NO142865C - ANALOGY PROCEDURE FOR THE PREPARATION OF NEW THERAPEUTIC ACTIVE CARBZOLS - Google Patents

ANALOGY PROCEDURE FOR THE PREPARATION OF NEW THERAPEUTIC ACTIVE CARBZOLS

Info

Publication number
NO142865C
NO142865C NO2975/73A NO297573A NO142865C NO 142865 C NO142865 C NO 142865C NO 2975/73 A NO2975/73 A NO 2975/73A NO 297573 A NO297573 A NO 297573A NO 142865 C NO142865 C NO 142865C
Authority
NO
Norway
Prior art keywords
carbzols
preparation
new therapeutic
therapeutic active
analogy procedure
Prior art date
Application number
NO2975/73A
Other languages
Norwegian (no)
Other versions
NO142865B (en
Inventor
Leo Berger
Alfred John Corraz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO142865B publication Critical patent/NO142865B/en
Publication of NO142865C publication Critical patent/NO142865C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • C07D209/82Carbazoles; Hydrogenated carbazoles
    • C07D209/88Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • C07D209/82Carbazoles; Hydrogenated carbazoles
    • C07D209/86Carbazoles; Hydrogenated carbazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO2975/73A 1972-07-24 1973-07-23 ANALOGY PROCEDURE FOR THE PREPARATION OF NEW THERAPEUTIC ACTIVE CARBZOLS NO142865C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US27414272A 1972-07-24 1972-07-24

Publications (2)

Publication Number Publication Date
NO142865B NO142865B (en) 1980-07-28
NO142865C true NO142865C (en) 1980-11-05

Family

ID=23046965

Family Applications (1)

Application Number Title Priority Date Filing Date
NO2975/73A NO142865C (en) 1972-07-24 1973-07-23 ANALOGY PROCEDURE FOR THE PREPARATION OF NEW THERAPEUTIC ACTIVE CARBZOLS

Country Status (26)

Country Link
JP (1) JPS5740144B2 (en)
KR (1) KR780000289B1 (en)
AR (1) AR205331A1 (en)
AT (1) AT325607B (en)
AU (1) AU475534B2 (en)
BE (1) BE802596A (en)
CA (1) CA1026348A (en)
CH (1) CH587819A5 (en)
DD (1) DD107681A5 (en)
DE (1) DE2337340C2 (en)
DK (1) DK138537B (en)
FI (1) FI59244C (en)
FR (1) FR2193611B1 (en)
GB (1) GB1385620A (en)
HK (1) HK49878A (en)
HU (1) HU167611B (en)
IE (1) IE37942B1 (en)
IL (1) IL42799A (en)
KE (1) KE2847A (en)
LU (1) LU68071A1 (en)
MY (1) MY7800315A (en)
NL (1) NL169877C (en)
NO (1) NO142865C (en)
SE (2) SE402283B (en)
SU (1) SU509220A3 (en)
ZA (1) ZA734047B (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4146542A (en) * 1978-06-12 1979-03-27 Hoffmann-La Roche Inc. Dihydrocarbazole acetic acid and esters thereof
US4150031A (en) * 1978-06-26 1979-04-17 Hoffmann-La Roche Inc. Hydroxy methyl carbazole acetic acid and esters
US4158007A (en) * 1978-08-21 1979-06-12 Hoffmann-La Roche Inc. Carbazole methyl malonates
US4501908A (en) * 1981-03-12 1985-02-26 Hoffmann-La Roche Inc. 2,3-Isopropylidene ribonic acid, 1,4-lactones
JPS6040256U (en) * 1983-08-25 1985-03-20 伊東 璋 Container cleaning machine
ATE61047T1 (en) * 1986-01-23 1991-03-15 Merck Frosst Canada Inc TETRAHYDROCARBAZOLE-1-ALKANOIC ACIDS.
EP0239306B1 (en) 1986-03-27 1993-06-02 Merck Frosst Canada Inc. Tetrahydrocarbazole esters
EP0307077A1 (en) * 1987-07-21 1989-03-15 Merck Frosst Canada Inc. Tetrahydrocarbazoles for the improvement of cyclosporin therapy
CA1326030C (en) * 1987-07-21 1994-01-11 John W. Gillard Cyclohept[b]indolealkanoic acids
PT95692A (en) * 1989-10-27 1991-09-13 American Home Prod PROCESS FOR THE PREPARATION OF INDOLE-, INDENO-, PYRANOINDOLE- AND TETRA-HYDROCARBAZOLE-ALCANOIC ACID DERIVATIVES, OR WHICH ARE USEFUL AS PLA2 INHIBITORS AND LIPOXIGENASE
JP2004010601A (en) * 2002-06-11 2004-01-15 Nippon Steel Chem Co Ltd Method for producing indole derivative and intermediate useful for the same
AU2004206796A1 (en) * 2003-01-14 2004-08-05 Merck & Co., Inc. Geminally di-substituted NSAID derivatives as Abeta 42 lowering agents
WO2005000457A2 (en) * 2003-05-06 2005-01-06 Air Products And Chemicals, Inc. Hydrogen storage reversible hydrogenated of pi-conjugated substrates
US20070069197A1 (en) * 2003-08-15 2007-03-29 Universite Laval Monomers, oligomers and polymers of 2-functionalized and 2,7-difunctionalized carbzoles
US7662831B2 (en) 2006-07-27 2010-02-16 Wyeth Llc Tetracyclic indoles as potassium channel modulators
US9447040B2 (en) * 2011-11-15 2016-09-20 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. Tricyclic compounds, compositions comprising them and uses thereof
JP5940036B2 (en) * 2013-10-08 2016-06-29 テックフィールズ バイオケム カンパニー リミテッド Positively charged water-soluble prodrugs of aryl- and heteroarylpropionic acids with very fast skin permeability
WO2021193708A1 (en) * 2020-03-25 2021-09-30 Jnc株式会社 Compound, liquid crystal composition, and liquid crystal display element

