MY139848A - Pyrazole derivatives for the inhibition of cdk's and gsk's - Google Patents

Pyrazole derivatives for the inhibition of cdk's and gsk's

Info

Publication number
MY139848A
MY139848A MYPI20060218A MY139848A MY 139848 A MY139848 A MY 139848A MY PI20060218 A MYPI20060218 A MY PI20060218A MY 139848 A MY139848 A MY 139848A
Authority
MY
Malaysia
Prior art keywords
cdk
gsk
inhibition
pyrazole derivatives
dichilorophenyl
Prior art date
Application number
Inventor
Valerio Berdini
Adrian Liam Gill
Gary Trewartha
Andrew James Woodhead
Paul Graham Wyatt
Original Assignee
Astex Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0501480A external-priority patent/GB0501480D0/en
Priority claimed from GB0501748A external-priority patent/GB0501748D0/en
Application filed by Astex Therapeutics Ltd filed Critical Astex Therapeutics Ltd
Publication of MY139848A publication Critical patent/MY139848A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

THE INVENTION PROVIDES A COMPOUND OF THE FORMULA (1): OR SALTS, TAUTOMERS, SOLVATES AND N-OXIDES THEREOF, WHEREIN: R1 IS 2,6-DICHILOROPHENYL; R2A AND R2B ARE BOTH HYDROGEN; AND R3 IS A GROUP: WHERE R4 IS CI-4 ALKYL. THE COMPOUNDS HAVE ACTIVITYAS INHIBITORS OF CDK KINASES AND INHIBIT THE PROLIFERATION OF CANCER CELLS.
MYPI20060218 2005-01-21 2006-01-18 Pyrazole derivatives for the inhibition of cdk's and gsk's MY139848A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US64621705P 2005-01-21 2005-01-21
GB0501480A GB0501480D0 (en) 2005-01-22 2005-01-22 Pharmaceutical compounds
GB0501748A GB0501748D0 (en) 2005-01-27 2005-01-27 Pharmaceutical compounds
US65133905P 2005-02-09 2005-02-09

Publications (1)

Publication Number Publication Date
MY139848A true MY139848A (en) 2009-11-30

Family

ID=45699652

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI20060218 MY139848A (en) 2005-01-21 2006-01-18 Pyrazole derivatives for the inhibition of cdk's and gsk's

Country Status (3)

Country Link
GT (3) GT200600015A (en)
MY (1) MY139848A (en)
TW (3) TW200640922A (en)

Also Published As

Publication number Publication date
GT200600014A (en) 2006-08-09
TW200639170A (en) 2006-11-16
GT200600016A (en) 2006-08-09
TW200640922A (en) 2006-12-01
GT200600015A (en) 2006-08-09
TW200637858A (en) 2006-11-01

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