MX3326E - Procedimiento para la preparacion de derivados de triazolocicloalquiltiadiazina - Google Patents
Procedimiento para la preparacion de derivados de triazolocicloalquiltiadiazinaInfo
- Publication number
- MX3326E MX3326E MX000332U MX33276U MX3326E MX 3326 E MX3326 E MX 3326E MX 000332 U MX000332 U MX 000332U MX 33276 U MX33276 U MX 33276U MX 3326 E MX3326 E MX 3326E
- Authority
- MX
- Mexico
- Prior art keywords
- carbon atoms
- chosen
- hydrogen
- see
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/12—Oxygen or sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
La presente invención se refiere a procedimiento para la preparación de derivados de triazolocicloalquiltiadiazina, que tiene la fórmula (VER FIGURA ) en donde R1, R2 y R3 se eligen de hidrógeno y alquilo inferior que tiene de 1 a 4 átomos de carbono; R4 se elige de hidrógeno, alquilo inferior que tiene de 1 a 4 átomos de carbono y oxo; R5 se elige de hidrógeno, alquilo que tiene de 1 a 15 átomos de carbono trifluorometilo, cicloalquilo que tine de 3 a 6 átomos de carbono, fenilo alcoxialquilo que tiene de 2 a 8 átomos de carbono y fenoxialquilo que tiene de 7 a 10 átomos de carbono; A es un enlace sigma o el radical -(CH2)8- en el cual n es un entero de 1 a 7; y una sal de adición de ácido farmacéuticamente aceptable de la misma, que comprende hacer reaccionar un 4-amino-4H-1,2, 4-triazol-3-tiol que tiene la fórmula: (VER FIGURA ) en la cual R5 es como se ha definido arriba con una 2-halocicloalcanona que tiene la fórmula: (VER FIGURA) en la cual R1,R2, R3, R4 y A son como se ha definido arriba y X es halógeno que se elige de cloro, bromo, y yodo, a una temperatura que varía de la temperatura ambiente a 150°C, y durante un período de tiempo que varía de una a doce horas.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/571,942 US3954984A (en) | 1975-04-28 | 1975-04-28 | Triazolocycloalkylthiadiazine derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX3326E true MX3326E (es) | 1980-09-26 |
Family
ID=24285695
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX000332U MX3326E (es) | 1975-04-28 | 1976-02-17 | Procedimiento para la preparacion de derivados de triazolocicloalquiltiadiazina |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US3954984A (es) |
| JP (1) | JPS51127095A (es) |
| BE (1) | BE838974A (es) |
| CA (1) | CA1051891A (es) |
| CH (1) | CH620217A5 (es) |
| DE (1) | DE2607626A1 (es) |
| DK (1) | DK140503B (es) |
| ES (1) | ES445008A1 (es) |
| FR (1) | FR2309230A1 (es) |
| GB (1) | GB1477127A (es) |
| IE (1) | IE42879B1 (es) |
| IL (1) | IL49072A (es) |
| MX (1) | MX3326E (es) |
| NL (1) | NL7602256A (es) |
| NO (1) | NO760418L (es) |
| PH (1) | PH11482A (es) |
| SE (1) | SE7601568L (es) |
| ZA (1) | ZA76939B (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4025510A (en) * | 1975-12-01 | 1977-05-24 | E. I. Du Pont De Nemours And Company | 2,4-Diaryl[1,3,4H]thiadiazines fused to quinoxalines |
| DE3433037A1 (de) * | 1984-09-08 | 1986-03-20 | Gödecke AG, 1000 Berlin | 1,2,4-benzothiadiazinoxid-derivate, verfahren zu deren herstellung und deren verwendung |
-
1975
- 1975-04-28 US US05/571,942 patent/US3954984A/en not_active Expired - Lifetime
-
1976
- 1976-02-09 ES ES445008A patent/ES445008A1/es not_active Expired
- 1976-02-10 DK DK52976AA patent/DK140503B/da unknown
- 1976-02-10 NO NO760418A patent/NO760418L/no unknown
- 1976-02-12 SE SE7601568A patent/SE7601568L/xx unknown
- 1976-02-13 IE IE292/76A patent/IE42879B1/en unknown
- 1976-02-17 CA CA245,924A patent/CA1051891A/en not_active Expired
- 1976-02-17 MX MX000332U patent/MX3326E/es unknown
- 1976-02-17 ZA ZA939A patent/ZA76939B/xx unknown
- 1976-02-19 IL IL49072A patent/IL49072A/xx unknown
- 1976-02-19 GB GB651176A patent/GB1477127A/en not_active Expired
- 1976-02-20 CH CH213676A patent/CH620217A5/de not_active IP Right Cessation
- 1976-02-24 FR FR7605112A patent/FR2309230A1/fr active Granted
- 1976-02-25 DE DE19762607626 patent/DE2607626A1/de not_active Withdrawn
- 1976-02-26 BE BE164677A patent/BE838974A/xx unknown
- 1976-03-04 NL NL7602256A patent/NL7602256A/xx not_active Application Discontinuation
- 1976-03-12 PH PH18200A patent/PH11482A/en unknown
- 1976-04-05 JP JP51037329A patent/JPS51127095A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| FR2309230A1 (fr) | 1976-11-26 |
| DK52976A (es) | 1976-10-29 |
| NL7602256A (nl) | 1976-11-01 |
| AU1138176A (en) | 1977-09-01 |
| ZA76939B (en) | 1977-01-26 |
| DE2607626A1 (de) | 1976-11-11 |
| NO760418L (es) | 1976-10-29 |
| DK140503B (da) | 1979-09-17 |
| CA1051891A (en) | 1979-04-03 |
| ES445008A1 (es) | 1977-06-01 |
| GB1477127A (en) | 1977-06-22 |
| SE7601568L (sv) | 1976-10-29 |
| BE838974A (fr) | 1976-06-16 |
| IL49072A0 (en) | 1976-04-30 |
| IE42879L (en) | 1976-10-28 |
| FR2309230B1 (es) | 1980-06-27 |
| IL49072A (en) | 1978-12-17 |
| IE42879B1 (en) | 1980-11-05 |
| US3954984A (en) | 1976-05-04 |
| DK140503C (es) | 1980-02-11 |
| JPS51127095A (en) | 1976-11-05 |
| PH11482A (en) | 1978-02-01 |
| CH620217A5 (es) | 1980-11-14 |
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