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD70880A (en) *
US3580926A (en) * 1969-11-10 1971-05-25 Parke Davis & Co Carbazole-4-alkanoic acids and tetrahydrocarbazole-4-alkanoic acids
ZA715217B (en) * 1970-08-20 1972-04-26 Org Nv Anti-inflammatory preparations

Also Published As

Publication number Publication date
FI59244C (en) 1981-07-10
FR2193611B1 (en) 1976-05-14
IL42799A (en) 1977-03-31
KR780000289B1 (en) 1978-08-10
IE37942L (en) 1974-01-24
LU68071A1 (en) 1975-04-11
SE402283B (en) 1978-06-26
JPS4943973A (en) 1974-04-25
CA1026348A (en) 1978-02-14
KE2847A (en) 1978-06-30
JPS5740144B2 (en) 1982-08-25
CH587819A5 (en) 1977-05-13
AR205331A1 (en) 1976-04-30
HU167611B (en) 1975-11-28
IE37942B1 (en) 1977-11-23
DK138537B (en) 1978-09-25
DD107681A5 (en) 1974-08-12
AT325607B (en) 1975-10-27
NL169877C (en) 1982-09-01
HK49878A (en) 1978-09-08
DK138537C (en) 1979-03-05
FI59244B (en) 1981-03-31
IL42799A0 (en) 1973-10-25
NL169877B (en) 1982-04-01
GB1385620A (en) 1975-02-26
NO142865B (en) 1980-07-28
BE802596A (en) 1974-01-21
AU475534B2 (en) 1976-08-26
SE7605813L (en) 1976-05-21
SU509220A3 (en) 1976-03-30
NL7310275A (en) 1974-01-28
MY7800315A (en) 1978-12-31
ATA649773A (en) 1975-01-15
AU5839073A (en) 1975-01-23
DE2337340C2 (en) 1985-05-02
FR2193611A1 (en) 1974-02-22
ZA734047B (en) 1974-03-27
DE2337340A1 (en) 1974-02-14

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