NO20061324L - Polymorfe former av en kjent antihyperlinemisk forbindelse - Google Patents
Polymorfe former av en kjent antihyperlinemisk forbindelseInfo
- Publication number
- NO20061324L NO20061324L NO20061324A NO20061324A NO20061324L NO 20061324 L NO20061324 L NO 20061324L NO 20061324 A NO20061324 A NO 20061324A NO 20061324 A NO20061324 A NO 20061324A NO 20061324 L NO20061324 L NO 20061324L
- Authority
- NO
- Norway
- Prior art keywords
- polymorphic forms
- antihyperlinemic
- compound
- preparation
- dihydroxyheptide
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
To nye polymorfe former av (E)-7-[4-(4-fIuorfenyl)-6-isopropyl-2-[metyl(metylsulfonyl)amino]pyrimidin 5-y1](3R,5S)-3,5-dihydroksyhept-6-ensyre tris(hydroksymetyl)metylammoniumsalt (1), metoder for fremstilling av disse og anvendelse av disse ved fremstilling av farmasøytisk anvendelige preparater ved behandling av, bl.a. hyperkolesterolermi, hyperlipoproteinemi og aterosklerose er beskrevet.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0321827.8A GB0321827D0 (en) | 2003-09-18 | 2003-09-18 | Chemical compounds |
PCT/GB2004/004133 WO2005028450A1 (en) | 2003-09-18 | 2004-09-17 | Polymorphic forms of a known antihyperlipemic agent |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20061324L true NO20061324L (no) | 2006-04-04 |
Family
ID=29227290
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20061324A NO20061324L (no) | 2003-09-18 | 2006-03-23 | Polymorfe former av en kjent antihyperlinemisk forbindelse |
Country Status (13)
Country | Link |
---|---|
US (1) | US20070105882A1 (no) |
EP (1) | EP1663990A1 (no) |
JP (1) | JP2007505879A (no) |
CN (1) | CN100439342C (no) |
AU (1) | AU2004274239B2 (no) |
BR (1) | BRPI0414499A (no) |
CA (1) | CA2538756A1 (no) |
GB (1) | GB0321827D0 (no) |
IL (1) | IL174164A0 (no) |
NO (1) | NO20061324L (no) |
NZ (1) | NZ546007A (no) |
WO (1) | WO2005028450A1 (no) |
ZA (1) | ZA200602263B (no) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0003305D0 (en) | 2000-02-15 | 2000-04-05 | Zeneca Ltd | Pyrimidine derivatives |
GB0011120D0 (en) | 2000-05-09 | 2000-06-28 | Avecia Ltd | Process |
NL1015744C2 (nl) * | 2000-07-19 | 2002-01-22 | Dsm Nv | Werkwijze voor de bereiding van 2-(6-gesubstitueerde-1,3-dioxan-4-yl) azijnzuurderivaten. |
HUP0401248A3 (en) | 2001-07-13 | 2004-11-29 | Astrazeneca Uk Ltd | Preparation of aminopyrimidine compounds and new intermediates |
EP1323717A1 (en) | 2001-12-27 | 2003-07-02 | Dsm N.V. | Process for the preparation of 2-(6-Substituted-1,3-Dioxane-4-yL) acetic acid derivatives |
EP1375493A1 (en) | 2002-06-17 | 2004-01-02 | Dsm N.V. | Process for the preparation of an dioxane acetic acid ester |
GB0218781D0 (en) | 2002-08-13 | 2002-09-18 | Astrazeneca Ab | Chemical process |
JP4579821B2 (ja) | 2002-12-16 | 2010-11-10 | アストラゼネカ・ユーケイ・リミテッド | ピリミジン化合物を製造するための方法 |
GB0312896D0 (en) * | 2003-06-05 | 2003-07-09 | Astrazeneca Ab | Chemical process |
UY28501A1 (es) | 2003-09-10 | 2005-04-29 | Astrazeneca Uk Ltd | Compuestos químicos |
GB0322552D0 (en) | 2003-09-26 | 2003-10-29 | Astrazeneca Uk Ltd | Therapeutic treatment |
GB0324791D0 (en) * | 2003-10-24 | 2003-11-26 | Astrazeneca Ab | Chemical process |
GB0428328D0 (en) * | 2004-12-24 | 2005-02-02 | Astrazeneca Uk Ltd | Chemical process |
GB0514078D0 (en) * | 2005-07-08 | 2005-08-17 | Astrazeneca Uk Ltd | Chemical process |
