EP3993878A4 - Beta adrenergic agonist and methods of using the same - Google Patents

Beta adrenergic agonist and methods of using the same Download PDF

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Publication number
EP3993878A4
EP3993878A4 EP20835619.6A EP20835619A EP3993878A4 EP 3993878 A4 EP3993878 A4 EP 3993878A4 EP 20835619 A EP20835619 A EP 20835619A EP 3993878 A4 EP3993878 A4 EP 3993878A4
Authority
EP
European Patent Office
Prior art keywords
methods
same
adrenergic agonist
beta adrenergic
beta
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
EP20835619.6A
Other languages
German (de)
French (fr)
Other versions
EP3993878A1 (en
Inventor
Anthony P. FORD
Jiaxin Yu
David Scott Carter
Wei Chen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Curasen Therapeutics Inc
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Curasen Therapeutics Inc
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Filing date
Publication date
Priority claimed from US16/831,285 external-priority patent/US11040944B2/en
Application filed by Curasen Therapeutics Inc filed Critical Curasen Therapeutics Inc
Publication of EP3993878A1 publication Critical patent/EP3993878A1/en
Publication of EP3993878A4 publication Critical patent/EP3993878A4/en
Pending legal-status Critical Current

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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
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    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
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    • C07D277/62—Benzothiazoles
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    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/06—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 2
    • C07D311/08—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 2 not hydrogenated in the hetero ring
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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US16/831,285 US11040944B2 (en) 2019-03-27 2020-03-26 Beta adrenergic agonist and methods of using the same
US16/831,370 US10947196B2 (en) 2019-03-27 2020-03-26 Beta adrenergic agonist and methods of using the same
US202063018431P 2020-04-30 2020-04-30
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CN115710158A (en) * 2021-08-23 2023-02-24 凯特立斯（深圳）科技有限公司 Method for preparing ticagrelor intermediate through asymmetric catalysis
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AU2022350660A1 (en) * 2021-09-23 2024-04-11 Curasen Therapeutics, Inc. Beta adrenergic agonist and methods of using the same
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CN115677577A (en) * 2021-11-03 2023-02-03 中国药科大学 Small molecular compound targeting SRSF6 protein, and preparation method and application thereof
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CN115521254A (en) * 2022-09-27 2022-12-27 中国药科大学 Indanterol derivative and preparation method and application thereof

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