NO165802C - ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOPYRIDINES. - Google Patents

ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOPYRIDINES.

Info

Publication number
NO165802C
NO165802C NO870251A NO870251A NO165802C NO 165802 C NO165802 C NO 165802C NO 870251 A NO870251 A NO 870251A NO 870251 A NO870251 A NO 870251A NO 165802 C NO165802 C NO 165802C
Authority
NO
Norway
Prior art keywords
preparation
therapeutic active
alkyl
hydrogen
analogue procedure
Prior art date
Application number
NO870251A
Other languages
Norwegian (no)
Other versions
NO165802B (en
NO870251D0 (en
NO870251L (en
Inventor
Pascal George
Claudie Giron
Jacques Froissant
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8600836A external-priority patent/FR2593181B1/en
Priority claimed from FR8601553A external-priority patent/FR2593818B1/en
Application filed by Synthelabo filed Critical Synthelabo
Publication of NO870251D0 publication Critical patent/NO870251D0/en
Publication of NO870251L publication Critical patent/NO870251L/en
Publication of NO165802B publication Critical patent/NO165802B/en
Publication of NO165802C publication Critical patent/NO165802C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Abstract

Compounds of general formula (I) <IMAGE> in which R1 is hydrogen or an alkyl or benzyl group and R2 is an alkyl, alkenyl, phenyl or benzyl group, or else R1 and R2 form an aliphatic chain, each of X1, X2 and X3 is hydrogen or a halogen or an alkyl, methoxy, alkylthio, methylsulphonyl, trifluoromethyl, carboxyl, cyano, nitro, amino or aminocarbonyl group, and Y is hydrogen or a halogen or a methyl, trifluoromethyl, carboxyl, cyano, amino or aminocarbonyl group. Application in therapeutics.y
NO870251A 1986-01-22 1987-01-21 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOPYRIDINES. NO165802C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8600836A FR2593181B1 (en) 1986-01-22 1986-01-22 IMIDAZO ACYLAMINOMETHYL-3 DERIVATIVES (1,2-A) PYRIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR8601553A FR2593818B1 (en) 1986-02-05 1986-02-05 IMIDAZO (1,2-A) PYRIDINE ACYLAMINOMETHYL-3 DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Publications (4)

Publication Number Publication Date
NO870251D0 NO870251D0 (en) 1987-01-21
NO870251L NO870251L (en) 1987-07-23
NO165802B NO165802B (en) 1991-01-02
NO165802C true NO165802C (en) 1991-04-10

Family

ID=26224973

Family Applications (1)

Application Number Title Priority Date Filing Date
NO870251A NO165802C (en) 1986-01-22 1987-01-21 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOPYRIDINES.

Country Status (15)

Country Link
EP (1) EP0234970B1 (en)
KR (1) KR870007174A (en)
AT (1) ATE62687T1 (en)
AU (1) AU586065B2 (en)
CA (1) CA1263390A (en)
DE (1) DE3769333D1 (en)
DK (1) DK32287A (en)
ES (1) ES2032455T3 (en)
FI (1) FI870254A (en)
GR (1) GR3002080T3 (en)
HU (1) HU196400B (en)
IL (1) IL81334A (en)
NO (1) NO165802C (en)
NZ (1) NZ219006A (en)
PT (1) PT84161B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0289371B1 (en) * 1987-03-27 1991-09-25 Synthelabo Imidazopyridine derivatives, their preparation and therapeutical use
FR2615513B1 (en) * 1987-05-21 1989-07-13 Synthelabo DERIVATIVES OF ACYLAMINOMETHYL-3 TETRAHYDRO-5,6,7,8 IMIDAZO (1,2-A) PYRIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
DE4405378A1 (en) * 1994-02-19 1995-08-24 Merck Patent Gmbh Adhesion receptor antagonists
US6596731B2 (en) 2001-03-27 2003-07-22 Hoffmann-La Roche Inc. Substituted imidazo[1,2-A] pyridine derivatives
WO2006051063A1 (en) * 2004-11-11 2006-05-18 Ferrer Internacional S. A. Imidazo[1,2-a]pyridine compounds, compositions, uses and methods related thereto
WO2009143156A2 (en) * 2008-05-19 2009-11-26 Sepracor Inc. IMIDAZO[1,2-a]PYRIDINE COMPOUNDS

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB991589A (en) * 1963-04-30 1965-05-12 Selvi & C Lab Bioterapico Novel [1,2-ª‡]imidazopyridines and a process for the manufacture thereof
US3408496A (en) * 1964-11-23 1968-10-29 Parametrics Inc Alpha ray excited composition analysis
ZA81219B (en) * 1980-01-23 1982-01-27 Schering Corp Imidazo (1,2-a) pyridines ,process for their preparation and pharmaceutical compositions containing them
FR2492382A1 (en) * 1980-10-22 1982-04-23 Synthelabo IMIDAZO (1,2-A) PYRIDINE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC USE THEREOF
FR2568880B1 (en) * 1984-08-07 1986-12-12 Synthelabo IMIDAZO ACYLAMINOMETHYL-3 DERIVATIVES (1,2-A) PYRIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR2600650B1 (en) * 1986-06-27 1988-09-09 Synthelabo PROCESS FOR THE PREPARATION OF IMIDAZOPYRIDINES AND INTERMEDIATE COMPOUNDS

Also Published As

Publication number Publication date
FI870254A (en) 1987-07-23
DE3769333D1 (en) 1991-05-23
ES2032455T3 (en) 1993-02-16
EP0234970A1 (en) 1987-09-02
DK32287A (en) 1987-07-23
AU6789587A (en) 1987-07-23
CA1263390A (en) 1989-11-28
DK32287D0 (en) 1987-01-21
ATE62687T1 (en) 1991-05-15
GR3002080T3 (en) 1992-12-30
NO165802B (en) 1991-01-02
PT84161B (en) 1989-07-31
HUT43064A (en) 1987-09-28
FI870254A0 (en) 1987-01-21
HU196400B (en) 1988-11-28
NO870251D0 (en) 1987-01-21
IL81334A (en) 1991-01-31
NO870251L (en) 1987-07-23
NZ219006A (en) 1989-05-29
EP0234970B1 (en) 1991-04-17
KR870007174A (en) 1987-08-17
IL81334A0 (en) 1987-08-31
PT84161A (en) 1987-02-01
AU586065B2 (en) 1989-06-29

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