MX365620B - Composiciones para el cuidado de la piel y metodos que comprenden agonistas selectivos del receptor de melanocortina 1. - Google Patents
Composiciones para el cuidado de la piel y metodos que comprenden agonistas selectivos del receptor de melanocortina 1.Info
- Publication number
- MX365620B MX365620B MX2015006342A MX2015006342A MX365620B MX 365620 B MX365620 B MX 365620B MX 2015006342 A MX2015006342 A MX 2015006342A MX 2015006342 A MX2015006342 A MX 2015006342A MX 365620 B MX365620 B MX 365620B
- Authority
- MX
- Mexico
- Prior art keywords
- skin care
- care compositions
- methods
- skin
- melanocortin
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/06—Tripeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/07—Tetrapeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/02—Cosmetics or similar toiletry preparations characterised by special physical form
- A61K8/04—Dispersions; Emulsions
- A61K8/06—Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/64—Proteins; Peptides; Derivatives or degradation products thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q17/00—Barrier preparations; Preparations brought into direct contact with the skin for affording protection against external influences, e.g. sunlight, X-rays or other harmful rays, corrosive materials, bacteria or insect stings
- A61Q17/04—Topical preparations for affording protection against sunlight or other radiation; Topical sun tanning preparations
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/004—Aftersun preparations
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/04—Preparations for care of the skin for chemically tanning the skin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/08—Anti-ageing preparations
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Dermatology (AREA)
- Medicinal Chemistry (AREA)
- Organic Chemistry (AREA)
- Epidemiology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Immunology (AREA)
- Gastroenterology & Hepatology (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Birds (AREA)
- Gerontology & Geriatric Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Dispersion Chemistry (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Abstract
La presente invención se refiere a los tri- y tetra-péptidos cortos de acuerdo con la siguiente Fórmula I Ar (CH2) mX1-X2-CO-X3-X4-X5-(Trp) n-NX6R son agonistas, selectivos, potentes del receptor de melanocortina 1 (MC1R). Se proporcionan en la presente composiciones para el cuidado de la piel incluyendo los agonistas de péptido de la Fórmula I de MC1R y métodos para regular una afección de la piel de un mamífero que incluye aplicar a una superficie de tratamiento del cuerpo una cantidad segura y efectiva de una composición para el cuidado de la piel que incluye un péptido de la Fórmula I. Los péptidos, composiciones para el cuidado de la piel, y métodos para el cuidado de la piel descritos en la presente son útiles en regular una afección de la piel de un mamífero asociado con la exposición de la radiación ultravioleta (UV), incluyendo quemadura solar, sensibilidad de UV, fotoenvejecimiento y pigmentación de la piel, particullarmente en ausencia de exposición al sol.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261729018P | 2012-11-21 | 2012-11-21 | |
PCT/US2013/071031 WO2014081845A2 (en) | 2012-11-21 | 2013-11-20 | Skin care compositions and methods comprising selective agonists of melanocortin 1 receptor |
Publications (2)
Publication Number | Publication Date |
---|---|
MX2015006342A MX2015006342A (es) | 2016-02-25 |
MX365620B true MX365620B (es) | 2019-06-07 |
Family
ID=50776668
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2015006342A MX365620B (es) | 2012-11-21 | 2013-11-20 | Composiciones para el cuidado de la piel y metodos que comprenden agonistas selectivos del receptor de melanocortina 1. |
MX2015006333A MX366171B (es) | 2012-11-21 | 2013-11-20 | Composiciones farmaceuticas y metodos terapeuticos de uso que comprenden agonistas selectivos del receptor de melanocortina. |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2015006333A MX366171B (es) | 2012-11-21 | 2013-11-20 | Composiciones farmaceuticas y metodos terapeuticos de uso que comprenden agonistas selectivos del receptor de melanocortina. |
Country Status (7)
Country | Link |
---|---|
US (3) | US9434764B2 (es) |
EP (2) | EP2922565B1 (es) |
AU (3) | AU2013348044B2 (es) |
CA (2) | CA2892134C (es) |
ES (2) | ES2768423T3 (es) |
MX (2) | MX365620B (es) |
