NO20060936L - Tiomorfolinsteroidforbindelser, anvendelse derav for fremstilling av meioseregulerende medikamenter og fremgangsmate for fremstilling derav - Google Patents

Tiomorfolinsteroidforbindelser, anvendelse derav for fremstilling av meioseregulerende medikamenter og fremgangsmate for fremstilling derav

Info

Publication number
NO20060936L
NO20060936L NO20060936A NO20060936A NO20060936L NO 20060936 L NO20060936 L NO 20060936L NO 20060936 A NO20060936 A NO 20060936A NO 20060936 A NO20060936 A NO 20060936A NO 20060936 L NO20060936 L NO 20060936L
Authority
NO
Norway
Prior art keywords
preparation
meiosis
thiomorpholine
steroid compounds
steroid
Prior art date
Application number
NO20060936A
Other languages
English (en)
Inventor
Thorsten Blume
Bernhard Lindenthal
Katja Prelle
Michaele Peters-Kottig
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of NO20060936L publication Critical patent/NO20060936L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Reproductive Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Epidemiology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)

Abstract

Foreliggende oppfinnelse gjelder tiomorfolinosteroidforbindelser med den generelle formel (I), som med fordel kan anvendes for stimulenng av meiosen i humane oocytter, hvor steroidet særpreges ved at en tiomorfohnogruppe er bundet til C'^ i steroidskjelettet via en alkylengruppe.
NO20060936A 2003-07-28 2006-02-27 Tiomorfolinsteroidforbindelser, anvendelse derav for fremstilling av meioseregulerende medikamenter og fremgangsmate for fremstilling derav NO20060936L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP03090237A EP1514874A1 (en) 2003-07-28 2003-07-28 Thiomorpholino steroid compounds, the use thereof for the preparation of meiosis regulating medicaments and method for the preparation thereof
PCT/EP2004/007737 WO2005014613A1 (en) 2003-07-28 2004-07-13 Thiomorpholino steroid compounds, the use thereof for the preparation of meiosis-regulating medicaments and method for the preparation thereof

Publications (1)

Publication Number Publication Date
NO20060936L true NO20060936L (no) 2006-02-27

Family

ID=34130263

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20060936A NO20060936L (no) 2003-07-28 2006-02-27 Tiomorfolinsteroidforbindelser, anvendelse derav for fremstilling av meioseregulerende medikamenter og fremgangsmate for fremstilling derav

Country Status (19)

Country Link
US (1) US20070078262A1 (no)
EP (2) EP1514874A1 (no)
JP (1) JP2007500140A (no)
KR (1) KR20060059991A (no)
CN (1) CN1829731A (no)
AT (1) ATE393772T1 (no)
AU (1) AU2004263252A1 (no)
BR (1) BRPI0412342A (no)
CA (1) CA2528904A1 (no)
DE (1) DE602004013453T2 (no)
DK (1) DK1664079T3 (no)
ES (1) ES2305813T3 (no)
IL (1) IL172085A0 (no)
NO (1) NO20060936L (no)
PL (1) PL1664079T3 (no)
PT (1) PT1664079E (no)
RU (1) RU2349597C2 (no)
WO (1) WO2005014613A1 (no)
ZA (1) ZA200601711B (no)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2813094A (en) * 1955-02-16 1957-11-12 Searle & Co Cyclic derivatives of 3-hydroxy-delta-pregnene-20-carboxamide
US2846432A (en) * 1957-10-31 1958-08-05 Searle & Co Heterocyclic derivatives of 20-amino-methyl-5-pregnen-3-ol
DE1930473A1 (de) * 1969-06-14 1970-12-17 Schering Ag 22-N-substituierte (20R)-23,24-dinor-cholanderivate
US3983111A (en) * 1972-05-05 1976-09-28 Glaxo Laboratories Limited Steroidal anaesthetics of the pregnane and 19-norpregnane series
GB9804861D0 (en) * 1998-03-06 1998-04-29 Res Inst Medicine Chem Chemical compounds
EP1245572A1 (en) * 2001-03-26 2002-10-02 Schering Aktiengesellschaft Aminosterol compounds, their use in the preparation of meiosis-regulating medicaments and method for their preparation

Also Published As

Publication number Publication date
CN1829731A (zh) 2006-09-06
RU2349597C2 (ru) 2009-03-20
PT1664079E (pt) 2008-07-14
BRPI0412342A (pt) 2006-09-05
IL172085A0 (en) 2009-02-11
EP1664079A1 (en) 2006-06-07
DK1664079T3 (da) 2008-08-04
ATE393772T1 (de) 2008-05-15
PL1664079T3 (pl) 2008-09-30
EP1664079B1 (en) 2008-04-30
EP1514874A1 (en) 2005-03-16
ZA200601711B (en) 2007-05-30
DE602004013453D1 (de) 2008-06-12
CA2528904A1 (en) 2005-02-17
WO2005014613A1 (en) 2005-02-17
ES2305813T3 (es) 2008-11-01
AU2004263252A1 (en) 2005-02-17
US20070078262A1 (en) 2007-04-05
JP2007500140A (ja) 2007-01-11
KR20060059991A (ko) 2006-06-02
RU2006105783A (ru) 2007-09-20
DE602004013453T2 (de) 2009-06-18

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application