MX381440B - Composicion farmaceutica para tratar colitis ulcerativa. - Google Patents
Composicion farmaceutica para tratar colitis ulcerativa.Info
- Publication number
- MX381440B MX381440B MX2017003780A MX2017003780A MX381440B MX 381440 B MX381440 B MX 381440B MX 2017003780 A MX2017003780 A MX 2017003780A MX 2017003780 A MX2017003780 A MX 2017003780A MX 381440 B MX381440 B MX 381440B
- Authority
- MX
- Mexico
- Prior art keywords
- ulcerative colitis
- pharmaceutical composition
- treatment
- pharmaceutically acceptable
- acceptable salt
- Prior art date
Links
- 206010009900 Colitis ulcerative Diseases 0.000 title abstract 3
- 201000006704 Ulcerative Colitis Diseases 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Se proporciona una composición farmacéutica para tratar colitis ulcerativa, que comprende un compuesto representado por una fórmula (1) o una sal farmacéuticamente aceptable del mismo, en donde el compuesto o la sal farmacéuticamente aceptable se administra en una cantidad de 600 mg o más por día a un paciente con colitis ulcerativa.(ver Fórmula).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2014198681 | 2014-09-29 | ||
| PCT/JP2015/059717 WO2016051828A1 (ja) | 2014-09-29 | 2015-03-27 | 潰瘍性大腸炎の治療用医薬組成物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX2017003780A MX2017003780A (es) | 2017-06-30 |
| MX381440B true MX381440B (es) | 2025-03-12 |
Family
ID=55629887
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2017003780A MX381440B (es) | 2014-09-29 | 2015-03-27 | Composicion farmaceutica para tratar colitis ulcerativa. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US10183022B2 (es) |
| JP (1) | JP6580053B2 (es) |
| KR (1) | KR102319078B1 (es) |
| AU (1) | AU2015326196B2 (es) |
| BR (1) | BR112017006272A2 (es) |
| CA (1) | CA2961311C (es) |
| EA (1) | EA034956B1 (es) |
| MX (1) | MX381440B (es) |
| WO (1) | WO2016051828A1 (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3514235B8 (de) * | 2018-01-18 | 2024-02-14 | Sterna Biologicals GmbH | Zusammensetzung zur behandlung eines an colitis ulcerosa leidenden patienten sowie verwendung der zusammensetzung als arzneimittel |
| CN112996786B (zh) | 2018-10-30 | 2024-08-20 | 吉利德科学公司 | 用于抑制α4β7整合素的化合物 |
| JP7189369B2 (ja) | 2018-10-30 | 2022-12-13 | ギリアード サイエンシーズ, インコーポレイテッド | アルファ4β7インテグリンの阻害のための化合物 |
| HUE070112T2 (hu) | 2018-10-30 | 2025-05-28 | Gilead Sciences Inc | 3-(Kinolin-8-il)-1,4-dihidropirido[3,4-d]pirimidin-2,4-dion-származékok mint alpha4beta7 integrin gátlók gyulladásos betegségek kezelésére |
| EP3873900B1 (en) | 2018-10-30 | 2025-01-08 | Gilead Sciences, Inc. | Imidazo[1,2-a]pyridine derivatives as alpha4beta7 integrin inhibitors for the treatment of inflammatory diseases |
| JP7491996B2 (ja) | 2019-08-14 | 2024-05-28 | ギリアード サイエンシーズ, インコーポレイテッド | α4β7インテグリンの阻害のための化合物 |
| GB202002926D0 (en) * | 2020-02-28 | 2020-04-15 | Benevolentai Tech Limited | Compositions and uses thereof |
| KR102758046B1 (ko) | 2021-11-05 | 2025-01-23 | (주) 넥셀 | 궤양성 대장염 예방 또는 치료용 재조합 단백질 및 이를 포함하는 궤양성 대장염 예방 또는 치료용 조성물 |
