IL231070A0 - Estrogen receptor ligands and methods of their use - Google Patents

Estrogen receptor ligands and methods of their use

Info

Publication number
IL231070A0
IL231070A0 IL231070A IL23107014A IL231070A0 IL 231070 A0 IL231070 A0 IL 231070A0 IL 231070 A IL231070 A IL 231070A IL 23107014 A IL23107014 A IL 23107014A IL 231070 A0 IL231070 A0 IL 231070A0
Authority
IL
Israel
Prior art keywords
methods
estrogen receptor
estrogen
receptor
Prior art date
Application number
IL231070A
Other languages
English (en)
Hebrew (he)
Original Assignee
Gtx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US13/215,679 external-priority patent/US9427418B2/en
Priority claimed from PCT/US2012/052141 external-priority patent/WO2013043304A1/en
Application filed by Gtx Inc filed Critical Gtx Inc
Publication of IL231070A0 publication Critical patent/IL231070A0/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4453Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
IL231070A 2011-08-23 2014-02-20 Estrogen receptor ligands and methods of their use IL231070A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13/215,679 US9427418B2 (en) 2009-02-23 2011-08-23 Estrogen receptor ligands and methods of use thereof
PCT/US2012/052141 WO2013043304A1 (en) 2009-02-23 2012-08-23 Estrogen receptor ligands and methods of use thereof

Publications (1)

Publication Number Publication Date
IL231070A0 true IL231070A0 (en) 2014-03-31

Family

ID=48444651

Family Applications (1)

Application Number Title Priority Date Filing Date
IL231070A IL231070A0 (en) 2011-08-23 2014-02-20 Estrogen receptor ligands and methods of their use

Country Status (10)

Country Link
EP (1) EP2747562A4 (enrdf_load_stackoverflow)
JP (1) JP2014524479A (enrdf_load_stackoverflow)
KR (1) KR20140064906A (enrdf_load_stackoverflow)
CN (1) CN103957706A (enrdf_load_stackoverflow)
AU (1) AU2012312902B2 (enrdf_load_stackoverflow)
CA (1) CA2845890A1 (enrdf_load_stackoverflow)
IL (1) IL231070A0 (enrdf_load_stackoverflow)
IN (1) IN2014DN01959A (enrdf_load_stackoverflow)
MX (1) MX2014002105A (enrdf_load_stackoverflow)
RU (1) RU2014111060A (enrdf_load_stackoverflow)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2018342909B2 (en) * 2017-09-27 2023-06-08 Targimmune Therapeutics Ag Castration resistant prostate cancer
CA3128331C (en) * 2019-01-30 2024-06-18 Margaret K. YU Anti-androgens for the treatment of metastatic castration-sensitive prostate cancer
WO2020157334A1 (en) * 2019-02-01 2020-08-06 Fondazione Per L'istituto Oncologico Di Ricerca (Ior) Methods of treating castrate-resistant prostate cancer

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8158828B2 (en) * 2005-11-28 2012-04-17 Gtx, Inc. Nuclear receptor binding agents
US8546451B2 (en) * 2005-11-28 2013-10-01 Gtx, Inc. Estrogen receptor ligands and methods of use thereof
EP2455362A1 (en) * 2005-11-28 2012-05-23 GTX, Inc. Nuclear receptor binding agents
KR20130101146A (ko) * 2009-02-23 2013-09-12 지티엑스, 인코포레이티드 에스트로겐 수용체 리간드 및 그 이용 방법

Also Published As

Publication number Publication date
AU2012312902A1 (en) 2013-05-23
KR20140064906A (ko) 2014-05-28
IN2014DN01959A (enrdf_load_stackoverflow) 2015-05-15
CN103957706A (zh) 2014-07-30
JP2014524479A (ja) 2014-09-22
MX2014002105A (es) 2014-09-25
EP2747562A1 (en) 2014-07-02
AU2012312902B2 (en) 2016-03-17
EP2747562A4 (en) 2015-05-06
RU2014111060A (ru) 2015-09-27
CA2845890A1 (en) 2013-03-28

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