MX2009011843A - Dosificacion intravenosa y oral de un inhibidor de p2y12 de accion directa y reversible. - Google Patents

Dosificacion intravenosa y oral de un inhibidor de p2y12 de accion directa y reversible.

Info

Publication number
MX2009011843A
MX2009011843A MX2009011843A MX2009011843A MX2009011843A MX 2009011843 A MX2009011843 A MX 2009011843A MX 2009011843 A MX2009011843 A MX 2009011843A MX 2009011843 A MX2009011843 A MX 2009011843A MX 2009011843 A MX2009011843 A MX 2009011843A
Authority
MX
Mexico
Prior art keywords
reversible
intravenous
inhibitor
acting
direct
Prior art date
Application number
MX2009011843A
Other languages
English (en)
Spanish (es)
Inventor
Anjali Pandey
Pamela B Conley
Patrick Andre
Daniel D Gretler
Athiwat Hutchaleelaha
David R Phillips
Huang Wolin
Robert M Scarborough
Original Assignee
Portola Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Portola Pharm Inc filed Critical Portola Pharm Inc
Publication of MX2009011843A publication Critical patent/MX2009011843A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Emergency Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MX2009011843A 2007-05-02 2008-05-02 Dosificacion intravenosa y oral de un inhibidor de p2y12 de accion directa y reversible. MX2009011843A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US91564907P 2007-05-02 2007-05-02
US94792107P 2007-07-03 2007-07-03
PCT/US2008/062518 WO2008137753A2 (en) 2007-05-02 2008-05-02 Intravenous and oral dosing of a direct-acting and reversible p2y12 inhibitor

Publications (1)

Publication Number Publication Date
MX2009011843A true MX2009011843A (es) 2010-04-22

Family

ID=39587015

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009011843A MX2009011843A (es) 2007-05-02 2008-05-02 Dosificacion intravenosa y oral de un inhibidor de p2y12 de accion directa y reversible.

Country Status (17)

Country Link
US (2) US20090048216A1 (https=)
EP (1) EP2079464A2 (https=)
JP (1) JP2010526101A (https=)
KR (1) KR20100029746A (https=)
CN (1) CN101795682A (https=)
AU (1) AU2008247483A1 (https=)
BR (1) BRPI0811476A2 (https=)
CA (1) CA2686203A1 (https=)
CO (1) CO6241104A2 (https=)
EA (1) EA200901473A1 (https=)
EC (1) ECSP099778A (https=)
GT (1) GT200900284A (https=)
IL (1) IL201834A0 (https=)
MA (1) MA31663B1 (https=)
MX (1) MX2009011843A (https=)
TN (1) TN2009000451A1 (https=)
WO (1) WO2008137753A2 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1951254E (pt) * 2005-11-03 2012-04-12 Portola Pharm Inc [4-(6-halo-7-substituído-2,4-dioxo-1,4-di-hidro-2hquinazolin- 3-il)-fenil]-5-cloro-tiofen-2-il-sulfonilureias e formas e métodos relacionados com as mesmas
CA2678492A1 (en) * 2007-03-06 2008-09-12 Novartis Ag Bicyclic organic compounds suitable for the treatment of inflammatory or allergic conditions
US20090156620A1 (en) * 2007-05-02 2009-06-18 Portola Pharmaceuticals, Inc. [4-(6-fluoro-7-methylamino-2,4-dioxo-1,4-dihydro-2h-quinazolin-3-yl)-phenyl]-5-chloro-thiophen-2-yl-sulfonylurea salts, forms and methods related thereto
WO2008137809A2 (en) * 2007-05-02 2008-11-13 Portola Pharmaceuticals, Inc. [4-(6-fluoro-7-methylamino-2,4-dioxo-1,4-dihydro-2h-quinazolin-3-yl)-phenyl] -5-chloro-thiophen-2-yl-sulfonylurea salts, in different crystalline forms, pharmaceutical compositions thereof
US9427448B2 (en) * 2009-11-11 2016-08-30 The Medicines Company Methods of treating, reducing the incidence of, and/or preventing ischemic events
MX2011006995A (es) * 2008-12-30 2011-09-27 Thrombologic Aps Metodos para identificar pacientes criticamente enfermos en riesgo incrementado de desarrollar nsuficiencia organica y compuestos para el tratamiento de la misma.
BR112012011298B1 (pt) 2009-11-11 2021-12-14 Chiesi Farmaceutici S.P.A. Uso de cangrelor e/ou bivalirudina na preparação de medicamentos e combinação de medicamentos
US10376532B2 (en) 2009-11-11 2019-08-13 Chiesi Farmaceutici, S.P.A. Methods of treating, reducing the incidence of, and/or preventing ischemic events
EP2633857B1 (en) * 2009-12-23 2015-08-12 ratiopharm GmbH Solid pharmaceutical dosage form of ticagrelor and acetylsalicylic acid
US20130165459A1 (en) 2010-01-12 2013-06-27 Norvartis Pharma Ag Pharmaceutical composition and dosage forms of elinogrel and methods of use thereof
WO2011137459A1 (en) * 2010-04-30 2011-11-03 Portola Pharmaceuticals, Inc. Dosage forms of elinogrel and methods of injectable administration thereof
EP2646827A1 (en) 2010-12-01 2013-10-09 INSERM (Institut National de la Santé et de la Recherche Médicale) Method and kits for determining platelet susceptibility to activation in a patient
JP2013544271A (ja) * 2010-12-03 2013-12-12 ポートラ ファーマシューティカルズ, インコーポレイテッド 式(i)の化合物の薬学的組成物、投薬形態、および新規の形態、ならびにその使用方法
MA49887A (fr) 2017-03-15 2020-06-24 Idorsia Pharmaceuticals Ltd Administration sous-cutanée d'un antagoniste du récepteur p2y12
MA49452A (fr) 2017-06-23 2021-05-05 Chiesi Farm Spa Procédé de prévention de thrombose de shunt de l'artère systémique-pulmonaire
CN107462648B (zh) * 2017-08-21 2019-09-27 盐城锦明药业有限公司 一种Cangrelor中间体腺苷-2-硫酮的高效液相色谱检测方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6906063B2 (en) 2000-02-04 2005-06-14 Portola Pharmaceuticals, Inc. Platelet ADP receptor inhibitors
PT1951254E (pt) 2005-11-03 2012-04-12 Portola Pharm Inc [4-(6-halo-7-substituído-2,4-dioxo-1,4-di-hidro-2hquinazolin- 3-il)-fenil]-5-cloro-tiofen-2-il-sulfonilureias e formas e métodos relacionados com as mesmas

