MX2021015850A - Agonista beta adrenergico y metodos de uso del mismo. - Google Patents

Agonista beta adrenergico y metodos de uso del mismo.

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Publication number
MX2021015850A
MX2021015850A MX2021015850A MX2021015850A MX2021015850A MX 2021015850 A MX2021015850 A MX 2021015850A MX 2021015850 A MX2021015850 A MX 2021015850A MX 2021015850 A MX2021015850 A MX 2021015850A MX 2021015850 A MX2021015850 A MX 2021015850A
Authority
MX
Mexico
Prior art keywords
methods
same
adrenergic agonist
beta adrenergic
compounds
Prior art date
Application number
MX2021015850A
Other languages
English (en)
Inventor
Wei Chen
Anthony P Ford
David Scott Carter
Jiaxin Yu
Original Assignee
Curasen Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US16/831,285 external-priority patent/US11040944B2/en
Application filed by Curasen Therapeutics Inc filed Critical Curasen Therapeutics Inc
Publication of MX2021015850A publication Critical patent/MX2021015850A/es

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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A61K31/366—Lactones having six-membered rings, e.g. delta-lactones
    • A61K31/37—Coumarins, e.g. psoralen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4704—2-Quinolinones, e.g. carbostyril
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Abstract

La presente revelación está dirigida a compuestos químicos y al uso de dichos compuestos en el tratamiento de enfermedades asociadas con un receptor adrenérgico.
MX2021015850A 2019-07-01 2020-06-30 Agonista beta adrenergico y metodos de uso del mismo. MX2021015850A (es)

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US16/831,285 US11040944B2 (en) 2019-03-27 2020-03-26 Beta adrenergic agonist and methods of using the same
US16/831,370 US10947196B2 (en) 2019-03-27 2020-03-26 Beta adrenergic agonist and methods of using the same
US202063018431P 2020-04-30 2020-04-30
PCT/US2020/040308 WO2021003161A1 (en) 2019-07-01 2020-06-30 Beta adrenergic agonist and methods of using the same

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GB202113594D0 (en) 2021-09-23 2021-11-10 Atrogi Ab New compounds and methods
CA3230482A1 (en) * 2021-09-23 2023-03-30 Jiaxin Yu Beta adrenergic agonist and methods of using the same
GB202113588D0 (en) 2021-09-23 2021-11-10 Atrogi Ab New compounds and methods
CN115677577A (zh) * 2021-11-03 2023-02-03 中国药科大学 靶向srsf6蛋白的小分子化合物及其制备方法和用途
GB202204085D0 (en) 2022-03-23 2022-05-04 Atrogi Ab New compounds and methods
GB202205895D0 (en) 2022-04-22 2022-06-08 Atrogi Ab New medical uses
CN115521254B (zh) * 2022-09-27 2024-05-31 中国药科大学 一种茚达特罗衍生物及其制备方法和应用

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