NO20063621L - Derivater av N-`(1,5-difenyl-1H-pyrazol-3-yl) sulfonamid med CB1 receptoraffinitet - Google Patents

Derivater av N-`(1,5-difenyl-1H-pyrazol-3-yl) sulfonamid med CB1 receptoraffinitet

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Publication number
NO20063621L
NO20063621L NO20063621A NO20063621A NO20063621L NO 20063621 L NO20063621 L NO 20063621L NO 20063621 A NO20063621 A NO 20063621A NO 20063621 A NO20063621 A NO 20063621A NO 20063621 L NO20063621 L NO 20063621L
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Norway
Prior art keywords
alkyl
pyrazol
sulfonamide
diphenyl
derivatives
Prior art date
Application number
NO20063621A
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English (en)
Inventor
Christian Congy
Francis Barth
Murielle Rinaldi-Carmona
Serge Martinez
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Sanofi Aventis
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Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of NO20063621L publication Critical patent/NO20063621L/no

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Abstract

Det beskrives forbindelser med formel (I) der Ri betyr (Ci-C) alkyl, (C-C) cykloalkyl som eventuelt er mono- eller polysubstituert, (C-C) cykloalkylmetyl som er eventuelt er mono- eller polysubstituert, fenyl som eventuelt er usubstituert eller substituert, benzyl som eventuelt er usubstituert eller mono- eller disubstituert, tienyl som eventuelt er usubstituert eller substituert; Rbetyr hydrogen eller (C-C) alkyl; Rbetyr hydrogen eller (C-C) alkyl; R, R, Rs, R, Rg og Rhver uavhengig av hverandre betyr hydrogen, halogen (C-C) alkyl, (C-C) alkoksy, trifiuormetyl eller S(0)„Alk; n betyr 0, 1 eller 2; og Alk betyr (C-C) alkyl.Videre beskrives fremgangsmåter for fremstilling av forbindelsen og deres anvendelse i medikamenter.
NO20063621A 2004-01-12 2006-08-10 Derivater av N-`(1,5-difenyl-1H-pyrazol-3-yl) sulfonamid med CB1 receptoraffinitet NO20063621L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0400257A FR2864958B1 (fr) 2004-01-12 2004-01-12 Derive de n-[(1,5-diphenyl-1h-pyrazol-3-yl)methyl] sulfonamide, leur preparation et leur application en therapeutique.
PCT/FR2005/000031 WO2005073197A1 (fr) 2004-01-12 2005-01-07 Derives de n-` (1,5-diphenyl-1h-pyrazol-3-yl) sulfonamide avec une affinite pour les recepteurs cb1

Publications (1)

Publication Number Publication Date
NO20063621L true NO20063621L (no) 2006-10-10

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US (1) US7294645B2 (no)
EP (1) EP1720837B1 (no)
JP (1) JP4723514B2 (no)
KR (1) KR20060105050A (no)
CN (1) CN1910157A (no)
AR (1) AR047096A1 (no)
AT (1) ATE465995T1 (no)
AU (1) AU2005209441B2 (no)
CA (1) CA2551141C (no)
CR (1) CR8468A (no)
CY (1) CY1110651T1 (no)
DE (1) DE602005020907D1 (no)
DK (1) DK1720837T3 (no)
EC (1) ECSP066695A (no)
ES (1) ES2344850T3 (no)
FR (1) FR2864958B1 (no)
HR (1) HRP20100283T8 (no)
IL (1) IL176710A0 (no)
MA (1) MA28422B1 (no)
NO (1) NO20063621L (no)
NZ (1) NZ548442A (no)
PL (1) PL1720837T3 (no)
PT (1) PT1720837E (no)
RS (1) RS51365B (no)
RU (1) RU2366657C2 (no)
SI (1) SI1720837T1 (no)
TN (1) TNSN06203A1 (no)
TW (1) TWI323255B (no)
UA (1) UA85079C2 (no)
WO (1) WO2005073197A1 (no)
ZA (1) ZA200605657B (no)

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FR2880890B1 (fr) * 2005-01-19 2007-03-30 Sanofi Aventis Sa Derives de n-[(4,5-diphenyl-2-thienyl)methyl]sulfonamide, leur preparation et leur application en therapeutique
FR2881744B1 (fr) * 2005-02-09 2007-04-27 Sanofi Aventis Sa Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique
FR2894579B1 (fr) * 2005-12-12 2008-01-18 Sanofi Aventis Sa Derives diaryltriazolmethylamine, leur preparation et leur application en therapeutique.
FR2894578B1 (fr) * 2005-12-12 2008-02-01 Sanofi Aventis Sa Derives heterocycliques, leur preparation et leur application en therapeutique.
EP1829867A1 (en) 2006-03-03 2007-09-05 Laboratorios Del Dr. Esteve, S.A. Imidazole compounds having pharmaceutical activity towards the sigma receptor
FR2899899A1 (fr) * 2006-04-14 2007-10-19 Sanofi Aventis Sa Derives d'aminomethyl pyridine, leur preparation et leur application en therapeutique
ATE469129T1 (de) * 2006-07-11 2010-06-15 Sanofi Aventis N-ä(1,5-diphenyl-1h-pyrazol-3- yl)methylüsulfonamid-derivate antagonisten der cb1 rezeptoren der cannabinoide
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JP2008019205A (ja) * 2006-07-12 2008-01-31 Sanofi-Aventis Ｎ−［（１，５−ジフェニル−１ｈ−ピラゾール−３−イル）メチル］スルホンアミド誘導体、その調製法および治療におけるその応用
WO2008062424A2 (en) * 2006-07-31 2008-05-29 Cadila Healthcare Limited Substituted 4,5-dihydro-1h-pyrazole derivatives as cannabinoid modulators
US7875647B2 (en) 2006-09-29 2011-01-25 Green Cross Corporation Heteroaryl-pyrazole derivatives as cannabinoid CB1 receptor antagonists
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US20070021486A1 (en) 2007-01-25
RU2006129297A (ru) 2008-02-20
PL1720837T3 (pl) 2010-09-30
EP1720837A1 (fr) 2006-11-15
FR2864958B1 (fr) 2006-02-24
US7294645B2 (en) 2007-11-13
HRP20100283T1 (hr) 2010-08-31
ZA200605657B (en) 2007-12-27
ES2344850T3 (es) 2010-09-08
IL176710A0 (en) 2006-10-31
KR20060105050A (ko) 2006-10-09
EP1720837B1 (fr) 2010-04-28
JP2007517839A (ja) 2007-07-05
HRP20100283T8 (en) 2010-10-31
CY1110651T1 (el) 2015-06-10
AR047096A1 (es) 2006-01-04
FR2864958A1 (fr) 2005-07-15
UA85079C2 (en) 2008-12-25
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CN1910157A (zh) 2007-02-07
JP4723514B2 (ja) 2011-07-13
AU2005209441A1 (en) 2005-08-11
RS51365B (en) 2011-02-28
DE602005020907D1 (de) 2010-06-10
WO2005073197A1 (fr) 2005-08-11
RU2366657C2 (ru) 2009-09-10
MA28422B1 (fr) 2007-02-01
ECSP066695A (es) 2006-10-31
CA2551141C (fr) 2011-06-07
NZ548442A (en) 2009-10-30
CR8468A (es) 2007-03-06
SI1720837T1 (sl) 2010-08-31
ATE465995T1 (de) 2010-05-15
PT1720837E (pt) 2010-05-14
TNSN06203A1 (en) 2007-11-15
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