Also Published As

Publication number Publication date
JP2010526101A (ja) 2010-07-29
KR20100029746A (ko) 2010-03-17
US20090048216A1 (en) 2009-02-19
CO6241104A2 (es) 2011-01-20
GT200900284A (es) 2012-01-31
WO2008137753A3 (en) 2009-02-12
CN101795682A (zh) 2010-08-04
EP2079464A2 (en) 2009-07-22
EA200901473A1 (ru) 2010-06-30
US20120009172A1 (en) 2012-01-12
TN2009000451A1 (en) 2011-03-31
BRPI0811476A2 (pt) 2014-11-04
AU2008247483A1 (en) 2008-11-13
MA31663B1 (fr) 2010-09-01
WO2008137753A2 (en) 2008-11-13
IL201834A0 (en) 2010-06-16
CA2686203A1 (en) 2008-11-13
ECSP099778A (es) 2010-01-29

Similar Documents

Publication Publication Date Title
MX2009011843A (es) Dosificacion intravenosa y oral de un inhibidor de p2y12 de accion directa y reversible.
ECSP099376A (es) Inhibidores de la actividad de la akt
HN2009003002A (es) Compuestos de piridopirimidinonas inhibidores de pi3k-alfa
PL1986669T3 (pl) Zastosowanie Bifidobacterium longum do zapobiegania i leczenia zapalenia
MX2015012432A (es) Inhibidores piridinicos de la cinasa cdk9.
IL211825A (en) Compounds based on pyridine and pyrimidine for use as wnt signal transducer inhibitors, pharmaceutical formulations containing such compounds and used as drugs for the treatment and / or cancer prevention
HRP20110451T1 (hr) Upotreba izotiocijanata kao sredstva protiv mieloma
MA33803B1 (fr) Inhibiteur de bromodomaine de benzodiazépine
MX2009004017A (es) Usos de los compuestos carboxi-amido triazol y sus sales.
MX341212B (es) Inhibidor de bromodominio de benzodiazepina.
MX2009011578A (es) 6-fenilpirimidinonas como moduladores de pim.
ECSP077980A (es) Inhibidores de la actividad akt
CL2013001136A1 (es) Un agente inhibitorio de la fosfodiesterasa 7 (pde7) para ser usado en el tratamiento o la reduccion de la posibilidad de una adiccion; y composicion farmaceutica, forma de dosificacion unitaria y kit farmaceutico que incluyen al inhibidor de fosfodiesterasa 7 (pde7) y un agente terapeutico adicional.
MX2009014235A (es) 4-bencilaminoquinolonas, composiciones farmaceuticas que las contiene y su uso.
PH12013500467A1 (en) Pharmaceutical composition
PH12014500386A1 (en) Combination treatment for hepatitis c
MX2009000657A (es) Composiciones y metodos para el tratamiento de mucositis.
MY177741A (en) Pharmaceutical compositions compring 4-amino-5-fluoro-3-[6-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-quinolin-2-one-lactate monohydrate.
UA109290C2 (uk) Спільні кристали і солі інгібіторів ccr3
MY140514A (en) Triazolopyridine derivatives as inhibitors of lipases and phospholipases
UA93709C2 (ru) 12-имидазолил-1-додеканол и его применение b изготовлении фармацевтических композиций
IN2012DN03428A (https=)
PH12013500695A1 (en) Pharmaceutical compositions containing a dgat1 inhibitor
MX2010005714A (es) Compuestos de piridina.
SG158091A1 (en) Imidazoazepinone compounds

Legal Events

Date Code Title Description
FA Abandonment or withdrawal