NO20070299L - Novel heterocyclic compounds - Google Patents

Novel heterocyclic compounds

Info

Publication number
NO20070299L
NO20070299L NO20070299A NO20070299A NO20070299L NO 20070299 L NO20070299 L NO 20070299L NO 20070299 A NO20070299 A NO 20070299A NO 20070299 A NO20070299 A NO 20070299A NO 20070299 L NO20070299 L NO 20070299L
Authority
NO
Norway
Prior art keywords
heterocyclic compounds
novel heterocyclic
novel
compounds
heterocyclic
Prior art date
Application number
NO20070299A
Other languages
English (en)
Inventor
Braj Bhushan Lohray
Vidya Bhushan Lohray
Brijesh Srivastava
Original Assignee
Cadila Healthcare Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cadila Healthcare Ltd filed Critical Cadila Healthcare Ltd
Publication of NO20070299L publication Critical patent/NO20070299L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • A61K31/4161,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • A61K31/41621,2-Diazoles condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO20070299A 2004-07-12 2007-01-17 Novel heterocyclic compounds NO20070299L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN745MU2004 2004-07-12
PCT/IN2005/000237 WO2006025069A2 (en) 2004-07-12 2005-07-08 Tricyclic pyrazole derivatives as cannabinoid receptor modulators

Publications (1)

Publication Number Publication Date
NO20070299L true NO20070299L (no) 2007-03-26

Family

ID=35636669

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20070299A NO20070299L (no) 2004-07-12 2007-01-17 Novel heterocyclic compounds

Country Status (20)

Country Link
US (2) US8030345B2 (no)
EP (2) EP1781668A2 (no)
JP (1) JP2008505965A (no)
KR (1) KR20070041717A (no)
CN (1) CN101014605A (no)
AP (1) AP2228A (no)
AU (1) AU2005278781B2 (no)
BR (1) BRPI0513104A (no)
CA (1) CA2586011C (no)
EA (1) EA011307B1 (no)
EC (1) ECSP077167A (no)
GE (1) GEP20094682B (no)
IL (1) IL180637A0 (no)
MX (1) MX2007000491A (no)
NO (1) NO20070299L (no)
NZ (2) NZ552670A (no)
TN (1) TNSN07006A1 (no)
UA (1) UA88910C2 (no)
WO (1) WO2006025069A2 (no)
ZA (1) ZA200700162B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1781668A2 (en) * 2004-07-12 2007-05-09 Cadila Healthcare Ltd. Tricyclic pyrazole derivatives as cannabinoid receptor modulators
IN2012DN02474A (no) 2009-08-28 2015-08-21 Arena Pharm Inc
US9597340B2 (en) 2011-02-25 2017-03-21 Arena Pharmaceuticals, Inc. Cannabinoid receptor modulators
US20140206649A1 (en) 2011-02-25 2014-07-24 Jayant Thatte Cannabinoid receptor modulators
JP5945554B2 (ja) 2011-02-25 2016-07-05 アリーナ ファーマシューティカルズ, インコーポレイテッド 縮合型アザ環の結晶形およびその調製プロセス(カンナビノイド受容体モジュレーター)
US10351576B2 (en) * 2015-04-30 2019-07-16 Novartis Ag Fused tricyclic pyrazole derivatives useful for farnesoid X receptors
EP3402780A1 (en) 2016-01-14 2018-11-21 Beth Israel Deaconess Medical Center, Inc. Mast-cell modulators and uses thereof
JP2021511364A (ja) * 2018-01-29 2021-05-06 カディラ ヘルスケア リミティド 抗菌剤として有用な複素環式化合物

