AU586065B2 - 3-(acylaminomethyl)imidazo``1,2-a`` pyridine derivatives their preparation and their application in therapy - Google Patents

3-(acylaminomethyl)imidazo``1,2-a`` pyridine derivatives their preparation and their application in therapy

Info

Publication number
AU586065B2
AU586065B2 AU67895/87A AU6789587A AU586065B2 AU 586065 B2 AU586065 B2 AU 586065B2 AU 67895/87 A AU67895/87 A AU 67895/87A AU 6789587 A AU6789587 A AU 6789587A AU 586065 B2 AU586065 B2 AU 586065B2
Authority
AU
Australia
Prior art keywords
application
acylaminomethyl
imidazo
therapy
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU67895/87A
Other versions
AU6789587A (en
Inventor
Jacques Froissant
Pascal George
Claudie Giron
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8600836A external-priority patent/FR2593181B1/en
Priority claimed from FR8601553A external-priority patent/FR2593818B1/en
Application filed by Synthelabo SA filed Critical Synthelabo SA
Publication of AU6789587A publication Critical patent/AU6789587A/en
Application granted granted Critical
Publication of AU586065B2 publication Critical patent/AU586065B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Abstract

Compounds of general formula (I) <IMAGE> in which R1 is hydrogen or an alkyl or benzyl group and R2 is an alkyl, alkenyl, phenyl or benzyl group, or else R1 and R2 form an aliphatic chain, each of X1, X2 and X3 is hydrogen or a halogen or an alkyl, methoxy, alkylthio, methylsulphonyl, trifluoromethyl, carboxyl, cyano, nitro, amino or aminocarbonyl group, and Y is hydrogen or a halogen or a methyl, trifluoromethyl, carboxyl, cyano, amino or aminocarbonyl group. Application in therapeutics.y
AU67895/87A 1986-01-22 1987-01-21 3-(acylaminomethyl)imidazo``1,2-a`` pyridine derivatives their preparation and their application in therapy Ceased AU586065B2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR8600836A FR2593181B1 (en) 1986-01-22 1986-01-22 IMIDAZO ACYLAMINOMETHYL-3 DERIVATIVES (1,2-A) PYRIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR8600836 1986-01-22
FR8601553 1986-02-05
FR8601553A FR2593818B1 (en) 1986-02-05 1986-02-05 IMIDAZO (1,2-A) PYRIDINE ACYLAMINOMETHYL-3 DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Publications (2)

Publication Number Publication Date
AU6789587A AU6789587A (en) 1987-07-23
AU586065B2 true AU586065B2 (en) 1989-06-29

Family

ID=26224973

Family Applications (1)

Application Number Title Priority Date Filing Date
AU67895/87A Ceased AU586065B2 (en) 1986-01-22 1987-01-21 3-(acylaminomethyl)imidazo``1,2-a`` pyridine derivatives their preparation and their application in therapy

Country Status (15)

Country Link
EP (1) EP0234970B1 (en)
KR (1) KR870007174A (en)
AT (1) ATE62687T1 (en)
AU (1) AU586065B2 (en)
CA (1) CA1263390A (en)
DE (1) DE3769333D1 (en)
DK (1) DK32287A (en)
ES (1) ES2032455T3 (en)
FI (1) FI870254A (en)
GR (1) GR3002080T3 (en)
HU (1) HU196400B (en)
IL (1) IL81334A (en)
NO (1) NO165802C (en)
NZ (1) NZ219006A (en)
PT (1) PT84161B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0289371B1 (en) * 1987-03-27 1991-09-25 Synthelabo Imidazopyridine derivatives, their preparation and therapeutical use
FR2615513B1 (en) * 1987-05-21 1989-07-13 Synthelabo DERIVATIVES OF ACYLAMINOMETHYL-3 TETRAHYDRO-5,6,7,8 IMIDAZO (1,2-A) PYRIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
DE4405378A1 (en) * 1994-02-19 1995-08-24 Merck Patent Gmbh Adhesion receptor antagonists
US6596731B2 (en) 2001-03-27 2003-07-22 Hoffmann-La Roche Inc. Substituted imidazo[1,2-A] pyridine derivatives
WO2006051063A1 (en) * 2004-11-11 2006-05-18 Ferrer Internacional S. A. Imidazo[1,2-a]pyridine compounds, compositions, uses and methods related thereto
WO2009143156A2 (en) * 2008-05-19 2009-11-26 Sepracor Inc. IMIDAZO[1,2-a]PYRIDINE COMPOUNDS

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU7477287A (en) * 1986-06-27 1988-01-07 Synthelabo Imidazo pyridines
AU575190B2 (en) * 1984-08-07 1988-07-21 Synthelabo 3-acylaminomethylimidazo (1,2-a) pyridine

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB991589A (en) * 1963-04-30 1965-05-12 Selvi & C Lab Bioterapico Novel [1,2-ª‡]imidazopyridines and a process for the manufacture thereof
US3408496A (en) * 1964-11-23 1968-10-29 Parametrics Inc Alpha ray excited composition analysis
ZA81219B (en) * 1980-01-23 1982-01-27 Schering Corp Imidazo (1,2-a) pyridines ,process for their preparation and pharmaceutical compositions containing them
FR2492382A1 (en) * 1980-10-22 1982-04-23 Synthelabo IMIDAZO (1,2-A) PYRIDINE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC USE THEREOF

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU575190B2 (en) * 1984-08-07 1988-07-21 Synthelabo 3-acylaminomethylimidazo (1,2-a) pyridine
AU7477287A (en) * 1986-06-27 1988-01-07 Synthelabo Imidazo pyridines

Also Published As

Publication number Publication date
FI870254A (en) 1987-07-23
DE3769333D1 (en) 1991-05-23
ES2032455T3 (en) 1993-02-16
EP0234970A1 (en) 1987-09-02
DK32287A (en) 1987-07-23
AU6789587A (en) 1987-07-23
CA1263390A (en) 1989-11-28
NO165802C (en) 1991-04-10
DK32287D0 (en) 1987-01-21
ATE62687T1 (en) 1991-05-15
GR3002080T3 (en) 1992-12-30
NO165802B (en) 1991-01-02
PT84161B (en) 1989-07-31
HUT43064A (en) 1987-09-28
FI870254A0 (en) 1987-01-21
HU196400B (en) 1988-11-28
NO870251D0 (en) 1987-01-21
IL81334A (en) 1991-01-31
NO870251L (en) 1987-07-23
NZ219006A (en) 1989-05-29
EP0234970B1 (en) 1991-04-17
KR870007174A (en) 1987-08-17
IL81334A0 (en) 1987-08-31
PT84161A (en) 1987-02-01

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