MX2023004955A - Compuestos de aminotiazol deuterados como compuestos antiviricos. - Google Patents

Compuestos de aminotiazol deuterados como compuestos antiviricos.

Info

Publication number
MX2023004955A
MX2023004955A MX2023004955A MX2023004955A MX2023004955A MX 2023004955 A MX2023004955 A MX 2023004955A MX 2023004955 A MX2023004955 A MX 2023004955A MX 2023004955 A MX2023004955 A MX 2023004955A MX 2023004955 A MX2023004955 A MX 2023004955A
Authority
MX
Mexico
Prior art keywords
compounds
deuterated
aminothiazole
antiviral
antiviral compounds
Prior art date
Application number
MX2023004955A
Other languages
English (en)
Spanish (es)
Inventor
Christian Gege
Gerald Kleymann
Original Assignee
Innovative Molecules Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Innovative Molecules Gmbh filed Critical Innovative Molecules Gmbh
Publication of MX2023004955A publication Critical patent/MX2023004955A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/54Nitrogen and either oxygen or sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C07B59/002Heterocyclic compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05Isotopically modified compounds, e.g. labelled

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
MX2023004955A 2020-10-29 2021-10-28 Compuestos de aminotiazol deuterados como compuestos antiviricos. MX2023004955A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP20204545 2020-10-29
PCT/EP2021/080023 WO2022090409A1 (en) 2020-10-29 2021-10-28 Deuterated aminothiazole compounds as antiviral compounds

Publications (1)

Publication Number Publication Date
MX2023004955A true MX2023004955A (es) 2023-05-17

Family

ID=73037895

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2023004955A MX2023004955A (es) 2020-10-29 2021-10-28 Compuestos de aminotiazol deuterados como compuestos antiviricos.

Country Status (9)

Country Link
US (1) US12552756B2 (enExample)
EP (1) EP4237414A1 (enExample)
JP (1) JP2023552274A (enExample)
KR (1) KR20230131177A (enExample)
CN (1) CN116783171A (enExample)
AU (1) AU2021367976A1 (enExample)
CA (1) CA3196645A1 (enExample)
MX (1) MX2023004955A (enExample)
WO (1) WO2022090409A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4466255A1 (en) 2022-01-17 2024-11-27 Innovative Molecules GmbH Solid crystalline forms of helicase-primase inhibitors and process of preparation thereof
IL325911A (en) 2023-07-17 2026-03-01 Innovative Molecules Gmbh Micronized crystalline hydrochloride salts of antiviral helicase-primase inhibitor compounds
WO2026078039A1 (en) 2024-10-09 2026-04-16 Innovative Molecules Gmbh Oral administration forms of antiviral helicase-primase inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DOP2000000109A (es) * 1999-12-23 2002-08-30 Gerald Kleymann Derivados de tiazolilamida
GEP20207128B (en) * 2016-04-06 2020-07-10 Molecules Gm Innovative Aminothiazole derivatives useful as antiviral agents
MX2020003369A (es) * 2017-10-05 2020-07-29 Innovative Molecules Gmbh Enantiomeros de tiazoles sustituidos como compuestos antivirales.
TW202038947A (zh) 2018-11-28 2020-11-01 德商創新分子有限責任公司 在與溶瘤病毒之組合療法中治療癌症的解旋酶引子酶抑制劑

Also Published As

Publication number Publication date
CN116783171A (zh) 2023-09-19
AU2021367976A9 (en) 2025-03-13
EP4237414A1 (en) 2023-09-06
KR20230131177A (ko) 2023-09-12
US20230391738A1 (en) 2023-12-07
WO2022090409A1 (en) 2022-05-05
US12552756B2 (en) 2026-02-17
AU2021367976A1 (en) 2023-06-08
JP2023552274A (ja) 2023-12-15
CA3196645A1 (en) 2022-05-05

Similar Documents

Publication Publication Date Title
CL2020002695A1 (es) Péptidos macrocíclicos contra actinetobacter baumannii
MX375099B (es) Derivados de aminotiazol útiles como agentes antivíricos.
CO2021012579A2 (es) Compuestos útiles en la terapia del vih
BR112022002496A2 (pt) Compostos deuterados para uso no tratamento de câncer
MX2023004955A (es) Compuestos de aminotiazol deuterados como compuestos antiviricos.
PH12018500904A1 (en) Peptide macrocycles against acinetobacter baumannii
UY35263A (es) Compuestos terapéuticos
UY37997A (es) Agentes antivirales contra la hepatitis b
CO6470845A2 (es) Derivados de pirimidina novedosos y su uso en el tratamiento del cancer y enfermedades adicionales
MX2018005890A (es) Composiciones para tratar atrofia muscular espinal.
BR112015004113A2 (pt) 6-aminoácido heteroarila diidropirimidinas para o tratamento e profilaxia da infecção pelo vírus da hepatite b
BR112017020837A2 (pt) compostos de carbamoilpiridona policíclicos e seu uso farmacêutico
CL2021001388A1 (es) Compuestos útiles en la terapia para el vih
BR112014006559A2 (pt) derivados do ácido betulínico com atividade antiviral
BR112023012947A2 (pt) Inibidores de lrrk2
CL2020003248A1 (es) Derivados de tetrahidrotienopiridina n-sustituidos y sus usos
CL2017002498A1 (es) Piridopirimidinonas y su uso como modulares del receptor nmda
MX2019011220A (es) Compuesto de pirrolopiridina novedoso, metodo de preparacion del mismo y uso del mismo.
BR112022010181A2 (pt) Composto tri-heterocíclico como inibidor de jak e uso do mesmo
CR20180615A (es) Nuevos derivados de [1,2,3]triazol[4,5-d]pirimidina
MX2021012544A (es) Compuestos novedosos y composiciones farmaceuticas de los mismos para el tratamiento de enfermedades renales.
MY197518A (en) Preventive and/or therapeutic agent of immune disease
BR112023010200A2 (pt) Inibidores enzimáticos
CO2022008835A2 (es) Agonistas del tlr7
BR112021019589A2 (pt) Derivados de isocromenos como inibidores de fosfoinositídeo 3-cinases