TW200831469A (en) * | 2006-12-01 | 2008-08-01 | Astrazeneca Uk Ltd | Chemical process |
WO2010082072A1 (en) * | 2009-01-15 | 2010-07-22 | Egis Gyógyszergyár | Process for the preparation of rosuvastatin salts |
WO2012073256A1 (en) | 2010-11-29 | 2012-06-07 | Cadila Healthcare Limited | Salts of rosuvastatin |
US9873677B2 (en) | 2014-03-06 | 2018-01-23 | Ptc Therapeutics, Inc. | Pharmaceutical compositions and salts of a 1,2,4-oxadiazole benzoic acid |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5026698A (en) * | 1988-11-02 | 1991-06-25 | Nissan Chemical Industries, Ltd. | Thienopyridine type mevalonolactones |
JP2648897B2 (ja) * | 1991-07-01 | 1997-09-03 | 塩野義製薬株式会社 | ピリミジン誘導体 |
US6278001B1 (en) * | 1995-11-28 | 2001-08-21 | L'oréal | Method for preparing (+) compactin and (+) mevinolin analog compounds having a β-hydroxy-δ-lactone grouping |
GB9903472D0 (en) * | 1999-02-17 | 1999-04-07 | Zeneca Ltd | Chemical process |
GB0003305D0 (en) * | 2000-02-15 | 2000-04-05 | Zeneca Ltd | Pyrimidine derivatives |
NL1015744C2 (nl) * | 2000-07-19 | 2002-01-22 | Dsm Nv | Werkwijze voor de bereiding van 2-(6-gesubstitueerde-1,3-dioxan-4-yl) azijnzuurderivaten. |
IL158525A0 (en) * | 2001-06-06 | 2004-05-12 | Bristol Myers Squibb Co | A process for preparing chiral diol sulfone derivatives |
KR20040026705A (ko) * | 2001-08-16 | 2004-03-31 | 테바 파마슈티컬 인더스트리즈 리미티드 | 스타틴의 칼슘 염 형태의 제조 방법 |
GB0218781D0 (en) * | 2002-08-13 | 2002-09-18 | Astrazeneca Ab | Chemical process |
WO2005054207A1 (en) * | 2003-12-04 | 2005-06-16 | Glenmark Pharmaceuticals Limited | Process for the preparation of pyrimidine derivatives |
US7241800B2 (en) * | 2004-03-17 | 2007-07-10 | Mai De Ltd. | Anhydrous amorphous form of fluvastatin sodium |
-
2003
- 2003-09-18 GB GBGB0321827.8A patent/GB0321827D0/en not_active Ceased
-
2004
- 2004-09-17 US US10/572,635 patent/US20070105882A1/en not_active Abandoned
- 2004-09-17 AU AU2004274239A patent/AU2004274239B2/en not_active Ceased
- 2004-09-17 WO PCT/GB2004/004133 patent/WO2005028450A1/en active Application Filing
- 2004-09-17 CN CNB2004800268240A patent/CN100439342C/zh not_active Expired - Fee Related
- 2004-09-17 JP JP2006526703A patent/JP2007505879A/ja not_active Withdrawn
- 2004-09-17 CA CA002538756A patent/CA2538756A1/en not_active Abandoned
- 2004-09-17 EP EP04768676A patent/EP1663990A1/en not_active Withdrawn
- 2004-09-17 BR BRPI0414499-6A patent/BRPI0414499A/pt not_active IP Right Cessation
- 2004-09-17 NZ NZ546007A patent/NZ546007A/en unknown
-
2006
- 2006-03-07 IL IL174164A patent/IL174164A0/en unknown
- 2006-03-23 NO NO20061324A patent/NO20061324L/no not_active Application Discontinuation
-
2007
- 2007-03-17 ZA ZA200602263A patent/ZA200602263B/en unknown
Also Published As
Publication number | Publication date |
---|---|
CN100439342C (zh) | 2008-12-03 |
EP1663990A1 (en) | 2006-06-07 |
WO2005028450A1 (en) | 2005-03-31 |
AU2004274239A1 (en) | 2005-03-31 |
AU2004274239B2 (en) | 2008-12-04 |
IL174164A0 (en) | 2006-08-01 |
CA2538756A1 (en) | 2005-03-31 |
NZ546007A (en) | 2008-11-28 |
US20070105882A1 (en) | 2007-05-10 |
BRPI0414499A (pt) | 2006-11-14 |
ZA200602263B (en) | 2007-11-28 |
CN1852899A (zh) | 2006-10-25 |
JP2007505879A (ja) | 2007-03-15 |
GB0321827D0 (en) | 2003-10-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |