NL6504085A - - Google Patents

Info

Publication number
NL6504085A
NL6504085A NL6504085A NL6504085A NL6504085A NL 6504085 A NL6504085 A NL 6504085A NL 6504085 A NL6504085 A NL 6504085A NL 6504085 A NL6504085 A NL 6504085A NL 6504085 A NL6504085 A NL 6504085A
Authority
NL
Netherlands
Application number
NL6504085A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to BE663693D priority Critical patent/BE663693A/fr
Priority to NL123139D priority patent/NL123139C/xx
Priority to FR940266A priority patent/FR3761M/fr
Application filed filed Critical
Publication of NL6504085A publication Critical patent/NL6504085A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NL6504085A 1962-07-04 1965-03-31 NL6504085A (cs)

Priority Applications (3)

Application Number Priority Date Filing Date Title
BE663693D BE663693A (cs) 1965-03-31
NL123139D NL123139C (cs) 1965-03-31
FR940266A FR3761M (fr) 1962-07-04 1963-07-03 Nouvelles dihydrothiéno-[3,4-d]-pyrimidines.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DET0022407 1962-07-04

Publications (1)

Publication Number Publication Date
NL6504085A true NL6504085A (cs) 1966-10-03

Family

ID=7550528

Family Applications (1)

Application Number Title Priority Date Filing Date
NL6504085A NL6504085A (cs) 1962-07-04 1965-03-31

Country Status (5)

Country Link
US (3) US3272811A (cs)
DE (1) DE1470336A1 (cs)
ES (1) ES301102A1 (cs)
GB (1) GB1048986A (cs)
NL (1) NL6504085A (cs)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3931204A (en) * 1971-07-13 1976-01-06 U.C.B. Societe Anonyme Thieno[3,4-d]pyrimidines
US3960860A (en) * 1973-01-08 1976-06-01 International Flavors & Fragrances Inc. 2-Methyl-5,7-dihydrothieno-[3,4d]-pyrimidine
US4287340A (en) * 1979-08-27 1981-09-01 Warner-Lambert Company Dihydro-oxo-pyrido[1,2-a]thienopyrimidine compounds
NL8300656A (nl) * 1982-02-25 1983-09-16 Maruko Pharmaceutical Co Thiopyranopyrimidineverbindingen en zuuradditiezouten daarvan.
DE3335472A1 (de) * 1983-09-30 1985-04-11 Gödecke AG, 1000 Berlin 5h-(1)benzopyrano-(2,3,-d)pyrimidin-derivate, verfahren zu deren herstellung sowie deren verwendung bei der bekaempfung von gastralen und duodenalen schleimhautlaesionen
DE3335473A1 (de) * 1983-09-30 1985-04-11 Gödecke AG, 1000 Berlin 4-thioxo-benzopyrano(2,3-d)pyrimidin-derivate sowie verfahren zu deren herstellung
US4670560A (en) * 1986-04-28 1987-06-02 Ortho Pharmaceutical Corporation Thienopyrimidine-2,4-dione derivatives and intermediates thereof
US4725599A (en) * 1986-09-08 1988-02-16 Pfizer Inc. Heterocyclic ring fused pyrimidine-4 (3H)-ones as anticoccidial agents
US4797486A (en) * 1986-09-08 1989-01-10 Pfizer Inc. Heterocyclic ring fused pyrimidine-4(3H)-ones as anticoccidial agents
EP0276057B1 (en) * 1987-01-21 1994-03-09 Merck & Co. Inc. Piperazinylpyrimidines as beta-adrenergic receptor blocking agents
US4871739A (en) * 1987-01-21 1989-10-03 Merck & Co., Inc. Substituted 6H-7,8-dihydrothiapyrano(3,2-D)-pyrimidines as hyopglycemic agents
US4889856A (en) * 1987-08-31 1989-12-26 Merck & Co., Inc. 7,8-dihydro-4-(1-pierazinyl)-6H-thiopyrano-[3,2-d] pyrimidines as β-blockers
US4994464A (en) * 1987-08-31 1991-02-19 Merck & Co., Inc. Piperazinylpyrimidines as β-adrenergic receptor blockers
US6232320B1 (en) * 1998-06-04 2001-05-15 Abbott Laboratories Cell adhesion-inhibiting antiinflammatory compounds
JP4497340B2 (ja) * 1998-08-27 2010-07-07 大日本住友製薬株式会社 ピリミジン誘導体
WO2000042025A1 (fr) * 1999-01-14 2000-07-20 Meiji Seika Kaisha, Ltd. Inhibiteurs de poly(adp-ribose) polymerase consistant en des derives de pyrimidine
NZ545717A (en) 2003-08-05 2009-12-24 Vertex Pharma Hydrogenated quinazoline derivatives as inhibitors of voltage-gated ion channels
TW200621257A (en) * 2004-10-20 2006-07-01 Astellas Pharma Inc Pyrimidine derivative fused with nonaromatic ring
ES2328400T3 (es) * 2005-04-21 2009-11-12 Boehringer Ingelheim International Gmbh Dihidrotienopirimidinas para el tratamiento de enfermedades inflamatorias.
EP1847543A1 (de) * 2006-04-19 2007-10-24 Boehringer Ingelheim Pharma GmbH & Co. KG Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen
CN103497201A (zh) * 2007-10-18 2014-01-08 贝林格尔.英格海姆国际有限公司 二氢噻吩并[3,2-d]嘧啶的制备中使用的中间体及其制备
DK2215092T3 (da) 2007-10-19 2012-05-07 Boehringer Ingelheim Int Substitueret piperidino-dihydrothienopyrimidin
CA2702524A1 (en) 2007-10-19 2009-04-23 Boehringer Ingelheim International Gmbh Heterocycle-substituted piperazino-dihydrothienopyrimidines
ATE537175T1 (de) 2007-10-19 2011-12-15 Boehringer Ingelheim Int Neue piperazino-dihydrothienopyrimidin-derivate
ME01465B (me) * 2008-05-13 2014-04-20 Boehringer Ingelheim Int Sinteza dihidrotieno[3 ,2-d]pirimidin diola i sličnih pirimidin diola
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma
US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
WO2014124860A1 (en) 2013-02-14 2014-08-21 Boehringer Ingelheim International Gmbh Specific pde4b-inhibitors for the treatment of diabetes mellitus
CN116925099B (zh) * 2023-07-21 2025-06-03 厦门大学 手性二氢噻吩并嘧啶亚砜的制备方法及其应用与其2、4位取代化合物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB617435A (en) * 1945-08-10 1949-02-07 Lederle Lab Inc Improvements in or relating to tetrahydro thieno uracils and method of preparing same
US2792394A (en) * 1954-01-25 1957-05-14 Phillips Petroleum Co Preparation of sulfenyl dithiocarbamates
NL226623A (cs) * 1954-10-05
US2937118A (en) * 1956-06-27 1960-05-17 Raschig Gmbh Dr F Aminopyridine compositions
US3063902A (en) * 1961-01-18 1962-11-13 Irwin Neisler & Co Analgesic aralkyl-pyridines
US3244594A (en) * 1962-01-12 1966-04-05 Egyt Gyogyszervegyeszeti Gyar 1, 6-bis-(beta-chloro-ethyl-amino)-1, 6-deoxy-d-mannitol heparinate

Also Published As

Publication number Publication date
US3318881A (en) 1967-05-09
US3318883A (en) 1967-05-09
ES301102A1 (es) 1965-01-16
DE1470336A1 (de) 1969-03-20
US3272811A (en) 1966-09-13
GB1048986A (en) 1966-11-23

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