ME02064B - Derivati kvinazolin-4(3h)-ona korisceni kao inhibitori pi3 kinaze - Google Patents
Derivati kvinazolin-4(3h)-ona korisceni kao inhibitori pi3 kinazeInfo
- Publication number
- ME02064B ME02064B MEP-2015-43A MEP4315A ME02064B ME 02064 B ME02064 B ME 02064B ME P4315 A MEP4315 A ME P4315A ME 02064 B ME02064 B ME 02064B
- Authority
- ME
- Montenegro
- Prior art keywords
- compound
- formula
- combination
- use according
- treatment
- Prior art date
Links
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- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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| TW099135360A TWI478923B (zh) | 2009-10-19 | 2010-10-18 | 喹唑啉酮化合物及其用途 |
| PCT/EP2010/065746 WO2011048111A1 (en) | 2009-10-19 | 2010-10-19 | Compounds |
| PCT/GB2011/052015 WO2012052753A1 (en) | 2010-10-18 | 2011-10-18 | Quinazolin-4 (3h) -one derivatives used as pi3 kinase inhibitors |
| EP11787742.3A EP2630149B1 (en) | 2010-10-18 | 2011-10-18 | Quinazolin-4(3h)-one derivatives used as pi3 kinase inhibitors |
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| EA029473B1 (ru) | 2011-12-15 | 2018-03-30 | Новартис Аг | Применение ингибиторов pi3k для лечения острой и церебральной малярии |
| TWI617561B (zh) | 2012-03-13 | 2018-03-11 | 瑞斯比維特有限公司 | 呈晶體型式之新穎化合物，包含其之醫藥組成物，製備該化合物之方法及包括該組成物之吸入裝置 |
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| CN104870017B (zh) | 2012-11-08 | 2020-08-14 | 理森制药股份公司 | 含有PDE4抑制剂和PI3δ或双重PI3δ-γ激酶抑制剂的药物组合物 |
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| WO2022017371A1 (zh) * | 2020-07-21 | 2022-01-27 | 中国医药研究开发中心有限公司 | 具有磷脂酰肌醇3-激酶δ和γ的双重抑制剂活性的杂环化合物及其医药用途 |
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| TWI617561B (zh) | 2012-03-13 | 2018-03-11 | 瑞斯比維特有限公司 | 呈晶體型式之新穎化合物，包含其之醫藥組成物，製備該化合物之方法及包括該組成物之吸入裝置 |
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