NL162081B - PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION WITH ANTIBACTERIAL PROPERTIES, FORMED PREPARATION AND PROCESS FOR THE PREPARATION OF AN ACTIVE SUBSTANCE SUITABLE FOR USE IN THE FIRST METHOD. - Google Patents

PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION WITH ANTIBACTERIAL PROPERTIES, FORMED PREPARATION AND PROCESS FOR THE PREPARATION OF AN ACTIVE SUBSTANCE SUITABLE FOR USE IN THE FIRST METHOD.

Info

Publication number
NL162081B
NL162081B NL7512465.A NL7512465A NL162081B NL 162081 B NL162081 B NL 162081B NL 7512465 A NL7512465 A NL 7512465A NL 162081 B NL162081 B NL 162081B
Authority
NL
Netherlands
Prior art keywords
preparation
active substance
antibacterial properties
substance suitable
pharmaceutical
Prior art date
Application number
NL7512465.A
Other languages
Dutch (nl)
Other versions
NL7512465A (en
NL162081C (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NL7512465A publication Critical patent/NL7512465A/en
Publication of NL162081B publication Critical patent/NL162081B/en
Application granted granted Critical
Publication of NL162081C publication Critical patent/NL162081C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/088Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/228Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to adjacent ring-carbon atoms of the cyclohexane rings
    • C07H15/23Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to adjacent ring-carbon atoms of the cyclohexane rings with only two saccharide radicals in the molecule, e.g. ambutyrosin, butyrosin, xylostatin, ribostamycin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NL7512465.A 1974-10-26 1975-10-24 PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION WITH ANTIBACTERIAL PROPERTIES, FORMED PREPARATION AND PROCESS FOR THE PREPARATION OF AN ACTIVE SUBSTANCE SUITABLE FOR USE IN THE FOREGOING PROCESS NL162081C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4641274A GB1464401A (en) 1974-10-26 1974-10-26 Aminoglycosides

Publications (3)

Publication Number Publication Date
NL7512465A NL7512465A (en) 1976-04-28
NL162081B true NL162081B (en) 1979-11-15
NL162081C NL162081C (en) 1980-04-15

Family

ID=10441164

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7512465.A NL162081C (en) 1974-10-26 1975-10-24 PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION WITH ANTIBACTERIAL PROPERTIES, FORMED PREPARATION AND PROCESS FOR THE PREPARATION OF AN ACTIVE SUBSTANCE SUITABLE FOR USE IN THE FOREGOING PROCESS

Country Status (28)

Country Link
JP (1) JPS5519237B2 (en)
AR (1) AR205593A1 (en)
AT (1) AT340051B (en)
BE (1) BE834864A (en)
BG (1) BG24821A3 (en)
CA (1) CA1039275A (en)
CH (1) CH601339A5 (en)
CS (1) CS195712B2 (en)
DD (1) DD122522A5 (en)
DE (1) DE2547738C3 (en)
DK (1) DK147075C (en)
EG (1) EG11975A (en)
ES (1) ES442051A1 (en)
FI (1) FI752951A (en)
FR (1) FR2289202A1 (en)
GB (1) GB1464401A (en)
HU (1) HU172060B (en)
IE (1) IE42452B1 (en)
IL (1) IL48263A (en)
LU (1) LU73644A1 (en)
NL (1) NL162081C (en)
NZ (1) NZ179050A (en)
PH (1) PH12782A (en)
PL (1) PL99933B1 (en)
RO (1) RO72878A (en)
SE (1) SE7511945L (en)
SU (1) SU617017A3 (en)
ZA (1) ZA756326B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0000473B1 (en) * 1977-06-24 1981-03-11 Scherico Ltd. Process for preparing aminoglycoside derivatives, novel derivatives obtained and pharmaceutical compositions containing such derivatives
JPS5488241A (en) * 1977-12-21 1979-07-13 Kyowa Hakko Kogyo Co Ltd Novel fortimicin a derivative
JPS57118475U (en) * 1981-01-14 1982-07-22

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH606076A5 (en) * 1973-08-06 1978-10-13 Scherico Ltd

Also Published As

Publication number Publication date
AR205593A1 (en) 1976-05-14
BG24821A3 (en) 1978-05-12
BE834864A (en) 1976-04-26
IL48263A0 (en) 1975-12-31
JPS5168543A (en) 1976-06-14
FR2289202B1 (en) 1978-11-10
IE42452L (en) 1976-04-26
IL48263A (en) 1978-03-10
RO72878B (en) 1983-06-30
ATA809575A (en) 1977-03-15
ZA756326B (en) 1976-09-29
SE7511945L (en) 1976-04-27
ES442051A1 (en) 1977-04-01
DK147075B (en) 1984-04-02
DE2547738C3 (en) 1978-08-03
JPS5519237B2 (en) 1980-05-24
AT340051B (en) 1977-11-25
HU172060B (en) 1978-05-28
EG11975A (en) 1978-06-30
CH601339A5 (en) 1978-07-14
GB1464401A (en) 1977-02-16
DK481175A (en) 1976-04-27
PH12782A (en) 1979-08-17
NL7512465A (en) 1976-04-28
LU73644A1 (en) 1977-05-31
RO72878A (en) 1983-07-07
DE2547738B2 (en) 1977-12-01
CS195712B2 (en) 1980-02-29
AU8598175A (en) 1976-12-09
PL99933B1 (en) 1978-08-31
DE2547738A1 (en) 1976-05-06
FR2289202A1 (en) 1976-05-28
NL162081C (en) 1980-04-15
FI752951A (en) 1976-04-27
DD122522A5 (en) 1976-10-12
IE42452B1 (en) 1980-08-13
SU617017A3 (en) 1978-07-25
NZ179050A (en) 1978-03-06
DK147075C (en) 1984-11-05
CA1039275A (en) 1978-09-26

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