GT200600014A - PHARMACEUTICAL COMPOUNDS - Google Patents

PHARMACEUTICAL COMPOUNDS

Info

Publication number
GT200600014A
GT200600014A GT200600014A GT200600014A GT200600014A GT 200600014 A GT200600014 A GT 200600014A GT 200600014 A GT200600014 A GT 200600014A GT 200600014 A GT200600014 A GT 200600014A GT 200600014 A GT200600014 A GT 200600014A
Authority
GT
Guatemala
Prior art keywords
pharmaceutical compounds
compounds
glucogeno
synthease
cycline
Prior art date
Application number
GT200600014A
Other languages
Spanish (es)
Inventor
Valerio Berdini
Adrian Liam Gill
Eva Figueroa Navarro
Michael Alistair O'brien
Theresa Rachel Phillips
Gary Trewartha
Andrew James Woodhead
Paul Graham Wyatt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0501480A external-priority patent/GB0501480D0/en
Priority claimed from GB0501748A external-priority patent/GB0501748D0/en
Application filed filed Critical
Publication of GT200600014A publication Critical patent/GT200600014A/en

Links

Abstract

LA PRESENTE INVENCION SE REFIERE A COMPUESTOS DE LA FORMULA GENERAL I EN LA QUE R1,R2A,R2B,R3, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS INHIBEN O MODULAN LA ACTIVIDAD DE QUINASAS DEPENDIENTE DE CICLINA (CDK) Y QUINASA GLUCOGENO SINTASA (GSK) POR LO QUE SON DE UTILIDAD CONTRA EL CRECIMIENTO CELULAR ANORMAL.THE PRESENT INVENTION REFERS TO COMPOUNDS OF GENERAL FORMULA I IN WHICH R1, R2A, R2B, R3, ARE FUNCTIONAL GROUPS DESCRIBED IN THE RECORD. THESE COMPOUNDS INHIBIT OR MODULATE THE ACTIVITY OF CYCLINE-DEPENDENT KINASES (CDK) AND GLUCOGENO SYNTHEASE KINASE (GSK) SO THEY ARE USEFUL AGAINST ABNORMAL CELLULAR GROWTH.

GT200600014A 2005-01-21 2006-01-11 PHARMACEUTICAL COMPOUNDS GT200600014A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US64621705P 2005-01-21 2005-01-21
GB0501480A GB0501480D0 (en) 2005-01-22 2005-01-22 Pharmaceutical compounds
GB0501748A GB0501748D0 (en) 2005-01-27 2005-01-27 Pharmaceutical compounds
US65133905P 2005-02-09 2005-02-09

Publications (1)

Publication Number Publication Date
GT200600014A true GT200600014A (en) 2006-08-09

Family

ID=45699652

Family Applications (3)

Application Number Title Priority Date Filing Date
GT200600015A GT200600015A (en) 2005-01-21 2006-01-11 PHARMACEUTICAL COMPOUNDS
GT200600014A GT200600014A (en) 2005-01-21 2006-01-11 PHARMACEUTICAL COMPOUNDS
GT200600016A GT200600016A (en) 2005-01-21 2006-01-11 PHARMACEUTICAL COMPOUNDS

Family Applications Before (1)

Application Number Title Priority Date Filing Date
GT200600015A GT200600015A (en) 2005-01-21 2006-01-11 PHARMACEUTICAL COMPOUNDS

Family Applications After (1)

Application Number Title Priority Date Filing Date
GT200600016A GT200600016A (en) 2005-01-21 2006-01-11 PHARMACEUTICAL COMPOUNDS

Country Status (3)

Country Link
GT (3) GT200600015A (en)
MY (1) MY139848A (en)
TW (3) TW200637858A (en)

Also Published As

Publication number Publication date
TW200640922A (en) 2006-12-01
GT200600016A (en) 2006-08-09
GT200600015A (en) 2006-08-09
TW200639170A (en) 2006-11-16
TW200637858A (en) 2006-11-01
MY139848A (en) 2009-11-30

Similar Documents

Publication Publication Date Title
GT200300292A (en) PIRIMIDINE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELLULAR GROWTH
GT200600174A (en) REPLACED PIRROLOPIRIDINS, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING AND USE PROCESS
GT200600197A (en) COMPOUNDS AND COMPOSITIONS AS PROTEIN QUINASA INHIBITORS
GT200500103A (en) 4-PHENYLAMINE-QUINAZOLIN-6-IL-AMIDAS
GT200800258A (en) PIRROLO-PYRIMIDINE COMPOUNDS AND THEIR USES
GT200300087A (en) 2- (2,6-DICLOROPHENYL) -DIARYLIMIDAZOLS
NO20083669L (en) 4-aryl-2amino-pyrimidines or 4-aryl-2-aminoalkylpyrimidines as jak-2 modulators and methods of use thereof
GT200500242A (en) PROCESSES FOR THE PREPARATION OF 2- (2,6-DIOXOPIPERIDIN-3-IL) -1-SUBSTITUTED OXOISOINDOLINES
UA95244C2 (en) Compounds and methods for kinase modulation, and indications therefor
GT200500272A (en) 2-ANILINOPIRIMIDINAS REPLACED AS INHIBITORS OF THE KINASE OF THE CELL CYCLE OR THE RECEIVER OF THE THYROSINE KINASE, ITS PREPARATION AND ITS USE AS MEDICATIONS
GT200700077A (en) 4-METHYLPIRIDOPIRIMIDINONE COMPOUNDS
CR20120356A (en) NEW ACTIVE HETEROCYCLIC COMPOUNDS AS BETA-LACTAMASAS INHIBITORS
GT200300289A (en) PIRROLOPIRIMIDINE DERIVATIVES
GT200600205A (en) NEW HERBICIDES
GT200300031A (en) SUBSTITUTE INDAZOLS, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING AND USE PROCEDURE
CR20110620A (en) DERIVATIVES OF N- (HETERO) ARIL-PIRROLIDINA DE PIRAZO-4-IL-PIRROLO [2,3-D] PIRIMIDINES AND PIRROL-3-IL-PIRROLO [2,3-D] PYRIMIDINES AS IHNIBITORS OF THE JANUS KINASE
HN2010002119A (en) 2,6-DIAMINO-PYRIMIDIN-5-IL-CARBOXAMIDS AS SYK OR JAK KINASAS INHIBITORS
ATE479687T1 (en) KINASE INHIBITORS
GT200600339A (en) MACROCICLIC INHIBITORS OF HEPATITIS C VIRUS
MX2009006688A (en) Compounds and methods for kinase modulation, and indications therefor.
GT200400092A (en) PREPARATION AND USE OF RENTAL DERIVATIVES FOR THE TREATMENT OF OBESITY
GT200500218A (en) DERIVATIVES OF TRIAZOLOPIRIDINILSULFANILO AS QUINASA MAP P38 INHIBITORS
GT200600306A (en) AGRECANASA GLUTAMATE INHIBITORS
DOP2006000234A (en) KINASE INHIBITORS
UY31984A (en) DERIVATIVES OF N-substituted 1- (3,4-difluorobenzyl) -6-oxo-1,6-dihydropyrimidin-5-carboxamides and 2- (3,4-difluorobenzyl) -3-oxo-2,3-dihydro- N-substituted 1H-pyrazol-4-carboxamides.