| CN114668775B (zh) * | 2022-02-28 | 2023-12-19 | 中国药科大学 | 纤维素衍生物在制备治疗溃疡性结肠炎药物中的应用 |
| US20250206825A1 (en) | 2022-03-11 | 2025-06-26 | Osaka University | Composition for preventing or treating myocarditis, comprising vla-4 inhibitor |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1325480C (zh) | 2000-08-18 | 2007-07-11 | 味之素株式会社 | 苯基丙氨酸衍生物 |
| JP4572832B2 (ja) | 2003-02-20 | 2010-11-04 | 味の素株式会社 | キナゾリンジオン骨格を有するフェニルアラニン誘導体の製造方法及び製造中間体 |
| ES2360064T3 (es) | 2003-11-14 | 2011-05-31 | Ajinomoto Co., Inc. | Dispersión sólida o preparación de dispersión sólida medicinal de un derivado de fenilalanina. |
| EP1683525B1 (en) | 2003-11-14 | 2017-05-17 | EA Pharma Co., Ltd. | Sustained-release phenylalanine derivative preparation for oral administration |
| WO2005051525A1 (en) | 2003-11-25 | 2005-06-09 | Polyvalor, Limited Partnership | Permeation barrier coating or layer with modulated properties and methods of making the same |
| EP1688410B1 (en) | 2003-11-27 | 2014-03-05 | Ajinomoto Co., Inc. | Crystal of phenylalanine derivative and process for producing the same |
| CA2613249A1 (en) | 2005-06-21 | 2006-12-28 | Ajinomoto Co., Inc. | Crystals of phenylalanine derivatives, production method thereof and use thereof |
| ATE549321T1 (de) | 2006-11-22 | 2012-03-15 | Ajinomoto Kk | Verfahren zur herstellung von phenylalaninderivaten mit chinazolindiongerüsten, und zwischenprodukte für die herstellung |
| US7987289B2 (en) | 2008-06-24 | 2011-07-26 | Microsoft Corporation | Participating in cloud as totally stubby edge |
| CN106963741A (zh) | 2010-03-29 | 2017-07-21 | Ea制药株式会社 | 含有苯基丙氨酸衍生物的医药制剂 |
| ES2549768T3 (es) * | 2010-03-29 | 2015-11-02 | Ajinomoto Co., Inc. | Cristal de sal hidrocloruro de derivado de fenilalanina |
-
2015
- 2015-03-27 EA EA201790726A patent/EA034956B1/ru not_active IP Right Cessation
- 2015-03-27 BR BR112017006272-0A patent/BR112017006272A2/pt not_active Application Discontinuation
- 2015-03-27 KR KR1020177011379A patent/KR102319078B1/ko not_active Expired - Fee Related
- 2015-03-27 CA CA2961311A patent/CA2961311C/en active Active
- 2015-03-27 MX MX2017003780A patent/MX381440B/es unknown
- 2015-03-27 WO PCT/JP2015/059717 patent/WO2016051828A1/ja not_active Ceased
- 2015-03-27 AU AU2015326196A patent/AU2015326196B2/en not_active Ceased
- 2015-03-27 JP JP2016551565A patent/JP6580053B2/ja active Active
-
2017
- 2017-03-28 US US15/471,745 patent/US10183022B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| CA2961311A1 (en) | 2016-04-07 |
| MX2017003780A (es) | 2017-06-30 |
| KR20170057435A (ko) | 2017-05-24 |
| AU2015326196B2 (en) | 2020-05-14 |
| KR102319078B1 (ko) | 2021-10-29 |
| CA2961311C (en) | 2022-12-06 |
| US20170196870A1 (en) | 2017-07-13 |
| US10183022B2 (en) | 2019-01-22 |
| WO2016051828A1 (ja) | 2016-04-07 |
| EA201790726A1 (ru) | 2017-11-30 |
| AU2015326196A1 (en) | 2017-03-23 |
| JPWO2016051828A1 (ja) | 2017-07-27 |
| EA034956B1 (ru) | 2020-04-10 |
| JP6580053B2 (ja) | 2019-09-25 |
| BR112017006272A2 (pt) | 2018-03-13 |
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