MX9705061A - Hidroximetilimidazodiazepinas y sus esteres. - Google Patents

Hidroximetilimidazodiazepinas y sus esteres.

Info

Publication number
MX9705061A
MX9705061A MX9705061A MX9705061A MX9705061A MX 9705061 A MX9705061 A MX 9705061A MX 9705061 A MX9705061 A MX 9705061A MX 9705061 A MX9705061 A MX 9705061A MX 9705061 A MX9705061 A MX 9705061A
Authority
MX
Mexico
Prior art keywords
hydrogen
hydroxymethylimidazodiazepines
esters
halogen
formula
Prior art date
Application number
MX9705061A
Other languages
English (en)
Other versions
MXPA97005061A (es
Inventor
Rene Borer
Bernd Buttelmann
Max Gerecke
Andre Szente
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MX9705061A publication Critical patent/MX9705061A/es
Publication of MXPA97005061A publication Critical patent/MXPA97005061A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La invencion está relacionada con hidroximetil-imidazodiazepinas y sus ésteres de formula general I. Estos compuestos pueden usarse como sustancias activas ansiolíticas y/o anticonvulsantes y/o relajantes musculares y/o sedativas-hipnoticas.
MXPA/A/1997/005061A 1995-01-06 1997-07-04 Hidroximetilimidazodiazepinas y sus esteres MXPA97005061A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH28/95-9 1995-01-06
CH2895 1995-01-06
PCT/CH1996/000001 WO1996020941A1 (de) 1995-01-06 1996-01-03 Hydroxymethyl-imidazodiazepine und deren ester

Publications (2)

Publication Number Publication Date
MX9705061A true MX9705061A (es) 1997-10-31
MXPA97005061A MXPA97005061A (es) 1998-07-03

Family

ID=

Also Published As

Publication number Publication date
DK0801651T3 (da) 2001-10-22
DE59607274D1 (de) 2001-08-16
BR9606823A (pt) 1997-12-30
JP3001979B2 (ja) 2000-01-24
GR3036867T3 (en) 2002-01-31
CA2209424A1 (en) 1996-07-11
PT801651E (pt) 2001-12-28
AU4296196A (en) 1996-07-24
ATE203026T1 (de) 2001-07-15
WO1996020941A1 (de) 1996-07-11
US6174881B1 (en) 2001-01-16
CN1168140A (zh) 1997-12-17
FI972865A0 (fi) 1997-07-04
JPH10500998A (ja) 1998-01-27
EP0801651A1 (de) 1997-10-22
ES2159714T3 (es) 2001-10-16
FI972865A (fi) 1997-09-03
EP0801651B1 (de) 2001-07-11
TR199700587T1 (xx) 1998-02-21

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