248T1 (de) 2010-08-15
CA2581921A1 (en) 2006-04-13
TW200626567A (en) 2006-08-01
WO2006037481A1 (en) 2006-04-13
AU2005291541A1 (en) 2006-04-13
EP1797051A1 (de) 2007-06-20
DE602005022896D1 (de) 2010-09-23
BRPI0516754A (pt) 2008-09-16
NZ553848A (en) 2010-01-29
RU2382036C2 (ru) 2010-02-20
RU2007110479A (ru) 2008-11-10

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application