MX2022014549A - Metodo para preparar 2-cloro-n-(1-cianociclopropil)-5-[2'-metil-5' -(pentafluoroetil)-4'-(trifluorometil)-2'h-1,3'-bipirazol-4-il]be nzamida. - Google Patents

Metodo para preparar 2-cloro-n-(1-cianociclopropil)-5-[2'-metil-5' -(pentafluoroetil)-4'-(trifluorometil)-2'h-1,3'-bipirazol-4-il]be nzamida.

Info

Publication number
MX2022014549A
MX2022014549A MX2022014549A MX2022014549A MX2022014549A MX 2022014549 A MX2022014549 A MX 2022014549A MX 2022014549 A MX2022014549 A MX 2022014549A MX 2022014549 A MX2022014549 A MX 2022014549A MX 2022014549 A MX2022014549 A MX 2022014549A
Authority
MX
Mexico
Prior art keywords
bipyrazol
cyanocyclopropyl
pentafluoroethyl
benzamide
chloro
Prior art date
Application number
MX2022014549A
Other languages
English (en)
Inventor
Werner Lindner
Birgit Keil
Britta Olenik
Franz-Josef Mais
Hildegard Scheithauer
Original Assignee
Vetoquinol Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vetoquinol Sa filed Critical Vetoquinol Sa
Publication of MX2022014549A publication Critical patent/MX2022014549A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J27/00—Catalysts comprising the elements or compounds of halogens, sulfur, selenium, tellurium, phosphorus or nitrogen; Catalysts comprising carbon compounds
    • B01J27/14—Phosphorus; Compounds thereof
    • B01J27/185—Phosphorus; Compounds thereof with iron group metals or platinum group metals
    • B01J27/1856—Phosphorus; Compounds thereof with iron group metals or platinum group metals with platinum group metals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

La presente invención se relaciona con un método para preparar 2-cloro-N-(1-cianociclopropil)-5-[2'-metil-5'-(pentafluoroetil)-4 '-(trifluorometil)-2'H-1,3'-bipirazol-4-il]benzamida, es decir, el compuesto de la Fórmula (I) y con un método para purificar el compuesto de la Fórmula I. La presente invención se relaciona además con nuevas formas cristalinas del compuesto de la Fórmula I.
MX2022014549A 2020-05-27 2021-05-26 Metodo para preparar 2-cloro-n-(1-cianociclopropil)-5-[2'-metil-5' -(pentafluoroetil)-4'-(trifluorometil)-2'h-1,3'-bipirazol-4-il]be nzamida. MX2022014549A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP20176774 2020-05-27
PCT/EP2021/064095 WO2021239835A1 (en) 2020-05-27 2021-05-26 Method for preparing 2-chloro-N-(1-cyanocyclopropyl)-5-[2'-methyl-5'-(pentafluoroethyl)-4'-(trifluoromethyl)-2'h-1,3'-bipyrazol-4-yl]benzamide

Publications (1)

Publication Number Publication Date
MX2022014549A true MX2022014549A (es) 2022-12-15

Family

ID=70861296

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2022014549A MX2022014549A (es) 2020-05-27 2021-05-26 Metodo para preparar 2-cloro-n-(1-cianociclopropil)-5-[2'-metil-5' -(pentafluoroetil)-4'-(trifluorometil)-2'h-1,3'-bipirazol-4-il]be nzamida.

Country Status (10)

Country Link
US (1) US20230203013A1 (es)
EP (1) EP4157830A1 (es)
JP (1) JP2023528015A (es)
KR (1) KR20230016672A (es)
CN (1) CN115605468A (es)
AU (1) AU2021279260A1 (es)
BR (1) BR112022023008A2 (es)
CA (1) CA3178621A1 (es)
MX (1) MX2022014549A (es)
WO (1) WO2021239835A1 (es)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014012975A1 (en) 2012-07-19 2014-01-23 Bayer Cropscience Ag Process for the preparation of 5-fluoro-1h-pyrazoles
PL2953942T3 (pl) 2013-02-06 2018-03-30 Bayer Cropscience Aktiengesellschaft Podstawione halogenem pochodne pirazolu jako środki do zwalczania szkodników
BR112016011899B1 (pt) 2013-11-27 2021-03-23 Bayer Animal Health Gmbh Processo para preparação de 5-fluoro-1h-pirazóis
WO2015078846A1 (en) 2013-11-27 2015-06-04 Bayer Cropscience Ag Process for the preparation of 5-fluoro-1h-pyrazoles
TWI694066B (zh) 2014-05-27 2020-05-21 德商拜耳動物保健有限公司 始於六氟丙烯之製備５-氟-１ｈ-吡唑的方法
AU2015306261B2 (en) 2014-08-19 2020-03-05 Bayer Animal Health Gmbh Process for the preparation of 5-fluoro-1H-pyrazoles starting from hexafluoropropene
WO2018177993A1 (de) * 2017-03-31 2018-10-04 Bayer Cropscience Aktiengesellschaft Pyrazole zur bekämpfung von arthropoden

Also Published As

Publication number Publication date
US20230203013A1 (en) 2023-06-29
CN115605468A (zh) 2023-01-13
KR20230016672A (ko) 2023-02-02
CA3178621A1 (en) 2021-12-02
EP4157830A1 (en) 2023-04-05
JP2023528015A (ja) 2023-07-03
AU2021279260A1 (en) 2022-12-15
WO2021239835A1 (en) 2021-12-02
BR112022023008A2 (pt) 2022-12-20

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