AR031032A1 - Uso de la tolterodina en el tratamiento del asma - Google Patents

Uso de la tolterodina en el tratamiento del asma

Info

Publication number
AR031032A1
AR031032A1 ARP010104944A ARP010104944A AR031032A1 AR 031032 A1 AR031032 A1 AR 031032A1 AR P010104944 A ARP010104944 A AR P010104944A AR P010104944 A ARP010104944 A AR P010104944A AR 031032 A1 AR031032 A1 AR 031032A1
Authority
AR
Argentina
Prior art keywords
asthma
tolterodine
treatment
copd
group
Prior art date
Application number
ARP010104944A
Other languages
English (en)
Original Assignee
Upjohn Co
Pharmacia Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co, Pharmacia Ab filed Critical Upjohn Co
Publication of AR031032A1 publication Critical patent/AR031032A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Otolaryngology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Emergency Medicine (AREA)
  • Immunology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Separation Using Semi-Permeable Membranes (AREA)

Abstract

Es un método para tratar un mamífero, seleccionado del grupo integrado por seres humanos y caballos, que sufre de asma, EPOC o rinitis alérgica y requiere dicho tratamiento, mediante la inhalacion de una dosis eficaz contra el asma, la EPOC o la rinitis alérgica, respectivamente, de un compuesto seleccionado del grupo integrado por la tolterodina, formula 1; la hidroxitolterodina y el 1-fenilciclopentanocarboxilato de 2-(diisopropilamino) etilo y sus sales farmacéuticamente aceptables.
ARP010104944A 2000-10-24 2001-10-22 Uso de la tolterodina en el tratamiento del asma AR031032A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24289900P 2000-10-24 2000-10-24
US28312001P 2001-04-11 2001-04-11
US31421801P 2001-08-22 2001-08-22

Publications (1)

Publication Number Publication Date
AR031032A1 true AR031032A1 (es) 2003-09-03

Family

ID=27399612

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP010104944A AR031032A1 (es) 2000-10-24 2001-10-22 Uso de la tolterodina en el tratamiento del asma

Country Status (9)

Country Link
US (1) US6538035B2 (es)
EP (1) EP1330241A2 (es)
JP (1) JP2004513099A (es)
AR (1) AR031032A1 (es)
AU (1) AU2002212962A1 (es)
CA (1) CA2422901A1 (es)
MX (1) MXPA03003592A (es)
PE (1) PE20020547A1 (es)
WO (1) WO2002034245A2 (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9203318D0 (sv) * 1992-11-06 1992-11-06 Kabi Pharmacia Ab Novel 3,3-diphenylpropylamines, their use and preparation
ATE418534T1 (de) * 2001-10-26 2009-01-15 Pharmacia & Upjohn Co Llc Quaternäre ammoniumverbindungen und deren verwendung als antimuscarinische wirkstoffe
MXPA04003806A (es) * 2001-11-05 2005-04-08 Upjohn Co Aerosol antimuscarinico.
WO2003070233A1 (en) * 2002-02-19 2003-08-28 Pharmacia Corporation Use of cyclooxygenase inhibitors and antimuscarinic agents for the treatment of incontinence
US7005449B2 (en) 2002-04-23 2006-02-28 Pharmacia & Upjohn Company Tolterodine salts
JP2006523676A (ja) * 2003-04-15 2006-10-19 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー 第四級アンモニウム化合物と、その抗ムスカリン性剤としての使用
CA2522666A1 (en) * 2003-04-18 2004-10-28 Pharmacia & Upjohn Company Llc Combination therapies for chronic obstructive pulmonary disease (copd)
US7629358B2 (en) * 2004-03-17 2009-12-08 Pfizer Inc Compounds useful for the treatment of diseases
ES2268987B1 (es) 2005-08-05 2008-02-01 Ragactives, S.L. Procedimiento para la obtencion de 3,3-difenilpropilaminas.
NZ570693A (en) * 2006-03-20 2011-02-25 Pfizer Ltd Amine derivatives
WO2009019599A2 (en) 2007-08-08 2009-02-12 Themis Laboratories Private Limited Extended release compositions comprising tolterodine
WO2009034432A2 (en) * 2007-09-14 2009-03-19 Pfizer Limited Novel compounds active as muscarinic receptor antagonists
KR101188333B1 (ko) 2008-02-20 2012-10-09 에스케이케미칼주식회사 안정성이 우수하고 경피제로 유용한 톨테로딘 결정성산부가염
CN110372571B (zh) * 2018-04-12 2022-11-15 中国科学院大连化学物理研究所 一种2-(2,2-二芳基乙基)-环胺衍生物或盐及合成和应用与组合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5382600A (en) 1988-01-22 1995-01-17 Pharmacia Aktiebolag 3,3-diphenylpropylamines and pharmaceutical compositions thereof
SE9203318D0 (sv) 1992-11-06 1992-11-06 Kabi Pharmacia Ab Novel 3,3-diphenylpropylamines, their use and preparation
EP0923536A1 (en) 1996-07-29 1999-06-23 Pharmacia & Upjohn Aktiebolag Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation
KR20000057548A (ko) 1996-12-13 2000-09-25 알프레드 엘. 미첼슨 광학적 전송물질 및 결합재

Also Published As

Publication number Publication date
MXPA03003592A (es) 2003-06-19
US6538035B2 (en) 2003-03-25
EP1330241A2 (en) 2003-07-30
US20020161054A1 (en) 2002-10-31
CA2422901A1 (en) 2002-05-02
WO2002034245A2 (en) 2002-05-02
AU2002212962A1 (en) 2002-05-06
PE20020547A1 (es) 2002-06-12
JP2004513099A (ja) 2004-04-30

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