Family Cites Families (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3260721A (en) * 1962-04-10 1966-07-12 American Cyanamid Co Heterocyclic derivatives of yohimbe alkaloids
EP0003115A1 (en) * 1978-01-16 1979-07-25 Sandoz Ag Penicillins, per se and for use as antibacterially active antibiotics and their production
DE3374166D1 (en) 1983-04-22 1987-12-03 Mitsubishi Rayon Co Apparatus for measuring gas partial pressure in living body
FR2692575B1 (fr) 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2713225B1 (fr) 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
CA2106642C (en) * 1992-10-14 2005-08-16 Peter Bod Carbazolone derivatives and process for preparing the same
FR2714057B1 (fr) 1993-12-17 1996-03-08 Sanofi Elf Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant.
US5547975A (en) 1994-09-20 1996-08-20 Talley; John J. Benzopyranopyrazolyl derivatives for the treatment of inflammation
FR2741621B1 (fr) 1995-11-23 1998-02-13 Sanofi Sa Nouveaux derives de pyrazole, procede pour leur preparation et compositions pharmaceutiques en contenant
FR2742148B1 (fr) 1995-12-08 1999-10-22 Sanofi Sa Nouveaux derives du pyrazole-3-carboxamide, procede pour leur preparation et compositions pharmaceutiques les contenant
FR2758723B1 (fr) 1997-01-28 1999-04-23 Sanofi Sa Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour la preparation de medicaments
FR2761266B1 (fr) 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates
FR2789079B3 (fr) 1999-02-01 2001-03-02 Sanofi Synthelabo Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant
FR2800375B1 (fr) 1999-11-03 2004-07-23 Sanofi Synthelabo Derives tricycliques d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant
FR2800372B1 (fr) * 1999-11-03 2001-12-07 Sanofi Synthelabo Derives tricycliques d'acide 1-benzylpyrazole-3- carboxylique, leur preparation, les medicaments en contenant
FR2804604B1 (fr) 2000-02-09 2005-05-27 Sanofi Synthelabo Utilisation d'un antagoniste des recepteurs aux cannabinoides centraux pour la preparation de medicaments utiles pour faciliter l'arret de la consommation de tabac
FR2809621B1 (fr) 2000-05-12 2002-09-06 Sanofi Synthelabo Utilisation d'un antagoniste des recepteurs aux cannabinoides centraux pour la preparation de medicaments utiles comme antidiarrheiques
FR2816938B1 (fr) 2000-11-22 2003-01-03 Sanofi Synthelabo Derives de 3-aroylindole, leur procede de preparation et les compositions pharmaceutiques en contenant
JP2005507875A (ja) 2001-08-31 2005-03-24 ユニバーシティ オブ コネチカット カンナビノイド受容体に作用する新規なピラゾール類似体
TWI231757B (en) 2001-09-21 2005-05-01 Solvay Pharm Bv 1H-Imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity
WO2003026648A1 (en) 2001-09-21 2003-04-03 Solvay Pharmaceuticals B.V. 4,5-dihydro-1h-pyrazole derivatives having potent cb1-antagonistic activity
ATE344663T1 (de) 2001-09-21 2006-11-15 Solvay Pharm Bv Neue 4,5-dihydro-1h-pyrazol-derivate mit cb1- antagonistischer wirkung
US6509367B1 (en) 2001-09-22 2003-01-21 Virginia Commonwealth University Pyrazole cannabinoid agonist and antagonists
CA2476665A1 (en) * 2002-02-19 2003-08-28 Pharmacia Corporation Tricyclic pyrazole derivatives for the treatment of inflammation
ITMI20041033A1 (it) * 2004-05-24 2004-08-24 Neuroscienze S C A R L Composti farmaceutici
EP1781668A2 (en) * 2004-07-12 2007-05-09 Cadila Healthcare Ltd. Tricyclic pyrazole derivatives as cannabinoid receptor modulators

Also Published As

Publication number Publication date
BRPI0513104A (pt) 2008-04-29
WO2006025069A2 (en) 2006-03-09
US20100273791A1 (en) 2010-10-28
ECSP077167A (es) 2007-05-30
CA2586011A1 (en) 2006-03-09
WO2006025069A8 (en) 2007-03-15
CN101014605A (zh) 2007-08-08
AU2005278781A1 (en) 2006-03-09
UA88910C2 (ru) 2009-12-10
EP2343302A1 (en) 2011-07-13
TNSN07006A1 (en) 2008-06-02
AU2005278781B2 (en) 2009-06-18
JP2008505965A (ja) 2008-02-28
ZA200700162B (en) 2009-09-30
IL180637A0 (en) 2007-06-03
AP2228A (en) 2011-04-01
WO2006025069A3 (en) 2006-04-27
KR20070041717A (ko) 2007-04-19
EA200700246A1 (ru) 2007-08-31
NZ580387A (en) 2011-06-30
US8030345B2 (en) 2011-10-04
US20080051386A1 (en) 2008-02-28
NZ552670A (en) 2010-02-26
EP1781668A2 (en) 2007-05-09
CA2586011C (en) 2011-07-19
EA011307B1 (ru) 2009-02-27
GEP20094682B (en) 2009-05-10
AP2007003880A0 (en) 2007-02-28
MX2007000491A (es) 2007-03-28

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