NO20054053L - Triazolforbindelser anvendbare i terapi. - Google Patents

Triazolforbindelser anvendbare i terapi.

Info

Publication number
NO20054053L
NO20054053L NO20054053A NO20054053A NO20054053L NO 20054053 L NO20054053 L NO 20054053L NO 20054053 A NO20054053 A NO 20054053A NO 20054053 A NO20054053 A NO 20054053A NO 20054053 L NO20054053 L NO 20054053L
Authority
NO
Norway
Prior art keywords
alkyl
optionally substituted
independently represent
ring
heterocyclic group
Prior art date
Application number
NO20054053A
Other languages
English (en)
Norwegian (no)
Other versions
NO20054053D0 (no
Inventor
Alan Stobie
Christopher Peter Wayman
Justin Stephen Bryans
Patrick Stephen Johnson
Rachel Jane Russel
Thomas Ryckmans
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB0303852.8A external-priority patent/GB0303852D0/en
Priority claimed from GBGB0317227.7A external-priority patent/GB0317227D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of NO20054053D0 publication Critical patent/NO20054053D0/no
Publication of NO20054053L publication Critical patent/NO20054053L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N2333/00—Assays involving biological materials from specific organisms or of a specific nature
    • G01N2333/435—Assays involving biological materials from specific organisms or of a specific nature from animals; from humans
    • G01N2333/705—Assays involving receptors, cell surface antigens or cell surface determinants
    • G01N2333/72—Assays involving receptors, cell surface antigens or cell surface determinants for hormones
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N2500/00—Screening for compounds of potential therapeutic value
    • G01N2500/04—Screening involving studying the effect of compounds C directly on molecule A (e.g. C are potential ligands for a receptor A, or potential substrates for an enzyme A)

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pulmonology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Urology & Nephrology (AREA)
  • Psychiatry (AREA)
  • Pregnancy & Childbirth (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Otolaryngology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Anesthesiology (AREA)
  • Vascular Medicine (AREA)
NO20054053A 2003-02-19 2005-08-31 Triazolforbindelser anvendbare i terapi. NO20054053L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0303852.8A GB0303852D0 (en) 2003-02-19 2003-02-19 Triazole compounds useful in therapy
GBGB0317227.7A GB0317227D0 (en) 2003-07-23 2003-07-23 Treatment of male sexual dysfunction
PCT/IB2004/000432 WO2004074291A1 (en) 2003-02-19 2004-02-09 Triazole compounds useful in therapy

Publications (2)

Publication Number Publication Date
NO20054053D0 NO20054053D0 (no) 2005-08-31
NO20054053L true NO20054053L (no) 2005-10-31

Family

ID=34889119

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20054053A NO20054053L (no) 2003-02-19 2005-08-31 Triazolforbindelser anvendbare i terapi.

Country Status (25)

