AU2012312902B2 - Estrogen receptor ligands and methods of use thereof - Google Patents
Estrogen receptor ligands and methods of use thereof Download PDFInfo
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- AU2012312902B2 AU2012312902B2 AU2012312902A AU2012312902A AU2012312902B2 AU 2012312902 B2 AU2012312902 B2 AU 2012312902B2 AU 2012312902 A AU2012312902 A AU 2012312902A AU 2012312902 A AU2012312902 A AU 2012312902A AU 2012312902 B2 AU2012312902 B2 AU 2012312902B2
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4453—Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Emergency Medicine (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13/215,679 | 2011-08-23 | ||
| US13/215,679 US9427418B2 (en) | 2009-02-23 | 2011-08-23 | Estrogen receptor ligands and methods of use thereof |
| PCT/US2012/052141 WO2013043304A1 (en) | 2009-02-23 | 2012-08-23 | Estrogen receptor ligands and methods of use thereof |
Publications (2)
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| AU2012312902B2 true AU2012312902B2 (en) | 2016-03-17 |
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| AU2018342909B2 (en) * | 2017-09-27 | 2023-06-08 | Targimmune Therapeutics Ag | Castration resistant prostate cancer |
| CA3128331C (en) * | 2019-01-30 | 2024-06-18 | Margaret K. YU | Anti-androgens for the treatment of metastatic castration-sensitive prostate cancer |
| WO2020157334A1 (en) * | 2019-02-01 | 2020-08-06 | Fondazione Per L'istituto Oncologico Di Ricerca (Ior) | Methods of treating castrate-resistant prostate cancer |
Citations (2)
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|---|---|---|---|---|
| US20070265296A1 (en) * | 2005-11-28 | 2007-11-15 | Dalton James T | Nuclear receptor binding agents |
| US20100267773A1 (en) * | 2005-11-28 | 2010-10-21 | Dalton James T | Estrogen receptor ligands and methods of use thereof |
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| EP2455362A1 (en) * | 2005-11-28 | 2012-05-23 | GTX, Inc. | Nuclear receptor binding agents |
| KR20130101146A (ko) * | 2009-02-23 | 2013-09-12 | 지티엑스, 인코포레이티드 | 에스트로겐 수용체 리간드 및 그 이용 방법 |
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2012
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- 2012-08-23 MX MX2014002105A patent/MX2014002105A/es unknown
- 2012-08-23 AU AU2012312902A patent/AU2012312902B2/en not_active Ceased
- 2012-08-23 CA CA2845890A patent/CA2845890A1/en not_active Abandoned
- 2012-08-23 RU RU2014111060/15A patent/RU2014111060A/ru not_active Application Discontinuation
- 2012-08-23 JP JP2014527312A patent/JP2014524479A/ja active Pending
- 2012-08-23 EP EP12834287.0A patent/EP2747562A4/en not_active Withdrawn
- 2012-08-23 CN CN201280051979.4A patent/CN103957706A/zh active Pending
- 2012-08-23 IN IN1959DEN2014 patent/IN2014DN01959A/en unknown
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2014
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Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20070265296A1 (en) * | 2005-11-28 | 2007-11-15 | Dalton James T | Nuclear receptor binding agents |
| US20100267773A1 (en) * | 2005-11-28 | 2010-10-21 | Dalton James T | Estrogen receptor ligands and methods of use thereof |
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| IL231070A0 (en) | 2014-03-31 |
| AU2012312902A1 (en) | 2013-05-23 |
| KR20140064906A (ko) | 2014-05-28 |
| IN2014DN01959A (enrdf_load_stackoverflow) | 2015-05-15 |
| CN103957706A (zh) | 2014-07-30 |
| JP2014524479A (ja) | 2014-09-22 |
| MX2014002105A (es) | 2014-09-25 |
| EP2747562A1 (en) | 2014-07-02 |
| EP2747562A4 (en) | 2015-05-06 |
| RU2014111060A (ru) | 2015-09-27 |
| CA2845890A1 (en) | 2013-03-28 |
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