MX9703363A - Nuevos derivados de pirimidiniloxi- y pirimidinilamino etilfenil-dioxolano. - Google Patents

Nuevos derivados de pirimidiniloxi- y pirimidinilamino etilfenil-dioxolano.

Info

Publication number
MX9703363A
MX9703363A MX9703363A MX9703363A MX9703363A MX 9703363 A MX9703363 A MX 9703363A MX 9703363 A MX9703363 A MX 9703363A MX 9703363 A MX9703363 A MX 9703363A MX 9703363 A MX9703363 A MX 9703363A
Authority
MX
Mexico
Prior art keywords
4alkyl
4alkoxy
aryl
pyrimidinylamino
pyrimidinyloxy
Prior art date
Application number
MX9703363A
Other languages
English (en)
Other versions
MXPA97003363A (es
Inventor
Clemens Lamberth
Fritz Schaub
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MXPA97003363A publication Critical patent/MXPA97003363A/es
Publication of MX9703363A publication Critical patent/MX9703363A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
    • C07C69/78—Benzoic acid esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/18—Radicals substituted by singly bound oxygen or sulfur atoms
    • C07D317/20—Free hydroxyl or mercaptan
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/18—Radicals substituted by singly bound oxygen or sulfur atoms
    • C07D317/22—Radicals substituted by singly bound oxygen or sulfur atoms etherified
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/18—Radicals substituted by singly bound oxygen or sulfur atoms
    • C07D317/24—Radicals substituted by singly bound oxygen or sulfur atoms esterified
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/28—Radicals substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

La invencion describe los 2-[4-(2-(pirimidin-4-iloxi- y -4- ilamino)- etil)- fenil]-dioxolanos de la formula I: en donde R1 es hidrogeno, alquilo C1-4, haloalquilo C1-4 o cicloalquilo C3-6, R2 es hidrogeno, alquilo C1-10, C1-8alcoxi- C1-4alquil, C3-8alqueniloxi-C1-4alquil, C3-8haloalqueniloxi- C1-4alquil, C3-8alquiniloxi-C1-4alquil, C1-8haloalcoxi- C1-4alquil, C1-8alquiltio-C1-4alquil, arilo, ariloxi-C1-4alquil, aril-C1-4alcoxi-C1-4alquil, heteroariloxi-C1-4alquil, C1-4alcoxi-C1-4alcoxi-C1-4alquil, o aril-C1-8alquil, R3 y R4 son en forma independiente halogeno, alquilo C1-4, alcoxi C1-4, C1-4alcoxi-C1-4alquil, C1-4alcoxicarbonil-C1-4alquil, C1-4alcoxicarbonil, ciano-C1-4alquil, ciano, o -COOH, o R3 y R4 juntos forman un miembro de puente seleccionado del 1,4-butadienileno, o 1-S-CH= CH -, cada uno substituido en forma opcional por uno o dos radicales seleccionados del halogeno o alquilo C1-4, y Z es NH u oxígeno; el uso de tales compuestos para el control de la acarina, hongos, e insectos no deseados, las composiciones para facilitar el uso, y la preparacion de los compuestos de la formula I.
MX9703363A 1994-12-07 1995-12-06 Nuevos derivados de pirimidiniloxi- y pirimidinilamino etilfenil-dioxolano. MX9703363A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9424676A GB9424676D0 (en) 1994-12-07 1994-12-07 Organic compounds
GB9424676.6 1994-12-07
PCT/EP1995/004795 WO1996017843A2 (en) 1994-12-07 1995-12-06 Novel pyrimidinyloxy- and pyrimidinylamino-ethylphenyl-dioxolane derivatives

Publications (2)

Publication Number Publication Date
MXPA97003363A MXPA97003363A (es) 1998-02-01
MX9703363A true MX9703363A (es) 1998-02-28

Family

ID=10765538

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9703363A MX9703363A (es) 1994-12-07 1995-12-06 Nuevos derivados de pirimidiniloxi- y pirimidinilamino etilfenil-dioxolano.

Country Status (9)

Country Link
EP (1) EP0796259A2 (es)
JP (1) JPH10512236A (es)
CN (1) CN1168671A (es)
AU (1) AU4260296A (es)
BR (1) BR9509877A (es)
CA (1) CA2206306A1 (es)
GB (1) GB9424676D0 (es)
MX (1) MX9703363A (es)
WO (1) WO1996017843A2 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2005290226A1 (en) 2004-07-16 2006-04-06 Sunesis Pharmaceuticals, Inc. Thienopyrimidines useful as Aurora kinase inhibitors
ATE516291T1 (de) * 2004-10-21 2011-07-15 Dow Agrosciences Llc Thenopyrimidin-verbindungen mit fungizider aktivität
EP1937691A1 (en) * 2005-10-21 2008-07-02 Dow Agrosciences LLC Thieno-pyrimidine compounds having fungicidal activity
NZ597929A (en) * 2009-07-30 2013-09-27 Merial Ltd Insecticidal 4-amino-thieno[2,3-d]-pyrimidine compounds and methods of their use
TWI566701B (zh) * 2012-02-01 2017-01-21 日本農藥股份有限公司 芳烷氧基嘧啶衍生物及包含該衍生物作為有效成分的農園藝用殺蟲劑及其使用方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU734184A1 (ru) * 1977-11-02 1980-05-15 Белорусский Ордена Трудового Красного Знамени Государственный Университет Им.В.И.Ленина Способ получени п-формилстирола
DE69500091T2 (de) * 1994-02-01 1997-05-15 Ube Industries 4-Phenylamino-Pyrimidin-Derivate, Verfahren zur Herstellung und diese enthaltende Schädlingsbekämpfungsmittel für Landwirtschaft und Gartenbau

Also Published As

Publication number Publication date
WO1996017843A3 (en) 1996-08-22
WO1996017843A2 (en) 1996-06-13
CN1168671A (zh) 1997-12-24
AU4260296A (en) 1996-06-26
CA2206306A1 (en) 1996-06-13
GB9424676D0 (en) 1995-02-01
EP0796259A2 (en) 1997-09-24
JPH10512236A (ja) 1998-11-24
BR9509877A (pt) 1997-09-30

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