NL167697C - PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION ACTING ON THE CENTRAL NERVOUS SYSTEM BASED ON 5-PHENYLBENZODIAZEPINE DERIVATIVES, AND METHOD FOR PREPARING 5-PHENYLBODODIA ZEPARIC THESE BEFORE USE THEREFORE - Google Patents

PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION ACTING ON THE CENTRAL NERVOUS SYSTEM BASED ON 5-PHENYLBENZODIAZEPINE DERIVATIVES, AND METHOD FOR PREPARING 5-PHENYLBODODIA ZEPARIC THESE BEFORE USE THEREFORE

Info

Publication number
NL167697C
NL167697C NL7016848A NL7016848A NL167697C NL 167697 C NL167697 C NL 167697C NL 7016848 A NL7016848 A NL 7016848A NL 7016848 A NL7016848 A NL 7016848A NL 167697 C NL167697 C NL 167697C
Authority
NL
Netherlands
Prior art keywords
preparation
zeparic
phenylbododia
phenylbenzodiazepine
derivatives
Prior art date
Application number
NL7016848A
Other languages
Dutch (nl)
Other versions
NL167697B (en
NL7016848A (en
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of NL7016848A publication Critical patent/NL7016848A/xx
Publication of NL167697B publication Critical patent/NL167697B/en
Application granted granted Critical
Publication of NL167697C publication Critical patent/NL167697C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NL7016848A 1969-11-18 1970-11-17 PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION ACTING ON THE CENTRAL NERVOUS SYSTEM BASED ON 5-PHENYLBENZODIAZEPINE DERIVATIVES, AND METHOD FOR PREPARING 5-PHENYLBODODIA ZEPARIC THESE BEFORE USE THEREFORE NL167697C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP44092366A JPS4910958B1 (en) 1969-11-18 1969-11-18

Publications (3)

Publication Number Publication Date
NL7016848A NL7016848A (en) 1971-05-21
NL167697B NL167697B (en) 1981-08-17
NL167697C true NL167697C (en) 1982-01-18

Family

ID=14052400

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7016848A NL167697C (en) 1969-11-18 1970-11-17 PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION ACTING ON THE CENTRAL NERVOUS SYSTEM BASED ON 5-PHENYLBENZODIAZEPINE DERIVATIVES, AND METHOD FOR PREPARING 5-PHENYLBODODIA ZEPARIC THESE BEFORE USE THEREFORE

Country Status (15)

Country Link
JP (2) JPS5010659B1 (en)
AT (2) AT300816B (en)
BE (1) BE759099A (en)
CH (2) CH549588A (en)
DE (2) DE2064926A1 (en)
DK (1) DK141846B (en)
ES (1) ES385641A1 (en)
FI (1) FI51701C (en)
FR (1) FR2073379B1 (en)
GB (2) GB1337737A (en)
NL (1) NL167697C (en)
NO (1) NO126085B (en)
SE (1) SE363111B (en)
YU (1) YU34898B (en)
ZA (1) ZA707644B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA713364B (en) * 1970-06-18 1972-01-26 Upjohn Co Prganic compounds and process
JPS494470B1 (en) * 1970-08-26 1974-02-01
CH545302A (en) * 1971-04-08 1974-01-13 Ciba Geigy Ag Triazolobenzodiazepine derivs - with anticonvulsant, cns depressant and muscle-relaxant activity
US3751426A (en) * 1971-04-28 1973-08-07 Upjohn Co 1-substituted-6-phenyl-4h-s-triazolo(4,3-a)(1,6)benzodiazepine compounds
GB1377230A (en) * 1971-09-13 1974-12-11 Upjohn Co 4h-s-triazolo -4,3-a- 1,4-benzodiazepines
BE790356A (en) * 1971-10-21 1973-04-20 Takeda Chemical Industries Ltd BENZODIAZEPINE DERIVATIVES
JPS5418280B2 (en) * 1971-10-30 1979-07-06
BE793629A (en) * 1972-01-03 1973-07-03 Upjohn Co NEW BENZODIAZEPINE DERIVATIVES AND THEIR PREPARATION
DE3021107A1 (en) * 1980-06-04 1981-12-17 Hoechst Ag, 6000 Frankfurt CARBAMOYLOXYAMINO-1,4-BENZODIAZEPINE, METHOD FOR IRER PRODUCTION AND MEDICINAL PRODUCTS CONTAINING THE SAME
CA1211437A (en) * 1981-08-12 1986-09-16 Rene Borer Benzazepines
CN111533745A (en) * 2020-05-20 2020-08-14 成都药明康德新药开发有限公司 Process for preparing tert-butyl-3- (aminomethyl) dihydro-5H-triazolodiazepine-8 (9H) -carboxylic acid ester

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI50981C (en) * 1968-11-05 1976-09-10 Takeda Chemical Industries Ltd Process for the preparation of s-triat solo- (4,3-a) (1,4) -benzodiazepines acting as hypnotics and sedatives.
US3987052A (en) * 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines

Also Published As

Publication number Publication date
AT300816B (en) 1972-08-10
ES385641A1 (en) 1973-10-01
DK141846B (en) 1980-06-30
NO126085B (en) 1972-12-18
FR2073379A1 (en) 1971-10-01
FR2073379B1 (en) 1974-08-23
FI51701C (en) 1977-03-10
CH551432A (en) 1974-07-15
JPS5010659B1 (en) 1975-04-23
SE363111B (en) 1974-01-07
BE759099A (en) 1971-04-30
YU282770A (en) 1979-10-31
NL167697B (en) 1981-08-17
ZA707644B (en) 1971-08-25
NL7016848A (en) 1971-05-21
GB1337737A (en) 1973-11-21
CH549588A (en) 1974-05-31
FI51701B (en) 1976-11-30
AT311993B (en) 1973-12-10
JPS4910958B1 (en) 1974-03-13
DK141846C (en) 1980-11-24
DE2064926A1 (en) 1971-07-22
YU34898B (en) 1980-04-30
GB1337736A (en) 1973-11-21
DE2056174A1 (en) 1971-06-24

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Legal Events

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V1 Lapsed because of non-payment of the annual fee