MX9303764A - 5'-indoliniloxazolidinonas utiles contra mycobacterium tuberculosis fundamento de la invencion. - Google Patents

5'-indoliniloxazolidinonas utiles contra mycobacterium tuberculosis fundamento de la invencion.

Info

Publication number
MX9303764A
MX9303764A MX9303764A MX9303764A MX9303764A MX 9303764 A MX9303764 A MX 9303764A MX 9303764 A MX9303764 A MX 9303764A MX 9303764 A MX9303764 A MX 9303764A MX 9303764 A MX9303764 A MX 9303764A
Authority
MX
Mexico
Prior art keywords
indolinyloxazolidinones
basis
mycobacterium tuberculosis
useful against
against mycobacterium
Prior art date
Application number
MX9303764A
Other languages
English (en)
Spanish (es)
Inventor
Steven Josjeph Brickner
Gary Edward Zurenko
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of MX9303764A publication Critical patent/MX9303764A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
MX9303764A 1992-07-08 1993-06-23 5'-indoliniloxazolidinonas utiles contra mycobacterium tuberculosis fundamento de la invencion. MX9303764A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US90938792A 1992-07-08 1992-07-08

Publications (1)

Publication Number Publication Date
MX9303764A true MX9303764A (es) 1994-01-31

Family

ID=25427164

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9303764A MX9303764A (es) 1992-07-08 1993-06-23 5'-indoliniloxazolidinonas utiles contra mycobacterium tuberculosis fundamento de la invencion.

Country Status (9)

Country Link
EP (1) EP0648119A1 (cs)
JP (1) JPH07508985A (cs)
KR (1) KR950702417A (cs)
AU (1) AU666740B2 (cs)
CA (1) CA2136324A1 (cs)
IL (1) IL106220A0 (cs)
MX (1) MX9303764A (cs)
TW (1) TW260608B (cs)
WO (1) WO1994001110A1 (cs)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
GB9702213D0 (en) * 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
GB9609919D0 (en) * 1996-05-11 1996-07-17 Zeneca Ltd Chemical compounds
GB9717807D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9717804D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9725244D0 (en) 1997-11-29 1998-01-28 Zeneca Ltd Chemical compounds
NZ508174A (en) 1998-06-05 2003-10-31 Astrazeneca Ab Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
GB9928568D0 (en) 1999-12-03 2000-02-02 Zeneca Ltd Chemical compounds
GB0009803D0 (en) 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
US7141588B2 (en) 2002-02-25 2006-11-28 Pfizer, Inc. N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
AR038536A1 (es) 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
ATE321760T1 (de) 2002-08-12 2006-04-15 Pharmacia & Upjohn Co Llc N-aryl-2-oxazolidinone und deren derivate
ATE344036T1 (de) 2002-11-21 2006-11-15 Pharmacia & Upjohn Co Llc N-(4-(piperazin-1-yl)-phenyl-2-oxazolidinon-5- carbonsäureamid-derivate und verwandte verbindungen als antibakterielle mittel
US7304050B2 (en) 2003-09-16 2007-12-04 Pfizer Inc. Antibacterial agents
WO2021258013A1 (en) 2020-06-18 2021-12-23 Akagera Medicines, Inc. Oxazolidinone compounds, liposome compositions comprising oxazolidinone compounds and methods of use thereof

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5314792A (en) * 1976-07-24 1978-02-09 Rubuobuna Buratsurabusukay Ara Copolymers of nnvinylmethylpyrazol and diivinyl crossslinking agent and process for producing same
JPS54110186A (en) * 1978-02-17 1979-08-29 Tokyo Yuuki Kagaku Kougiyou Kk Method of mamufacturing weak basic anion exchange resin
DE3324835A1 (de) * 1983-07-09 1985-01-17 Cassella Ag, 6000 Frankfurt Vernetztes copolymerisat, verfahren zu seiner herstellung und seine verwendung als sorptionsmittel
JPS6023854A (ja) * 1983-07-19 1985-02-06 Konishiroku Photo Ind Co Ltd 写真要素
DE3434137A1 (de) * 1984-09-18 1986-03-20 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von unloeslichen, nur wenig quellbaren pulverfoermigen polymeren
JPS63130605A (ja) * 1986-11-20 1988-06-02 Tokuyama Soda Co Ltd 陰イオン交換体の製造方法
US4889632A (en) * 1987-12-10 1989-12-26 Ceskoslovenska Akademie Ved Macroporous polymeric membranes for the separation of polymers and a method of their application
DE68929303T2 (de) * 1988-09-15 2002-05-02 Pharmacia & Upjohn Co., Kalamazoo 3-(Stickstoff substituierte)phenyl-5-beta-amidomethyloxazoliden-2-one
GB8829835D0 (en) * 1988-12-21 1989-02-15 Smith Kline French Lab Compounds
JPH03708A (ja) * 1989-05-29 1991-01-07 Koei Chem Co Ltd 吸水性材料

Also Published As

Publication number Publication date
EP0648119A1 (en) 1995-04-19
AU4386593A (en) 1994-01-31
CA2136324A1 (en) 1994-01-20
KR950702417A (ko) 1995-07-29
JPH07508985A (ja) 1995-10-05
IL106220A0 (en) 1993-11-15
WO1994001110A1 (en) 1994-01-20
AU666740B2 (en) 1996-02-22
TW260608B (cs) 1995-10-21

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