MX173858B - Procedimiento para la preparacion de derivados del acido amino-pimelico y compuestos obtenidos - Google Patents
Procedimiento para la preparacion de derivados del acido amino-pimelico y compuestos obtenidosInfo
- Publication number
- MX173858B MX173858B MX013643A MX1364388A MX173858B MX 173858 B MX173858 B MX 173858B MX 013643 A MX013643 A MX 013643A MX 1364388 A MX1364388 A MX 1364388A MX 173858 B MX173858 B MX 173858B
- Authority
- MX
- Mexico
- Prior art keywords
- denotes
- hydrogen atom
- radical
- amino
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/08—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Oncology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biophysics (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Communicable Diseases (AREA)
- Analytical Chemistry (AREA)
- Biochemistry (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Virology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Indole Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Saccharide Compounds (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
Abstract
La presente invención se refiere a procedimiento para preparar compuestos de fórmula (I): caracterizado porque se somete un compuesto de fórmula (II): a la acción de un halogenuro de alcanosulfonilo o arenosulfonilo de fórmula (III) HalSO2alc4 y luego a la acción de un agente de reducción, posteriormetne se somete, si se desea, a la totalidad o a una parte solamente de las operaciones siguientes en cualquier orden: a) desprotección de la función amino; b) hidrólisis de las funciones esteres y luego, llegado el caso, descarboxilación cuando X represente un radical -XO2alc3; c) reducción del doble enlace; d) esterificación o salificación por una base de las funciones carboxi; e) salificación de las funciones amina con un ácido; f) amidación de las funciones aminas libres por un aminoácido o un peptido constituído por 2, 3 o 4 aminoácidos o un peptido constituído por 2, 3 o 4 aminoácidos cuya función amina está protegida y luego desprotección de esta función amina.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8715209A FR2622578B1 (fr) | 1987-11-03 | 1987-11-03 | Nouveaux derives de l'acide aminopimelique, leur procede de preparation et leur application comme medicaments |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX13643A MX13643A (es) | 1993-09-01 |
| MX173858B true MX173858B (es) | 1994-04-07 |
Family
ID=9356421
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX013643A MX173858B (es) | 1987-11-03 | 1988-11-01 | Procedimiento para la preparacion de derivados del acido amino-pimelico y compuestos obtenidos |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US5030715A (es) |
| EP (1) | EP0315519B1 (es) |
| JP (1) | JPH01151543A (es) |
| AT (1) | ATE87299T1 (es) |
| AU (1) | AU615229B2 (es) |
| CA (1) | CA1310445C (es) |
| DE (1) | DE3879622T2 (es) |
| DK (1) | DK607688A (es) |
| ES (1) | ES2053787T3 (es) |
| FR (1) | FR2622578B1 (es) |
| GR (1) | GR3007597T3 (es) |
| HU (1) | HU202471B (es) |
| MX (1) | MX173858B (es) |
| PT (1) | PT88926B (es) |
| ZA (1) | ZA888200B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6077915A (en) * | 1990-07-23 | 2000-06-20 | Exxon Research & Engineering | Carbonyl containing compounds |
| DK1257541T3 (da) * | 2000-01-11 | 2009-01-19 | Molecular Insight Pharm Inc | Farmakoforiske stoffer |
| CN113072456B (zh) * | 2021-04-12 | 2022-04-19 | 中国科学技术大学 | 一种手性α-二氟甲基氨基酸类化合物及其制备方法 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2566410A1 (fr) * | 1984-06-20 | 1985-12-27 | Delalande Sa | Nouveaux derives de l'acide diaminopimelique, leur procede de preparation et leur application en therapeutique |
-
1987
- 1987-11-03 FR FR8715209A patent/FR2622578B1/fr not_active Expired - Fee Related
-
1988
- 1988-11-01 DK DK607688A patent/DK607688A/da not_active Application Discontinuation
- 1988-11-01 MX MX013643A patent/MX173858B/es unknown
- 1988-11-02 EP EP88402741A patent/EP0315519B1/fr not_active Expired - Lifetime
- 1988-11-02 HU HU885678A patent/HU202471B/hu not_active IP Right Cessation
- 1988-11-02 AT AT88402741T patent/ATE87299T1/de not_active IP Right Cessation
- 1988-11-02 CA CA000581930A patent/CA1310445C/fr not_active Expired - Lifetime
- 1988-11-02 AU AU24582/88A patent/AU615229B2/en not_active Ceased
- 1988-11-02 ZA ZA888200A patent/ZA888200B/xx unknown
- 1988-11-02 JP JP63276337A patent/JPH01151543A/ja active Pending
- 1988-11-02 DE DE88402741T patent/DE3879622T2/de not_active Expired - Fee Related
- 1988-11-02 ES ES88402741T patent/ES2053787T3/es not_active Expired - Lifetime
- 1988-11-03 US US07/267,190 patent/US5030715A/en not_active Expired - Fee Related
- 1988-11-03 PT PT88926A patent/PT88926B/pt not_active IP Right Cessation
-
1993
- 1993-04-09 GR GR920402861T patent/GR3007597T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ATE87299T1 (de) | 1993-04-15 |
| FR2622578B1 (fr) | 1990-03-16 |
| MX13643A (es) | 1993-09-01 |
| EP0315519B1 (fr) | 1993-03-24 |
| JPH01151543A (ja) | 1989-06-14 |
| DK607688A (da) | 1989-06-20 |
| EP0315519A3 (en) | 1990-02-28 |
| DK607688D0 (da) | 1988-11-01 |
| GR3007597T3 (es) | 1993-08-31 |
| AU2458288A (en) | 1989-05-25 |
| FR2622578A1 (fr) | 1989-05-05 |
| US5030715A (en) | 1991-07-09 |
| DE3879622T2 (de) | 1993-09-30 |
| PT88926A (pt) | 1988-12-01 |
| PT88926B (pt) | 1993-01-29 |
| HUT48568A (en) | 1989-06-28 |
| EP0315519A2 (fr) | 1989-05-10 |
| ES2053787T3 (es) | 1994-08-01 |
| ZA888200B (en) | 1990-01-31 |
| AU615229B2 (en) | 1991-09-26 |
| CA1310445C (fr) | 1992-11-17 |
| HU202471B (en) | 1991-03-28 |
| DE3879622D1 (de) | 1993-04-29 |
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