MXPA03005372A - Androgenos 14 (15) -insaturados, 15- y/o 16-sustituidos, con perfil de actividad mixto androgenico-progestacional. - Google Patents
Androgenos 14 (15) -insaturados, 15- y/o 16-sustituidos, con perfil de actividad mixto androgenico-progestacional.Info
- Publication number
- MXPA03005372A MXPA03005372A MXPA03005372A MXPA03005372A MXPA03005372A MX PA03005372 A MXPA03005372 A MX PA03005372A MX PA03005372 A MXPA03005372 A MX PA03005372A MX PA03005372 A MXPA03005372 A MX PA03005372A MX PA03005372 A MXPA03005372 A MX PA03005372A
- Authority
- MX
- Mexico
- Prior art keywords
- profile
- progestational
- unsaturated
- androgen
- mixed
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
- C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines Containing Plant Substances (AREA)
Abstract
Se describen esteroides relacionados con androgeno, que tienen una doble ligadura ?14 y que llevan un sustituyente en cualquiera de los atomos de carbono numeros 15 y 16, o en ambos. Los esteroides de la presente estan caracterizados porque poseen un perfil mixto de actividades androgenicas y progestagenicas. Esto hace que estos compuestos sean adecuados para terapia de reemplazo hormonal masculino o femenino, asi como para anticoncepcion masculina.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP00204543 | 2000-12-15 | ||
PCT/EP2001/014776 WO2002048169A1 (en) | 2000-12-15 | 2001-12-10 | 14(15)-unsaturated 15- and/or 16- substituted androgens with mixed androgen-progestational profile |
Publications (1)
Publication Number | Publication Date |
---|---|
MXPA03005372A true MXPA03005372A (es) | 2004-04-20 |
Family
ID=8172438
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MXPA03005372A MXPA03005372A (es) | 2000-12-15 | 2001-12-10 | Androgenos 14 (15) -insaturados, 15- y/o 16-sustituidos, con perfil de actividad mixto androgenico-progestacional. |
Country Status (12)
Country | Link |
---|---|
US (1) | US20040059140A1 (es) |
EP (1) | EP1343804A1 (es) |
JP (1) | JP2004520300A (es) |
CN (1) | CN1481388A (es) |
AR (1) | AR034194A1 (es) |
AU (1) | AU2002229663A1 (es) |
BR (1) | BR0116127A (es) |
CA (1) | CA2431328A1 (es) |
IL (1) | IL156208A0 (es) |
MX (1) | MXPA03005372A (es) |
PE (1) | PE20020752A1 (es) |
WO (1) | WO2002048169A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JO2492B1 (en) | 2003-04-28 | 2009-10-05 | شيرينج ايه جي | A pharmaceutical formula in the form of aqueous gel for the skin use of its active ingredients |
TW200745156A (en) * | 2005-06-17 | 2007-12-16 | Organon Nv | Steroids having a mixed androgenic and progestagenic profile |
CN110294782B (zh) * | 2018-03-22 | 2023-06-23 | 天津药业研究院股份有限公司 | 一种11烯甾体化合物的制备方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3042689A (en) * | 1960-11-21 | 1962-07-03 | Searle & Co | 16-hydrocarbon substituted 16,17-dihydroxyestren-3-ones, their esters and ethers, and intermediates for their production |
US3577410A (en) * | 1968-07-30 | 1971-05-04 | American Home Prod | 13beta-alkyl-17-hydroxygona-4,14-dien-3-ones |
ZA712312B (en) * | 1970-04-28 | 1972-01-26 | Ochsner Med Found Alton | 4,14-estradiene compounds |
US3766224A (en) * | 1971-06-03 | 1973-10-16 | Sandoz Ag | 15-methyl-substituted steroids |
DE2920184A1 (de) * | 1979-05-17 | 1980-11-27 | Schering Ag | 16 alpha -alkylsteroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate |
US5952319A (en) * | 1997-11-26 | 1999-09-14 | Research Triangle Institute | Androgenic steroid compounds and a method of making and using the same |
DE19827522A1 (de) * | 1998-06-22 | 1999-12-23 | Jenapharm Gmbh | 14,15-Cyclopropanosteroide der 19-Nor-Androstanreihe, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Präparate |
-
2001
- 2001-12-10 AU AU2002229663A patent/AU2002229663A1/en not_active Abandoned
- 2001-12-10 MX MXPA03005372A patent/MXPA03005372A/es unknown
- 2001-12-10 CA CA002431328A patent/CA2431328A1/en not_active Abandoned
- 2001-12-10 US US10/450,693 patent/US20040059140A1/en not_active Abandoned
- 2001-12-10 IL IL15620801A patent/IL156208A0/xx unknown
- 2001-12-10 EP EP01990564A patent/EP1343804A1/en not_active Withdrawn
- 2001-12-10 JP JP2002549700A patent/JP2004520300A/ja not_active Withdrawn
- 2001-12-10 BR BR0116127-0A patent/BR0116127A/pt not_active Application Discontinuation
- 2001-12-10 WO PCT/EP2001/014776 patent/WO2002048169A1/en not_active Application Discontinuation
- 2001-12-10 CN CNA018205801A patent/CN1481388A/zh active Pending
- 2001-12-14 AR ARP010105802A patent/AR034194A1/es unknown
- 2001-12-14 PE PE2001001255A patent/PE20020752A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AR034194A1 (es) | 2004-02-04 |
CA2431328A1 (en) | 2002-06-20 |
AU2002229663A1 (en) | 2002-06-24 |
PE20020752A1 (es) | 2002-08-22 |
IL156208A0 (en) | 2003-12-23 |
WO2002048169A1 (en) | 2002-06-20 |
EP1343804A1 (en) | 2003-09-17 |
BR0116127A (pt) | 2003-11-04 |
JP2004520300A (ja) | 2004-07-08 |
US20040059140A1 (en) | 2004-03-25 |
CN1481388A (zh) | 2004-03-10 |
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