NO20051009L - Syntese av indoliziner - Google Patents
Syntese av indolizinerInfo
- Publication number
- NO20051009L NO20051009L NO20051009A NO20051009A NO20051009L NO 20051009 L NO20051009 L NO 20051009L NO 20051009 A NO20051009 A NO 20051009A NO 20051009 A NO20051009 A NO 20051009A NO 20051009 L NO20051009 L NO 20051009L
- Authority
- NO
- Norway
- Prior art keywords
- following formula
- indolizines
- represented
- synthesis
- reacting
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Abstract
Det er beskrevet fremgangsmåter for fremstilling av substituerte indoliziner representert ved følgende formel: omfattende omsetning av et substrat representert ved følgende formel: med enten sykliseringsreagens med følgende fonnel: eller, et reagens fremstilt ved omsetning av forbindelsene representert ved formelen nedenfor med et alkyleringsmiddel: Variablene i ovennevnte formler er definert heri.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US41067902P | 2002-09-13 | 2002-09-13 | |
PCT/US2003/028252 WO2004024727A2 (en) | 2002-09-13 | 2003-09-10 | Synthesis of indolizines |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20051009L true NO20051009L (no) | 2005-04-04 |
Family
ID=31994182
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20051009A NO20051009L (no) | 2002-09-13 | 2005-02-24 | Syntese av indoliziner |
Country Status (10)
Country | Link |
---|---|
US (1) | US20040152897A1 (no) |
EP (1) | EP1537105A2 (no) |
JP (1) | JP2006504692A (no) |
KR (1) | KR20050052498A (no) |
CN (1) | CN1681813A (no) |
AU (1) | AU2003267071A1 (no) |
CA (1) | CA2496764A1 (no) |
MX (1) | MXPA05002745A (no) |
NO (1) | NO20051009L (no) |
WO (1) | WO2004024727A2 (no) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102060806A (zh) | 2003-09-11 | 2011-05-18 | iTherX药品公司 | 细胞因子抑制剂 |
WO2005099824A1 (en) * | 2004-03-30 | 2005-10-27 | Synta Pharmaceuticals, Corp. | 1-glyoxylamide indolizines for treating lung and ovarian cancer |
JP2010501562A (ja) | 2006-08-21 | 2010-01-21 | シンタ ファーマシューティカルズ コーポレーション | 増殖性障害を治療するための化合物 |
US8581004B2 (en) | 2008-02-21 | 2013-11-12 | Synta Pharmaceuticals Corp. | Compounds for treating proliferative disorders |
US8673460B2 (en) * | 2009-09-10 | 2014-03-18 | Lg Chem, Ltd. | Heterocyclic derivative and organic light emitting device using same |
JOP20190024A1 (ar) | 2016-08-26 | 2019-02-19 | Gilead Sciences Inc | مركبات بيروليزين بها استبدال واستخداماتها |
US10836769B2 (en) | 2018-02-26 | 2020-11-17 | Gilead Sciences, Inc. | Substituted pyrrolizine compounds and uses thereof |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1996003383A1 (en) * | 1994-07-21 | 1996-02-08 | Eli Lilly And Company | INDOLIZINE sPLA2 INHIBITORS |
WO1998047507A1 (en) * | 1997-04-24 | 1998-10-29 | Shionogi & Co., Ltd. | Method for the treatment of stroke using n-heterocyclic glyoxylamide compounds |
EP1007525A1 (en) * | 1997-08-29 | 2000-06-14 | Zeneca Limited | Aminometyl oxooxazolidinyl benzene derivatives |
ATE300542T1 (de) * | 2001-09-13 | 2005-08-15 | Synta Pharmaceuticals Corp | 1-glyoxlylamidindolizine zur behandlung von krebs |
-
2003
- 2003-09-10 JP JP2004536391A patent/JP2006504692A/ja not_active Withdrawn
- 2003-09-10 KR KR1020057004319A patent/KR20050052498A/ko not_active Application Discontinuation
- 2003-09-10 AU AU2003267071A patent/AU2003267071A1/en not_active Abandoned
- 2003-09-10 CN CNA038217406A patent/CN1681813A/zh active Pending
- 2003-09-10 CA CA002496764A patent/CA2496764A1/en not_active Abandoned
- 2003-09-10 MX MXPA05002745A patent/MXPA05002745A/es not_active Application Discontinuation
- 2003-09-10 EP EP03749545A patent/EP1537105A2/en not_active Withdrawn
- 2003-09-10 WO PCT/US2003/028252 patent/WO2004024727A2/en active Application Filing
- 2003-09-11 US US10/660,358 patent/US20040152897A1/en not_active Abandoned
-
2005
- 2005-02-24 NO NO20051009A patent/NO20051009L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AU2003267071A1 (en) | 2004-04-30 |
CA2496764A1 (en) | 2004-03-25 |
KR20050052498A (ko) | 2005-06-02 |
WO2004024727A2 (en) | 2004-03-25 |
WO2004024727A3 (en) | 2004-06-03 |
CN1681813A (zh) | 2005-10-12 |
EP1537105A2 (en) | 2005-06-08 |
JP2006504692A (ja) | 2006-02-09 |
MXPA05002745A (es) | 2005-06-03 |
US20040152897A1 (en) | 2004-08-05 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |