MX9705815A - AGONISTAS beta-ADRENERGICOS. - Google Patents

AGONISTAS beta-ADRENERGICOS.

Info

Publication number
MX9705815A
MX9705815A MX9705815A MX9705815A MX9705815A MX 9705815 A MX9705815 A MX 9705815A MX 9705815 A MX9705815 A MX 9705815A MX 9705815 A MX9705815 A MX 9705815A MX 9705815 A MX9705815 A MX 9705815A
Authority
MX
Mexico
Prior art keywords
compounds
formula
animals
lean meat
relates
Prior art date
Application number
MX9705815A
Other languages
English (en)
Other versions
MXPA97005815A (es
Inventor
Robert Lee Dow
Kristin Marie Lundy
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX9705815A publication Critical patent/MX9705815A/es
Publication of MXPA97005815A publication Critical patent/MXPA97005815A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
  • Indole Compounds (AREA)

Abstract

La presente invencion se refiere a ciertos compuestos de formula (I), a las mezclas racémico-enantioméricas y a isomeros opticos de dichos compuestos, a sus profármacos y a las sales farmacéuticamente aceptables, representadas a continuacion, que son agonistas de receptor beta-adrenérgico y por consiguiente, tienen utilidad como, inter alia, agentes hipoglucémicos y contra la obesidad. La invencion se refiere además a procedimientos de uso de los compuestos y a composiciones que los contienen. Los compuestos de al presente invencion poseen además utilidad para aumentar al deposicion de carne magra y/o mejorar la relacion de carne magra a grasa en animales, por ejemplo animales ungulado, animales de compañía, especialmente perros y aves de corral. Los compuestos de formula (I) tienen la siguiente estructura (Ver Formula) en la que R1, R2, R3, R4 y R5 son como se han definido en la memoria descriptiva.
MXPA/A/1997/005815A 1996-07-31 1997-07-30 Agonistasó-adrenergicos MXPA97005815A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2282796P 1996-07-31 1996-07-31
US022827 1996-07-31

Publications (2)

Publication Number Publication Date
MX9705815A true MX9705815A (es) 1998-08-30
MXPA97005815A MXPA97005815A (es) 1998-11-12

Family

ID=

Also Published As

Publication number Publication date
US5859044A (en) 1999-01-12
CA2211866A1 (en) 1998-01-31
EP0822185A1 (en) 1998-02-04
JPH1087615A (ja) 1998-04-07

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