NO145576C - Analogifremgangsmaate ved fremstilling av terapeutisk aktive penicillinderivater - Google Patents

Analogifremgangsmaate ved fremstilling av terapeutisk aktive penicillinderivater

Info

Publication number
NO145576C
NO145576C NO741227A NO741227A NO145576C NO 145576 C NO145576 C NO 145576C NO 741227 A NO741227 A NO 741227A NO 741227 A NO741227 A NO 741227A NO 145576 C NO145576 C NO 145576C
Authority
NO
Norway
Prior art keywords
preparation
therapeutically active
penicillin derivatives
analogy procedure
active penicillin
Prior art date
Application number
NO741227A
Other languages
English (en)
Norwegian (no)
Other versions
NO145576B (no
NO741227L (no
Inventor
Hisao Tobiki
Hirotada Yamada
Kozo Shimago
Iwao Nakatsuka
Takenari Nakagome
Norihiko Tanno
Original Assignee
Sumitomo Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Co filed Critical Sumitomo Chemical Co
Publication of NO741227L publication Critical patent/NO741227L/no
Publication of NO145576B publication Critical patent/NO145576B/no
Publication of NO145576C publication Critical patent/NO145576C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO741227A 1973-04-05 1974-04-04 Analogifremgangsmaate ved fremstilling av terapeutisk aktive penicillinderivater NO145576C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP48039358A JPS5751837B2 (es) 1973-04-05 1973-04-05

Publications (3)

Publication Number Publication Date
NO741227L NO741227L (no) 1974-10-08
NO145576B NO145576B (no) 1982-01-11
NO145576C true NO145576C (no) 1982-04-21

Family

ID=12550837

Family Applications (1)

Application Number Title Priority Date Filing Date
NO741227A NO145576C (no) 1973-04-05 1974-04-04 Analogifremgangsmaate ved fremstilling av terapeutisk aktive penicillinderivater

Country Status (16)

Country Link
US (1) US3945995A (es)
JP (1) JPS5751837B2 (es)
AR (1) AR202297A1 (es)
BE (1) BE813356A (es)
CA (1) CA1026749A (es)
CH (1) CH594681A5 (es)
DD (1) DD110502A5 (es)
DE (1) DE2416449C2 (es)
DK (1) DK145157C (es)
FR (1) FR2224132B1 (es)
GB (1) GB1470188A (es)
HU (1) HU168314B (es)
NL (1) NL7404679A (es)
NO (1) NO145576C (es)
SE (2) SE422942B (es)
ZA (1) ZA742186B (es)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1074784A (en) * 1974-09-06 1980-04-01 Sumitomo Chemical Company N-ACYLAMINO-.alpha.-ARYLACETAMIDO CEPHALOSPORINS
FR2288521A1 (fr) * 1974-10-25 1976-05-21 Merck Patent Gmbh Nouvelles penicillines et procede pour leur preparation
DE2525541C2 (de) * 1975-06-07 1984-01-12 Bayer Ag, 5090 Leverkusen β-Lactam-Antibiotica, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel
JPS5195090A (en) * 1975-02-14 1976-08-20 66 * dd22 * 33 hidorokishipiridajin 44 karubokishiamido * 22 * paraahidorokishifueniru * asetoamido * penishiransanno seiho
US4111932A (en) * 1975-09-08 1978-09-05 Mitsubishi Chemical Industries Limited Amino acid derivatives of 6-(2-amino-2-arylacetamido)penicillanic acids
US4053609A (en) * 1975-09-12 1977-10-11 Tanabe Seiyaku Co., Ltd. Penicillins and processes for preparing the same
GB1568962A (en) * 1975-10-31 1980-06-11 Beecham Group Ltd Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
JPS5285143A (en) * 1976-01-05 1977-07-15 Takeda Chem Ind Ltd Antimicrobial agents and method of preparing same
NZ184434A (en) * 1976-06-30 1979-03-28 Dainippon Pharmaceutical Co Penicillins with a substituted p-hydroxy-benzyl side-chain, and injectable pharmaceutical compositions
JPS5346997A (en) * 1976-10-06 1978-04-27 Bristol Myers Co Antiibacterial agent
US4081441A (en) * 1976-10-06 1978-03-28 Bristol-Myers Company Antibacterial agents
JPS53124295A (en) * 1977-04-04 1978-10-30 Mitsubishi Chem Ind Ltd Penicillin derivatives
EP0001041A3 (en) * 1977-07-27 1979-06-27 Sandoz Ag Alpha(pyridonecarboxylamino)-alpha substituted acetamido penicillins and -cephalosporins, process for their preparation, their use in pharmaceuticals; pyridones used in the process
US4198504A (en) * 1978-11-02 1980-04-15 Bristol-Myers Company [3-(Pyridinium)-7-(naphthyiridinyl carbonylamino)acetamido]cephalosporanic acid derivatives
JPS5573686A (en) * 1978-11-28 1980-06-03 Mitsui Toatsu Chem Inc Novel penicillin
US4231928A (en) * 1979-04-24 1980-11-04 Bristol-Myers Company Antibacterial agents
US4241062A (en) * 1979-05-29 1980-12-23 Merck & Co., Inc. Antibacterial penicillins
JPS5651488A (en) * 1979-10-02 1981-05-09 Meiji Seika Kaisha Ltd Penicillin derivative and its preparation
JPS5665874A (en) * 1979-11-01 1981-06-03 Mitsui Toatsu Chem Inc Novel quinoline derivative
US4288590A (en) * 1980-02-14 1981-09-08 Bristol-Myers Company 7-[Dα-(4-Hydroxy-1,5-naphthyridine-3-carboxamido)-α-arylacetamido]-3-(N,N-dimethyl-aminomethylpyridinium) methyl-3-cephem-4-carboxylates
IT1215277B (it) * 1985-05-27 1990-01-31 Pomezia Roma A Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi.
DE4102234A1 (de) * 1991-01-23 1992-07-30 Dresden Arzneimittel Neue (alpha)-aminochinolinoyl-(3)-penicilline, verfahren zu deren herstellung und diese enthaltende antibakterielle mittel
WO1993008196A1 (en) * 1991-10-15 1993-04-29 Fujisawa Pharmaceutical Co., Ltd. Penicillin g ester
AU1532802A (en) * 2000-10-12 2002-04-22 Merck & Co Inc Aza- and polyaza-naphthalenyl-carboxamides useful as hiv integrase inhibitors
SK4322003A3 (en) * 2000-10-12 2003-09-11 Merck & Co Inc Aza- and polyaza-naphthalenyl carboxamides useful as HIV integrase inhibitors
JP2004517860A (ja) * 2000-10-12 2004-06-17 メルク エンド カムパニー インコーポレーテッド Hivインテグラーゼ阻害薬として有用なアザ−およびポリアザ−ナフタレニルカルボキサミド類
JP4494020B2 (ja) 2002-03-15 2010-06-30 メルク・シャープ・エンド・ドーム・コーポレイション Hivインテグラーゼ阻害剤として有用なn−(置換ベンジル)−8−ヒドロキシ−1,6−ナフチリジン−7−カルボキサミド
AU2005279050A1 (en) * 2004-07-30 2006-03-09 Centre National De La Recherche Scientifique (Cnrs) Hybrid molecules QA where Q is an aminoquinoline and A is an antibiotic residue, and the synthesis and uses thereof as antibacterial agents

