MX2017005042A - Formas de dosificacion oral de magnesio de liberacion controlada, de alta carga y metodos para elaborar y utilizar las mismas. - Google Patents

Formas de dosificacion oral de magnesio de liberacion controlada, de alta carga y metodos para elaborar y utilizar las mismas.

Info

Publication number
MX2017005042A
MX2017005042A MX2017005042A MX2017005042A MX2017005042A MX 2017005042 A MX2017005042 A MX 2017005042A MX 2017005042 A MX2017005042 A MX 2017005042A MX 2017005042 A MX2017005042 A MX 2017005042A MX 2017005042 A MX2017005042 A MX 2017005042A
Authority
MX
Mexico
Prior art keywords
methods
dosage forms
magnesium
controlled
oral dosage
Prior art date
Application number
MX2017005042A
Other languages
English (en)
Inventor
F Brandon Stephen
A Okerholm Richard
J Legg Thomas
Original Assignee
Pharmalyte Solutions Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=58578872&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2017005042(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US15/132,461 external-priority patent/US9707253B2/en
Application filed by Pharmalyte Solutions Llc filed Critical Pharmalyte Solutions Llc
Publication of MX2017005042A publication Critical patent/MX2017005042A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00Medicinal preparations containing inorganic active ingredients
    • A61K33/06Aluminium, calcium or magnesium; Compounds thereof, e.g. clay
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Inorganic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Physiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se describen formas de dosificación de alta carga, de liberación controlada para administración oral de sales de magnesio. Por ejemplo, una forma de dosificación oral puede comprender desde aproximadamente 80% hasta aproximadamente 95% de lactato de magnesio y uno o más componentes. Como otro ejemplo, una forma de dosificación oral puede comprender por lo menos aproximadamente 50% de sal de magnesio y exhibe un perfil de disolución de liberación controlada. También se describen métodos para elaborar formas de dosificación de liberación controlada para administración oral de una cantidad terapéuticamente efectiva de sal de magnesio a un mamífero. También se describen métodos para tratar un trastorno caracterizado por deficiencia de magnesio y métodos para prevenir o aliviar bajos niveles de magnesio.
MX2017005042A 2016-04-19 2017-04-18 Formas de dosificacion oral de magnesio de liberacion controlada, de alta carga y metodos para elaborar y utilizar las mismas. MX2017005042A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US15/132,461 US9707253B2 (en) 2008-05-19 2016-04-19 High-loading, controlled-release magnesium oral dosage forms and methods for making and using same

Publications (1)

Publication Number Publication Date
MX2017005042A true MX2017005042A (es) 2018-08-20

Family

ID=58578872

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2017005042A MX2017005042A (es) 2016-04-19 2017-04-18 Formas de dosificacion oral de magnesio de liberacion controlada, de alta carga y metodos para elaborar y utilizar las mismas.

Country Status (12)

Country Link
EP (1) EP3243507A1 (es)
JP (1) JP2017214352A (es)
KR (1) KR20170119651A (es)
AR (1) AR108235A1 (es)
AU (1) AU2017202534B1 (es)
CA (1) CA2964581C (es)
CL (1) CL2017000957A1 (es)
MX (1) MX2017005042A (es)
MY (1) MY185460A (es)
RU (1) RU2017113518A (es)
SG (1) SG10201703206TA (es)
ZA (1) ZA201702773B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4212149A1 (en) * 2022-01-18 2023-07-19 Rijksuniversiteit Groningen Oral dosage forms of acid-labile salt and methods and uses related thereto

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5002774A (en) * 1989-06-08 1991-03-26 Erbamont, Inc. Sustained release pharmaceutical tablet
CN102098921A (zh) * 2008-05-19 2011-06-15 温顿制药有限公司 高载量、控释镁口服制剂及其制备和使用方法

Also Published As

Publication number Publication date
SG10201703206TA (en) 2017-11-29
AU2017202534B1 (en) 2017-06-08
JP2017214352A (ja) 2017-12-07
KR20170119651A (ko) 2017-10-27
AR108235A1 (es) 2018-08-01
ZA201702773B (en) 2018-11-28
RU2017113518A (ru) 2018-10-19
CA2964581A1 (en) 2017-10-19
MY185460A (en) 2021-05-19
EP3243507A1 (en) 2017-11-15
CL2017000957A1 (es) 2017-12-15
CA2964581C (en) 2020-06-16

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