Country Link
EP (1) EP1597260B1 (pt)
JP (2) JP4033886B2 (pt)
KR (1) KR100750028B1 (pt)
AP (1) AP2005003376A0 (pt)
AT (1) ATE349449T1 (pt)
AU (1) AU2004213242B2 (pt)
BR (1) BRPI0407676A (pt)
CA (1) CA2516557C (pt)
DE (1) DE602004003914T2 (pt)
DK (1) DK1597260T3 (pt)
EA (1) EA009460B1 (pt)
EC (1) ECSP055973A (pt)
ES (1) ES2277237T3 (pt)
GE (1) GEP20074089B (pt)
HR (1) HRP20050681A2 (pt)
IS (1) IS2450B (pt)
MA (1) MA27712A1 (pt)
MX (1) MXPA05008923A (pt)
NO (1) NO20054053L (pt)
OA (1) OA13029A (pt)
PL (1) PL378747A1 (pt)
PT (1) PT1597260E (pt)
RS (1) RS20050638A (pt)
SI (1) SI1597260T1 (pt)
TN (1) TNSN05200A1 (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200904403A (en) * 2007-04-25 2009-02-01 Daiichi Sankyo Co Ltd Tricyclic aryl compounds
CN102812011A (zh) * 2009-11-16 2012-12-05 梅利科技公司 [1,5]-二氮杂环辛间四烯衍生物
US8420633B2 (en) * 2010-03-31 2013-04-16 Hoffmann-La Roche Inc. Aryl-cyclohexyl-tetraazabenzo[e]azulenes
US8461151B2 (en) * 2010-04-13 2013-06-11 Hoffmann-La Roche Inc. Aryl-/heteroaryl-cyclohexenyl-tetraazabenzo[e]azulenes
US8492376B2 (en) * 2010-04-21 2013-07-23 Hoffmann-La Roche Inc. Heteroaryl-cyclohexyl-tetraazabenzo[e]azulenes
US8481528B2 (en) * 2010-04-26 2013-07-09 Hoffmann-La Roche Inc. Heterobiaryl-cyclohexyl-tetraazabenzo[e]azulenes
US9006450B2 (en) 2010-07-01 2015-04-14 Boehringer Ingelheim International Gmbh Compounds, pharmaceutical compositions and uses thereof
SI3077396T1 (sl) * 2013-12-05 2021-08-31 F. Hoffmann-La Roche Ag Sinteza trans-8-kloro-5-metil-1-(4-(piridin-2-iloksi)-cikloheksil)-5,6- dihidro-4H-2,3,5,10b-tetraaza-benzo(e)azulena in njegovih kristalnih oblik
HU231206B1 (hu) * 2017-12-15 2021-10-28 Richter Gedeon Nyrt. Triazolobenzazepinek

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8823475D0 (en) * 1988-10-06 1988-11-16 Merck Sharp & Dohme Chemical compounds
US5438035A (en) * 1994-06-24 1995-08-01 American Cyanamid Company Methods for controlling undesirable plant species with benzodiazepine compounds
US5753648A (en) * 1995-01-17 1998-05-19 American Cyanamid Company Tricyclic benzazepine vasopressin antagonists
DE69725182T2 (de) * 1996-11-01 2004-06-24 Wyeth 5H PYRROLO[2,1-c][1,4]BENZODIAZEPIN-3-CARBOXAMIDDERIVATE
TR200102069T2 (tr) * 1999-01-19 2001-11-21 Ortho-Mcneil Pharmaceutical, Inc. Vasopresin reseptörü antagonistleri olarak trisiklik benzodiazepinler.
US7109193B2 (en) * 2001-04-12 2006-09-19 Wyeth Tricyclic diazepines tocolytic oxytocin receptor antagonists
GB0224919D0 (en) * 2002-10-25 2002-12-04 Pfizer Ltd Triazole compounds useful in therapy

Also Published As

Publication number Publication date
ATE349449T1 (de) 2007-01-15
GEP20074089B (en) 2007-04-10
IS2450B (is) 2008-11-15
JP2007045838A (ja) 2007-02-22
TNSN05200A1 (fr) 2007-06-11
SI1597260T1 (sl) 2007-04-30
MXPA05008923A (es) 2006-03-09
EA200501136A1 (ru) 2006-06-30
EP1597260B1 (en) 2006-12-27
AU2004213242A1 (en) 2004-09-02
HRP20050681A2 (en) 2005-12-31
DK1597260T3 (da) 2007-04-02
MA27712A1 (fr) 2006-01-02
PT1597260E (pt) 2007-01-31
IS7957A (is) 2005-07-25
JP4033886B2 (ja) 2008-01-16
AP2005003376A0 (en) 2005-09-30
CA2516557A1 (en) 2004-09-02
AU2004213242B2 (en) 2007-04-19
NO20054053D0 (no) 2005-08-31
EP1597260A1 (en) 2005-11-23
OA13029A (en) 2006-11-10
PL378747A1 (pl) 2006-05-15
DE602004003914D1 (de) 2007-02-08
KR20050106443A (ko) 2005-11-09
EA009460B1 (ru) 2007-12-28
RS20050638A (en) 2007-12-31
BRPI0407676A (pt) 2006-03-01
KR100750028B1 (ko) 2007-08-16
ECSP055973A (es) 2006-01-16
ES2277237T3 (es) 2007-07-01
DE602004003914T2 (de) 2007-05-31
JP2006517921A (ja) 2006-08-03
CA2516557C (en) 2008-11-18

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