MX2014002105A - Ligandos de receptor de estrogeno y metodos de uso de los mismos. - Google Patents
Ligandos de receptor de estrogeno y metodos de uso de los mismos.Info
- Publication number
- MX2014002105A MX2014002105A MX2014002105A MX2014002105A MX2014002105A MX 2014002105 A MX2014002105 A MX 2014002105A MX 2014002105 A MX2014002105 A MX 2014002105A MX 2014002105 A MX2014002105 A MX 2014002105A MX 2014002105 A MX2014002105 A MX 2014002105A
- Authority
- MX
- Mexico
- Prior art keywords
- compound
- another embodiment
- prostate cancer
- levels
- castration
- Prior art date
Links
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- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4453—Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
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- A—HUMAN NECESSITIES
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- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
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US13/215,679 US9427418B2 (en) | 2009-02-23 | 2011-08-23 | Estrogen receptor ligands and methods of use thereof |
PCT/US2012/052141 WO2013043304A1 (en) | 2009-02-23 | 2012-08-23 | Estrogen receptor ligands and methods of use thereof |
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AU2018342909B2 (en) * | 2017-09-27 | 2023-06-08 | Targimmune Therapeutics Ag | Castration resistant prostate cancer |
CA3128331C (en) * | 2019-01-30 | 2024-06-18 | Margaret K. YU | Anti-androgens for the treatment of metastatic castration-sensitive prostate cancer |
WO2020157334A1 (en) * | 2019-02-01 | 2020-08-06 | Fondazione Per L'istituto Oncologico Di Ricerca (Ior) | Methods of treating castrate-resistant prostate cancer |
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US8158828B2 (en) * | 2005-11-28 | 2012-04-17 | Gtx, Inc. | Nuclear receptor binding agents |
US8546451B2 (en) * | 2005-11-28 | 2013-10-01 | Gtx, Inc. | Estrogen receptor ligands and methods of use thereof |
EP2455362A1 (en) * | 2005-11-28 | 2012-05-23 | GTX, Inc. | Nuclear receptor binding agents |
KR20130101146A (ko) * | 2009-02-23 | 2013-09-12 | 지티엑스, 인코포레이티드 | 에스트로겐 수용체 리간드 및 그 이용 방법 |
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2012
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- 2012-08-23 MX MX2014002105A patent/MX2014002105A/es unknown
- 2012-08-23 AU AU2012312902A patent/AU2012312902B2/en not_active Ceased
- 2012-08-23 CA CA2845890A patent/CA2845890A1/en not_active Abandoned
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AU2012312902A1 (en) | 2013-05-23 |
KR20140064906A (ko) | 2014-05-28 |
IN2014DN01959A (enrdf_load_stackoverflow) | 2015-05-15 |
CN103957706A (zh) | 2014-07-30 |
JP2014524479A (ja) | 2014-09-22 |
EP2747562A1 (en) | 2014-07-02 |
AU2012312902B2 (en) | 2016-03-17 |
EP2747562A4 (en) | 2015-05-06 |
RU2014111060A (ru) | 2015-09-27 |
CA2845890A1 (en) | 2013-03-28 |
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