WO (2) | WO2014081846A2 (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016187264A1 (en) * | 2015-05-18 | 2016-11-24 | The Arizona Board Of Regents On Behalf Of The University Of Arizona | Enhanced melanoma cancer prevention by novel melanotropins |
US10086035B2 (en) | 2016-02-04 | 2018-10-02 | ALASTIN Skincare, Inc. | Compositions and methods for invasive and non-invasive procedural skincare |
JP7039814B2 (ja) * | 2016-10-04 | 2022-03-23 | ディーエスエム アイピー アセッツ ビー.ブイ. | メラノコルチン-1-受容体アゴニスト |
CN111182914A (zh) | 2017-08-03 | 2020-05-19 | 阿拉斯廷护肤公司 | 用于改善皮肤松弛和身体轮廓的组合物和方法 |
BR112020008175A2 (pt) * | 2017-10-30 | 2020-10-20 | Dsm Ip Assets B.V. | compostos inovadores |
JP7296642B2 (ja) * | 2018-02-27 | 2023-06-23 | リポトゥルー,エセ.エレ. | 化粧料および医薬に使用するためのペプチドおよび組成物 |
WO2020028694A1 (en) | 2018-08-02 | 2020-02-06 | ALASTIN Skincare, Inc. | Liposomal compositions and methods of use |
BR112022025115A2 (pt) * | 2020-06-10 | 2023-02-07 | Mitsubishi Tanabe Pharma Corp | Agente profilático ou terapêutico para fotodermatose |
CN116925182A (zh) * | 2022-04-02 | 2023-10-24 | 肽鼎生物科技(深圳)有限公司 | 多肽药物及凝胶制剂的应用 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2002536295A (ja) | 1998-12-14 | 2002-10-29 | パラチン テクノロジーズ, インク. | 金属ペプチド組合せライブラリ及びその利用法 |
US6579968B1 (en) | 1999-06-29 | 2003-06-17 | Palatin Technologies, Inc. | Compositions and methods for treatment of sexual dysfunction |
CA2453515A1 (en) * | 2001-07-11 | 2003-01-23 | Palatin Technologies, Inc. | Linear and cyclic melanocortin receptor-specific peptides |
US7034004B2 (en) * | 2002-05-07 | 2006-04-25 | University Of Florida | Peptides and methods for the control of obesity |
WO2005048967A1 (en) | 2003-11-24 | 2005-06-02 | Clinuvel Pharmaceuticals Limited | A method of inducing melanogenesis in humans with mc1r variant alleles |
EP2368562B1 (en) | 2004-10-08 | 2015-06-17 | Clinuvel Pharmaceuticals Limited | Compositions and methods for inducing melanogenesis in a subject |
CA2702169A1 (en) * | 2007-10-12 | 2009-04-16 | Decode Genetics Ehf | Sequence variants for inferring human pigmentation patterns |
MX356295B (es) | 2008-05-27 | 2018-05-22 | Genzyme Corp | Análogos de péptido de la hormona de estimulación de alfa-melanocito. |
EA021897B1 (ru) * | 2009-11-23 | 2015-09-30 | Палатин Текнолоджиз, Инк. | Циклические пептиды, специфичные к рецептору меланокортина-1 |
-
2013
- 2013-11-20 AU AU2013348044A patent/AU2013348044B2/en active Active
- 2013-11-20 WO PCT/US2013/071033 patent/WO2014081846A2/en active Application Filing
- 2013-11-20 AU AU2013348043A patent/AU2013348043B2/en active Active
- 2013-11-20 CA CA2892134A patent/CA2892134C/en active Active
- 2013-11-20 US US14/646,407 patent/US9434764B2/en active Active
- 2013-11-20 EP EP13856556.9A patent/EP2922565B1/en active Active
- 2013-11-20 EP EP13857618.6A patent/EP2925340B8/en active Active
- 2013-11-20 ES ES13856556T patent/ES2768423T3/es active Active
- 2013-11-20 MX MX2015006342A patent/MX365620B/es active IP Right Grant
- 2013-11-20 MX MX2015006333A patent/MX366171B/es active IP Right Grant
- 2013-11-20 US US14/646,410 patent/US9834580B2/en active Active
- 2013-11-20 CA CA2892144A patent/CA2892144C/en active Active
- 2013-11-20 ES ES13857618T patent/ES2738555T3/es active Active
- 2013-11-20 WO PCT/US2013/071031 patent/WO2014081845A2/en active Application Filing
-
2017
- 2017-10-26 US US15/794,301 patent/US10301355B2/en active Active
-
2018
- 2018-06-12 AU AU2018204153A patent/AU2018204153B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
CA2892134C (en) | 2022-10-04 |
US20180066016A1 (en) | 2018-03-08 |
CA2892144C (en) | 2020-04-28 |
ES2738555T3 (es) | 2020-01-23 |
US20150297667A1 (en) | 2015-10-22 |
WO2014081845A3 (en) | 2015-07-30 |
EP2925340A4 (en) | 2017-01-04 |
US10301355B2 (en) | 2019-05-28 |
WO2014081845A2 (en) | 2014-05-30 |
WO2014081846A3 (en) | 2015-11-19 |
EP2922565A2 (en) | 2015-09-30 |
EP2922565A4 (en) | 2016-06-15 |
US9434764B2 (en) | 2016-09-06 |
MX366171B (es) | 2019-07-01 |
ES2768423T3 (es) | 2020-06-22 |
AU2013348044A1 (en) | 2015-06-04 |
AU2018204153B2 (en) | 2019-04-18 |
WO2014081846A2 (en) | 2014-05-30 |
CA2892134A1 (en) | 2014-05-30 |
AU2013348043B2 (en) | 2017-11-02 |
AU2018204153A1 (en) | 2018-06-28 |
US9834580B2 (en) | 2017-12-05 |
EP2925340A2 (en) | 2015-10-07 |
EP2922565B1 (en) | 2019-11-13 |
EP2925340B1 (en) | 2019-05-08 |
EP2925340B8 (en) | 2019-07-24 |
US20150299251A1 (en) | 2015-10-22 |
MX2015006342A (es) | 2016-02-25 |
AU2013348043A1 (en) | 2015-06-04 |
CA2892144A1 (en) | 2014-05-30 |
AU2013348044B2 (en) | 2018-03-15 |
MX2015006333A (es) | 2016-01-20 |
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