NO20044970L - Indolderivater, fremgangsmate for fremstilling av de samme og farmasoytiske preparater inneholdende de samme - Google Patents

Indolderivater, fremgangsmate for fremstilling av de samme og farmasoytiske preparater inneholdende de samme

Info

Publication number
NO20044970L
NO20044970L NO20044970A NO20044970A NO20044970L NO 20044970 L NO20044970 L NO 20044970L NO 20044970 A NO20044970 A NO 20044970A NO 20044970 A NO20044970 A NO 20044970A NO 20044970 L NO20044970 L NO 20044970L
Authority
NO
Norway
Prior art keywords
same
indole derivatives
preparing
processes
pharmaceutical compositions
Prior art date
Application number
NO20044970A
Other languages
English (en)
Inventor
Francis Barth
Carole Guillaumont
Murielle Rinaldi-Carmona
Claude Vernhet
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of NO20044970L publication Critical patent/NO20044970L/no

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Virology (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Psychology (AREA)
  • Otolaryngology (AREA)

Abstract

Oppfinnelsen vedrører forbindelse med formel (I) og deres fremstilling og farmasøytiske preparater inneholdende de samme. Forbindelsene er cannabinoid CB2 reseptor-ligander.
NO20044970A 2002-05-17 2004-11-15 Indolderivater, fremgangsmate for fremstilling av de samme og farmasoytiske preparater inneholdende de samme NO20044970L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0206133A FR2839718B1 (fr) 2002-05-17 2002-05-17 Derives d'indole, leur procede de preparation et les compositions pharmaceutiques en contenant
PCT/FR2003/001470 WO2003097597A2 (fr) 2002-05-17 2003-05-15 Derives d'indole et leur utilisation en tant que ligands des recepteurs cb2

Publications (1)

Publication Number Publication Date
NO20044970L true NO20044970L (no) 2005-02-17

Family

ID=29286599

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20044970A NO20044970L (no) 2002-05-17 2004-11-15 Indolderivater, fremgangsmate for fremstilling av de samme og farmasoytiske preparater inneholdende de samme

Country Status (20)

Country Link
US (1) US7138424B2 (no)
EP (1) EP1507758B1 (no)
JP (1) JP2005530797A (no)
KR (1) KR20040106560A (no)
CN (1) CN1668588A (no)
AT (1) ATE308518T1 (no)
AU (1) AU2003258762A1 (no)
BR (1) BR0311185A (no)
CA (1) CA2482756A1 (no)
DE (1) DE60302156T2 (no)
EA (1) EA200401315A1 (no)
FR (1) FR2839718B1 (no)
HR (1) HRP20041073A2 (no)
IL (1) IL164941A0 (no)
IS (1) IS7513A (no)
MA (1) MA27203A1 (no)
MX (1) MXPA04011387A (no)
NO (1) NO20044970L (no)
PL (1) PL374111A1 (no)
WO (1) WO2003097597A2 (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7067539B2 (en) * 2001-02-08 2006-06-27 Schering Corporation Cannabinoid receptor ligands
UY27939A1 (es) 2002-08-21 2004-03-31 Glaxo Group Ltd Compuestos
TW200505902A (en) * 2003-03-20 2005-02-16 Schering Corp Cannabinoid receptor ligands
GB0402355D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
TW200533657A (en) * 2004-02-17 2005-10-16 Esteve Labor Dr Substituted pyrazoline compounds, their preparation and use as medicaments
MX2007006102A (es) * 2004-11-22 2007-07-11 Threshold Pharmaceuticals Inc Agentes anti-cancer de union a tubulina y profarmacos de los mismos.
EP1743892A1 (en) * 2005-07-15 2007-01-17 Laboratorios del Dr. Esteve S.A. Substituted pyrazoline compounds, their preparation and use as medicaments
FR2893615B1 (fr) 2005-11-18 2008-03-07 Sanofi Aventis Sa Derives de 3-acylindole, leur preparation et leur application en therapeutique
GB0702862D0 (en) * 2007-02-14 2007-03-28 Univ Aberdeen Therapeutic compounds
EP2408761B1 (en) * 2007-08-29 2014-01-01 Merck Sharp & Dohme Corp. Substituted indole derivatives and methods of use thereof
FR2933697B1 (fr) 2008-07-11 2010-08-13 Sanofi Aventis Derives de 1-benzyl-cinnolin-4-(1h)-one substitues, leur preparation et leur application en therapeutique
FR2950055A1 (fr) 2009-09-17 2011-03-18 Sanofi Aventis Derives de 3-amino-cinnolin-4(1h)-one substitues, leur preparation et leur application en therapeutique
FR2983859B1 (fr) 2011-12-12 2014-01-17 Sanofi Sa Derives de 1,3,5-triazine-2-amine, leur preparation et leur application en diagnostique et en therapeutique

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2735774B1 (fr) 1995-06-21 1997-09-12 Sanofi Sa Utilisation de composes agonistes du recepteur cb2 humain pour la preparation de medicaments immunomodulateurs, nouveaux composes agonistes du recepteur cb2 et les compositions pharmaceutiques les contenant
AU1095101A (en) * 1999-10-18 2001-04-30 University Of Connecticut, The Cannabimimetic indole derivatives

Also Published As

Publication number Publication date
AU2003258762A1 (en) 2003-12-02
DE60302156D1 (de) 2005-12-08
BR0311185A (pt) 2005-02-22
ATE308518T1 (de) 2005-11-15
HRP20041073A2 (en) 2004-12-31
CA2482756A1 (fr) 2003-11-27
CN1668588A (zh) 2005-09-14
EP1507758B1 (fr) 2005-11-02
US7138424B2 (en) 2006-11-21
FR2839718B1 (fr) 2004-06-25
MXPA04011387A (es) 2005-02-14
KR20040106560A (ko) 2004-12-17
IS7513A (is) 2004-10-20
DE60302156T2 (de) 2006-07-20
JP2005530797A (ja) 2005-10-13
WO2003097597A2 (fr) 2003-11-27
IL164941A0 (en) 2005-12-18
US20060089345A1 (en) 2006-04-27
MA27203A1 (fr) 2005-01-03
EA200401315A1 (ru) 2005-04-28
PL374111A1 (en) 2005-10-03
WO2003097597A3 (fr) 2004-04-01
EP1507758A2 (fr) 2005-02-23
FR2839718A1 (fr) 2003-11-21

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