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3248387A (en) * 1963-02-07 1966-04-26 American Home Prod Amino-acylamino-penicillanic acids
GB1053415A (es) * 1964-07-29
GB1130445A (en) * 1966-04-26 1968-10-16 Beecham Group Ltd Penicillins
DE2104580C3 (de) * 1971-02-01 1981-04-02 Bayer Ag, 5090 Leverkusen Acylureidopenicilline
DE2165462C2 (de) * 1971-12-29 1984-12-13 Sumitomo Chemical Co., Ltd., Osaka Penicilline, Verfahren zu ihrer Herstellung und sie enthaltende Arzneimittel
AR204162A1 (es) * 1972-05-08 1975-11-28 Yamanouchi Pharma Co Ltd Proceso para la preparacion de derivados de ampicilina
JPS5417754B2 (es) * 1972-12-15 1979-07-02

Also Published As

Publication number Publication date
DE2416449A1 (de) 1974-10-24
NO145576B (no) 1982-01-11
DK145157B (da) 1982-09-20
AU6761374A (en) 1975-10-09
AR202297A1 (es) 1975-05-30
DE2416449C2 (de) 1982-10-07
SE422943B (sv) 1982-04-05
HU168314B (es) 1976-03-28
DD110502A5 (es) 1974-12-20
CH594681A5 (es) 1978-01-31
GB1470188A (en) 1977-04-14
ZA742186B (en) 1975-05-28
SE422942B (sv) 1982-04-05
CA1026749A (en) 1978-02-21
US3945995A (en) 1976-03-23
SE7701836L (sv) 1977-02-18
NO741227L (no) 1974-10-08
DK145157C (da) 1983-04-11
FR2224132A1 (es) 1974-10-31
BE813356A (fr) 1974-10-07
NL7404679A (es) 1974-10-08
FR2224132B1 (es) 1977-05-06
JPS49125387A (es) 1974-11-30
JPS5751837B2 (es) 1982-11-04

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